Palladium-Catalyzed γ‑Selective Arylation of Zincated Boc-Allylamines

The regio- and diastereoselective arylation of Boc-protected allylamines was performed via a one-pot lithiation/transmetalation to zinc/cross-coupling sequence, through an appropriate choice of a phosphine ligand. A variety of γ-arylated products were obtained in moderate to good yield, and the prod...

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Veröffentlicht in:	Organic letters 2014-08, Vol.16 (15), p.3998-4000
Hauptverfasser:	Millet, Anthony, Baudoin, Olivier
Format:	Artikel
Sprache:	eng
Schlagworte:	Chemical Sciences Organic chemistry
Online-Zugang:	Volltext
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