Bisubstrate Ether‐Linked Uridine‐Peptide Conjugates as O‐GlcNAc Transferase Inhibitors

The O‐linked β‐N‐acetylglucosamine (O‐GlcNAc) transferase (OGT) is a master regulator of installing O‐GlcNAc onto serine or threonine residues on a multitude of target proteins. Numerous nuclear and cytosolic proteins of varying functional classes, including translational factors, transcription fact...

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