INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS

Provided herein are compounds of formula (V) that bind to BF3 of an androgen receptor (AR), which can modulate the AR for the treatment of Kennedy's disease. L'invention concerne des composés de formule (V) qui se lient au BF3 d'un récepteur des androgènes (RA), qui peuvent moduler le...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: BAKARY-BARRY, Toure, GALLOP, Mark, BARSANTI, Paul
Format: Patent
Sprache:eng ; fre
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
container_end_page
container_issue
container_start_page
container_title
container_volume
creator BAKARY-BARRY, Toure
GALLOP, Mark
BARSANTI, Paul
description Provided herein are compounds of formula (V) that bind to BF3 of an androgen receptor (AR), which can modulate the AR for the treatment of Kennedy's disease. L'invention concerne des composés de formule (V) qui se lient au BF3 d'un récepteur des androgènes (RA), qui peuvent moduler le RA pour le traitement de la maladie de Kennedy.
format Patent
fullrecord <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_WO2022020342A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>WO2022020342A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_WO2022020342A13</originalsourceid><addsrcrecordid>eNrjZDDw9HPx93FVcPb3DfAP9XMJVnAEIj-XIH93Vz-FIFdn14AQ_yAFX3-XUB9HICuYh4E1LTGnOJUXSnMzKLu5hjh76KYW5MenFhckJqfmpZbEh_sbGRgBkYGxiZGjoTFxqgDXiSdM</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS</title><source>esp@cenet</source><creator>BAKARY-BARRY, Toure ; GALLOP, Mark ; BARSANTI, Paul</creator><creatorcontrib>BAKARY-BARRY, Toure ; GALLOP, Mark ; BARSANTI, Paul</creatorcontrib><description>Provided herein are compounds of formula (V) that bind to BF3 of an androgen receptor (AR), which can modulate the AR for the treatment of Kennedy's disease. L'invention concerne des composés de formule (V) qui se lient au BF3 d'un récepteur des androgènes (RA), qui peuvent moduler le RA pour le traitement de la maladie de Kennedy.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2022</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20220127&amp;DB=EPODOC&amp;CC=WO&amp;NR=2022020342A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76289</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20220127&amp;DB=EPODOC&amp;CC=WO&amp;NR=2022020342A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>BAKARY-BARRY, Toure</creatorcontrib><creatorcontrib>GALLOP, Mark</creatorcontrib><creatorcontrib>BARSANTI, Paul</creatorcontrib><title>INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS</title><description>Provided herein are compounds of formula (V) that bind to BF3 of an androgen receptor (AR), which can modulate the AR for the treatment of Kennedy's disease. L'invention concerne des composés de formule (V) qui se lient au BF3 d'un récepteur des androgènes (RA), qui peuvent moduler le RA pour le traitement de la maladie de Kennedy.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2022</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZDDw9HPx93FVcPb3DfAP9XMJVnAEIj-XIH93Vz-FIFdn14AQ_yAFX3-XUB9HICuYh4E1LTGnOJUXSnMzKLu5hjh76KYW5MenFhckJqfmpZbEh_sbGRgBkYGxiZGjoTFxqgDXiSdM</recordid><startdate>20220127</startdate><enddate>20220127</enddate><creator>BAKARY-BARRY, Toure</creator><creator>GALLOP, Mark</creator><creator>BARSANTI, Paul</creator><scope>EVB</scope></search><sort><creationdate>20220127</creationdate><title>INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS</title><author>BAKARY-BARRY, Toure ; GALLOP, Mark ; BARSANTI, Paul</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2022020342A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2022</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>BAKARY-BARRY, Toure</creatorcontrib><creatorcontrib>GALLOP, Mark</creatorcontrib><creatorcontrib>BARSANTI, Paul</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>BAKARY-BARRY, Toure</au><au>GALLOP, Mark</au><au>BARSANTI, Paul</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS</title><date>2022-01-27</date><risdate>2022</risdate><abstract>Provided herein are compounds of formula (V) that bind to BF3 of an androgen receptor (AR), which can modulate the AR for the treatment of Kennedy's disease. L'invention concerne des composés de formule (V) qui se lient au BF3 d'un récepteur des androgènes (RA), qui peuvent moduler le RA pour le traitement de la maladie de Kennedy.</abstract><oa>free_for_read</oa></addata></record>
fulltext fulltext_linktorsrc
identifier
ispartof
issn
language eng ; fre
recordid cdi_epo_espacenet_WO2022020342A1
source esp@cenet
subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS
url https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-04T13%3A42%3A17IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=BAKARY-BARRY,%20Toure&rft.date=2022-01-27&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EWO2022020342A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true