Chemical scaffold recycling: Structure-guided conversion of an HIV integrase inhibitor into a potent influenza virus RNA-dependent RNA polymerase inhibitor designed to minimize resistance potential

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Veröffentlicht in:European journal of medicinal chemistry 2023-02, Vol.247 (C)
Hauptverfasser: Slavish, Peter J., Cuypers, Maxime G., Rimmer, Mary Ashley, Abdolvahabi, Alireza, Jeevan, Trushar, Kumar, Gyanendra, Jarusiewicz, Jamie A., Vaithiyalingam, Sivaraja, Jones, Jeremy C., Bowling, John J., Price, Jeanine E., DuBois, Rebecca M., Min, Jaeki, Webby, Richard J., Rankovic, Zoran, White, Stephen W.
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container_issue C
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container_title European journal of medicinal chemistry
container_volume 247
creator Slavish, Peter J.
Cuypers, Maxime G.
Rimmer, Mary Ashley
Abdolvahabi, Alireza
Jeevan, Trushar
Kumar, Gyanendra
Jarusiewicz, Jamie A.
Vaithiyalingam, Sivaraja
Jones, Jeremy C.
Bowling, John J.
Price, Jeanine E.
DuBois, Rebecca M.
Min, Jaeki
Webby, Richard J.
Rankovic, Zoran
White, Stephen W.
description Not provided.
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subjects Pharmacology & Pharmacy
title Chemical scaffold recycling: Structure-guided conversion of an HIV integrase inhibitor into a potent influenza virus RNA-dependent RNA polymerase inhibitor designed to minimize resistance potential
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