Discovery of 4-benzoyl-1-[(4-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)oxoacetyl]-2-(R)-methylpi p erazine (BMS-378806): A novel HIV-1 attachment inhibitor that interferes with CD4-gp120 interactions

Discovery of 4-benzoyl-1-[(4-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)oxoacetyl]-2-(R)-methylpi p erazine (BMS-378806): A novel HIV-1 attachment inhibitor that interferes with CD4-gp120 interactions

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Veröffentlicht in:Journal of medicinal chemistry 2003, Vol.46 (20), p.4236-4239
Hauptverfasser: TAO WANG, ZHONGXING ZHANG, RANADIVE, Sunanda, ROBINSON, Brett S, GONG, Yi-Fei, RICARRDI, Keith, SPICER, Timothy P, DEMINIE, Carol, ROSE, Ronald, WANG, Hwei-Gene Heidi, BLAIR, Wade S, SHI, Pei-Yong, WALLACE, Owen B, LIN, Pin-Fang, COLONNO, Richard J, MEANWELL, Nicholas A, DESHPANDE, Milind, HAIQUAN FANG, ZHENG YANG, ZADJURA, Lisa M, TWEEDIE, Donald L, HUANG, Stella, FANG ZHAO
Format: Artikel
Sprache:eng
Schlagworte:
Antibiotics. Antiinfectious agents. Antiparasitic agents
Antiviral agents
Biological and medical sciences
Medical sciences
Pharmacology. Drug treatments
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container_end_page 4239
container_issue 20
container_start_page 4236
container_title Journal of medicinal chemistry
container_volume 46
creator TAO WANG
ZHONGXING ZHANG
RANADIVE, Sunanda
ROBINSON, Brett S
GONG, Yi-Fei
RICARRDI, Keith
SPICER, Timothy P
DEMINIE, Carol
ROSE, Ronald
WANG, Hwei-Gene Heidi
BLAIR, Wade S
SHI, Pei-Yong
WALLACE, Owen B
LIN, Pin-Fang
COLONNO, Richard J
MEANWELL, Nicholas A
DESHPANDE, Milind
HAIQUAN FANG
ZHENG YANG
ZADJURA, Lisa M
TWEEDIE, Donald L
HUANG, Stella
FANG ZHAO
description
format Article
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source American Chemical Society Journals
subjects Antibiotics. Antiinfectious agents. Antiparasitic agents
Antiviral agents
Biological and medical sciences
Medical sciences
Pharmacology. Drug treatments
title Discovery of 4-benzoyl-1-[(4-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)oxoacetyl]-2-(R)-methylpi p erazine (BMS-378806): A novel HIV-1 attachment inhibitor that interferes with CD4-gp120 interactions
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