Quinolidene-rhodanine conjugates: Facile synthesis and biological evaluation

A series of rhodanine incorporated quinoline derivatives were efficiently synthesized using reusable DBU acetate as ionic liquid and evaluated for their in vitro antitubercular activity against Mycobacterium tuberculosis H37Ra (MTB) (ATCC 25177) and Mycobacterium bovis BCG (ATCC 35743) both in activ...

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Veröffentlicht in:	European journal of medicinal chemistry 2017-01, Vol.125, p.385-399
Hauptverfasser:	Subhedar, Dnyaneshwar D., Shaikh, Mubarak H., Shingate, Bapurao B., Nawale, Laxman, Sarkar, Dhiman, Khedkar, Vijay M., Kalam Khan, Firoz A., Sangshetti, Jaiprakash N.
Format:	Artikel
Sprache:	eng
Schlagworte:	[DBUH][OAc] ionic liquid Animals Antibacterial activity Antifungal Antitubercular Antitubercular Agents - chemical synthesis Antitubercular Agents - chemistry Antitubercular Agents - pharmacology Bacterial Proteins - metabolism Cell Line Cytotoxicity Humans Metalloproteases - metabolism Molecular Docking Simulation Molecular docking study Mycobacterium bovis - drug effects Mycobacterium bovis - metabolism Mycobacterium Infections - drug therapy Mycobacterium Infections - veterinary Mycobacterium tuberculosis - drug effects Mycobacterium tuberculosis - metabolism Quinolines - chemical synthesis Quinolines - chemistry Quinolines - pharmacology Rhodanine - analogs & derivatives Rhodanine - chemical synthesis Rhodanine - chemistry Rhodanine - pharmacology
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