BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAMS
The invention provides novel compounds having the general formula (I) wherein R1, R2, R3, R4, R5 and X are as described herein, compositions including the compounds and methods of using the compounds. L'invention concerne de nouveaux composés de formule générale (I) dans laquelle R1, R2, R3, R4...
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| creator | KNOFLACH, Frédéric RUNTZ-SCHMITT, Valerie HERNANDEZ, Maria-Clemencia ZORN, Nicolas KOBLET, Andreas OLIVARES MORALES, Andres Miguel WAMSTEEKER CUSULIN, Jaclyn Ivy GOBBI, Luca CECERE, Giuseppe REUTLINGER, Michael O`CONNOR, Eoin Cornelius |
| description | The invention provides novel compounds having the general formula (I) wherein R1, R2, R3, R4, R5 and X are as described herein, compositions including the compounds and methods of using the compounds.
L'invention concerne de nouveaux composés de formule générale (I) dans laquelle R1, R2, R3, R4, R5 et X sont tels que mentionnés dans la description, des compositions comprenant les composés et des procédés d'utilisation des composés. |
| format | Patent |
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L'invention concerne de nouveaux composés de formule générale (I) dans laquelle R1, R2, R3, R4, R5 et X sont tels que mentionnés dans la description, des compositions comprenant les composés et des procédés d'utilisation des composés.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2021</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20211007&DB=EPODOC&CC=WO&NR=2021198124A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25563,76318</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20211007&DB=EPODOC&CC=WO&NR=2021198124A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>KNOFLACH, Frédéric</creatorcontrib><creatorcontrib>RUNTZ-SCHMITT, Valerie</creatorcontrib><creatorcontrib>HERNANDEZ, Maria-Clemencia</creatorcontrib><creatorcontrib>ZORN, Nicolas</creatorcontrib><creatorcontrib>KOBLET, Andreas</creatorcontrib><creatorcontrib>OLIVARES MORALES, Andres Miguel</creatorcontrib><creatorcontrib>WAMSTEEKER CUSULIN, Jaclyn Ivy</creatorcontrib><creatorcontrib>GOBBI, Luca</creatorcontrib><creatorcontrib>CECERE, Giuseppe</creatorcontrib><creatorcontrib>REUTLINGER, Michael</creatorcontrib><creatorcontrib>O`CONNOR, Eoin Cornelius</creatorcontrib><title>BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAMS</title><description>The invention provides novel compounds having the general formula (I) wherein R1, R2, R3, R4, R5 and X are as described herein, compositions including the compounds and methods of using the compounds.
L'invention concerne de nouveaux composés de formule générale (I) dans laquelle R1, R2, R3, R4, R5 et X sont tels que mentionnés dans la description, des compositions comprenant les composés et des procédés d'utilisation des composés.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2021</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZDBwcvWL8nfxdIxyDfD0c1VwcQ3yDHMM8QxzDVZwDFZwd3RyVHAEUr6-joYKAY6-wTwMrGmJOcWpvFCam0HZzTXE2UM3tSA_PrW4IDE5NS-1JD7c38jAyNDQ0sLQyMTR0Jg4VQCgSSbF</recordid><startdate>20211007</startdate><enddate>20211007</enddate><creator>KNOFLACH, Frédéric</creator><creator>RUNTZ-SCHMITT, Valerie</creator><creator>HERNANDEZ, Maria-Clemencia</creator><creator>ZORN, Nicolas</creator><creator>KOBLET, Andreas</creator><creator>OLIVARES MORALES, Andres Miguel</creator><creator>WAMSTEEKER CUSULIN, Jaclyn Ivy</creator><creator>GOBBI, Luca</creator><creator>CECERE, Giuseppe</creator><creator>REUTLINGER, Michael</creator><creator>O`CONNOR, Eoin Cornelius</creator><scope>EVB</scope></search><sort><creationdate>20211007</creationdate><title>BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAMS</title><author>KNOFLACH, Frédéric ; RUNTZ-SCHMITT, Valerie ; HERNANDEZ, Maria-Clemencia ; ZORN, Nicolas ; KOBLET, Andreas ; OLIVARES MORALES, Andres Miguel ; WAMSTEEKER CUSULIN, Jaclyn Ivy ; GOBBI, Luca ; CECERE, Giuseppe ; REUTLINGER, Michael ; O`CONNOR, Eoin Cornelius</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2021198124A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2021</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>KNOFLACH, Frédéric</creatorcontrib><creatorcontrib>RUNTZ-SCHMITT, Valerie</creatorcontrib><creatorcontrib>HERNANDEZ, Maria-Clemencia</creatorcontrib><creatorcontrib>ZORN, Nicolas</creatorcontrib><creatorcontrib>KOBLET, Andreas</creatorcontrib><creatorcontrib>OLIVARES MORALES, Andres Miguel</creatorcontrib><creatorcontrib>WAMSTEEKER CUSULIN, Jaclyn Ivy</creatorcontrib><creatorcontrib>GOBBI, Luca</creatorcontrib><creatorcontrib>CECERE, Giuseppe</creatorcontrib><creatorcontrib>REUTLINGER, Michael</creatorcontrib><creatorcontrib>O`CONNOR, Eoin Cornelius</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>KNOFLACH, Frédéric</au><au>RUNTZ-SCHMITT, Valerie</au><au>HERNANDEZ, Maria-Clemencia</au><au>ZORN, Nicolas</au><au>KOBLET, Andreas</au><au>OLIVARES MORALES, Andres Miguel</au><au>WAMSTEEKER CUSULIN, Jaclyn Ivy</au><au>GOBBI, Luca</au><au>CECERE, Giuseppe</au><au>REUTLINGER, Michael</au><au>O`CONNOR, Eoin Cornelius</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAMS</title><date>2021-10-07</date><risdate>2021</risdate><abstract>The invention provides novel compounds having the general formula (I) wherein R1, R2, R3, R4, R5 and X are as described herein, compositions including the compounds and methods of using the compounds.
L'invention concerne de nouveaux composés de formule générale (I) dans laquelle R1, R2, R3, R4, R5 et X sont tels que mentionnés dans la description, des compositions comprenant les composés et des procédés d'utilisation des composés.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAMS |
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