Dopamine/serotonin receptor ligands. 10:1 SAR studies on azecine-type dopamine receptor ligands by functional screening at human cloned D1, D2L, and D5 receptors with a microplate reader based calcium assay lead to a novel potent D1/D5 selective antagonist

Dopamine/serotonin receptor ligands. 10:1 SAR studies on azecine-type dopamine receptor ligands by functional screening at human cloned D1, D2L, and D5 receptors with a microplate reader based calcium assay lead to a novel potent D1/D5 selective antagonist

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Veröffentlicht in:Journal of medicinal chemistry 2006, Vol.49 (2), p.760-769
Hauptverfasser: HOEFGEN, Barbara, DECKER, Michael, MOHR, Patrick, SCHRARNM, Astrid M, ROSTOM, Sherif A. F, EL-SUBBAGH, Hussein, SCHWEIKERT, Peter M, RUDOLF, Dirk R, KASSACK, Matthias U, LEHMANN, Jochen
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Biological and medical sciences
Catecholaminergic system
Medical sciences
Neuropharmacology
Neurotransmitters. Neurotransmission. Receptors
Pharmacology. Drug treatments
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container_title Journal of medicinal chemistry
container_volume 49
creator HOEFGEN, Barbara
DECKER, Michael
MOHR, Patrick
SCHRARNM, Astrid M
ROSTOM, Sherif A. F
EL-SUBBAGH, Hussein
SCHWEIKERT, Peter M
RUDOLF, Dirk R
KASSACK, Matthias U
LEHMANN, Jochen
description
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source ACS Publications
subjects Biological and medical sciences
Catecholaminergic system
Medical sciences
Neuropharmacology
Neurotransmitters. Neurotransmission. Receptors
Pharmacology. Drug treatments
title Dopamine/serotonin receptor ligands. 10:1 SAR studies on azecine-type dopamine receptor ligands by functional screening at human cloned D1, D2L, and D5 receptors with a microplate reader based calcium assay lead to a novel potent D1/D5 selective antagonist
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