Selective Iodine-Catalyzed Intermolecular Oxidative Amination of C(sp3)H Bonds with ortho-Carbonyl-Substituted Anilines to Give Quinazolines

Access to quinazolines: The selective amination of C(sp3)H bonds adjacent to nitrogen or oxygen atoms of N‐alkylamides, ethers, or alcohols with ortho‐carbonyl‐substituted anilines constitutes the first step in a tandem annulation that leads to quinazolines in good to excellent yields (see scheme;...

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