Copper-Catalyzed Direct Amination of Quinoline N‑Oxides via C–H Bond Activation under Mild Conditions

A highly efficient and concise one-pot strategy for the direct amination of quinoline N-oxides via copper-catalyzed dehydrogenative C–N coupling has been developed. The desired products were obtained in good to excellent yields for 22 examples starting from the parent aliphatic amines. This methodol...

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Veröffentlicht in:	Organic letters 2014-04, Vol.16 (7), p.1840-1843
Hauptverfasser:	Zhu, Chongwei, Yi, Meiling, Wei, Donghui, Chen, Xuan, Wu, Yangjie, Cui, Xiuling
Format:	Artikel
Sprache:	eng
Schlagworte:	Amination Aminoquinolines - chemical synthesis Aminoquinolines - chemistry Catalysis Copper - chemistry Molecular Structure Oxides - chemistry
Online-Zugang:	Volltext
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