Stereoselective inhibition of the binding of ( super(3)H)PK 11195 to peripheral-type benzodiazepine binding sites by a quinoline-propanamide derivative

The specific binding of ( super(3)H)PK 11195 to the peripheral-type benzodiazepine binding site is inhibited by the 1-enantiomer of N,N-diethyl- alpha -methyl-2-phenyl-4-quinoline-propanamide ((-)Q sub(1)) but not by its d-enantiomer ((+)Q sub(1)). (-)Q sub(1) inhibited ( super(3)H)PK 11195 binding...

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Veröffentlicht in:	European journal of pharmacology 1986-01, Vol.128 (3), p.269-272
Hauptverfasser:	Dubroeucq, M-C, Benavides, J, Doble, A, Guilloux, F, Allam, D, Vaucher, N, Bertrand, P, Gueremy, C, Le Fur, G
Format:	Artikel
Sprache:	eng
Online-Zugang:	Volltext
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