Syntheses of SGLT2 Inhibitors by Ni- and Pd-Catalyzed Fukuyama Coupling Reactions

Nickel- and palladium-catalyzed Fukuyama coupling reactions of a d-gluconolactone-derived thioester with arylzinc reagents at ambient temperature provided the corresponding multifunctional aryl ketones in high yield. Ligand screening for the nickel-catalyzed Fukuyama coupling reactions indicated tha...

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Veröffentlicht in:	Journal of organic chemistry 2020-10, Vol.85 (19), p.12382-12392
Hauptverfasser:	Talode, Jalindar, Kato, Daiki, Nagae, Haruki, Tsurugi, Hayato, Seki, Masahiko, Mashima, Kazushi
Format:	Artikel
Sprache:	eng
Online-Zugang:	Volltext
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