N-Arylpiperazine-1-carboxamide Derivatives

A novel series of N-arylpiperazine-1-carboxamide derivatives was synthesized and their androgen receptor (AR) antagonist activities and in vivo antiandrogenic properties were evaluated. Reporter assays indicated that trans-2,5-dimethylpiperazine derivatives are potent AR antagonists, and in this ser...

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Veröffentlicht in:	Chemical & pharmaceutical bulletin 2005-04, Vol.53 (4), p.402
Hauptverfasser:	Kinoyama, Isao, Taniguchi, Nobuaki, Kawaminami, Eiji, Nozawa, Eisuke, Koutoku, Hiroshi, Furutani, Takashi, Kudoh, Masafumi, Okada, Minoru
Format:	Artikel
Sprache:	eng
Online-Zugang:	Volltext
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