Crystalline form of dihydro-2,3-benzodiazepine derivative

A physical form of (R)-7-acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-7H-1,3-dioxolo[4,5-h][2,3]benzodiazepine having an X-ray powder diffraction pattern with d spacings at 12.78, 9.48, 8.99, 8.64, 8.23, 6.39, 6.27. 5.73, 4.01 and 3.96 Å. The compound is useful as an AMPA antagonist.

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Hauptverfasser: ZMIJEWSKI, MILTON JOSEPH, JR, DAVID LEE VARIE, MARVIN MARTIN HANSEN, EDWARD GRANT GROLEAU, JEFFREY THOMAS VINCENZI, BENJAMIN ALAN ANDERSON
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creator ZMIJEWSKI, MILTON JOSEPH, JR
DAVID LEE VARIE
MARVIN MARTIN HANSEN
EDWARD GRANT GROLEAU
JEFFREY THOMAS VINCENZI
BENJAMIN ALAN ANDERSON
description A physical form of (R)-7-acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-7H-1,3-dioxolo[4,5-h][2,3]benzodiazepine having an X-ray powder diffraction pattern with d spacings at 12.78, 9.48, 8.99, 8.64, 8.23, 6.39, 6.27. 5.73, 4.01 and 3.96 Å. The compound is useful as an AMPA antagonist.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
title Crystalline form of dihydro-2,3-benzodiazepine derivative
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