Diastereoselective synthesis of substituted diaziridines from simple ketones and aldehydes

Diastereopure substituted diaziridines from simple ketones, aldehydes and amines are here reported. These important chemical scaffolds are obtained in the presence of a weak inorganic base and hydroxylamine O-sulfonic acid (HOSA). This method introduces three stereocenters in one step to provide a w...

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Veröffentlicht in:	Chemical communications (Cambridge, England) England), 2015-09, Vol.51 (70), p.13511-13514
Hauptverfasser:	Beebe, Alexander W, Dohmeier, Emma F, Moura-Letts, Gustavo
Format:	Artikel
Sprache:	eng
Schlagworte:	Aldehydes Amines Hydroxides Ketones Scaffolds Synthesis
Online-Zugang:	Volltext
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