Synthesis of succinic monoamide avermectin esters

Synthesis of succinic monoamide avermectin esters

Reaction of avermectin B 1 hemisuccinate with N -hydroxysuccinimide and N , N ’-dicyclohexylcarbodiimide followed by amination provided succinic monoamide avermectine esters that are potential antiparasitics.

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Veröffentlicht in:Russian chemical bulletin 2019-05, Vol.68 (5), p.1116-1121
Hauptverfasser: Shchetinina, M. A., Chernoburova, E. I., Kolotyrkina, N. G., Dzhafarov, M. Kh, Vasilevich, F. I., Zavarzin, I. V.
Format: Artikel
Sprache:eng
Schlagworte:
Chemistry
Chemistry and Materials Science
Chemistry/Food Science
Esters
Full Article
Inorganic Chemistry
Organic Chemistry
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Zusammenfassung:Reaction of avermectin B 1 hemisuccinate with N -hydroxysuccinimide and N , N ’-dicyclohexylcarbodiimide followed by amination provided succinic monoamide avermectine esters that are potential antiparasitics.
ISSN:1066-5285
1573-9171
DOI:10.1007/s11172-019-2528-x