PHARMACEUTICAL COMPOSITION COMPRISING AMORPHOUS SELEXIPAG

The present invention is directed to solid state forms of selexipag (Formula (I)), including an amorphous form of selexipag and a selexipag-containing premix, to methods for their preparation, to pharmaceutical compositions comprising them and to their use in medicine, particularly for the treatment...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: MALHOTRA, Geena, PUPPALA, Ravikumar, GANGRADE, Manish Gopaldas, PATHI, Srinivas Laxminarayan, RAO, Dharmaraj Ramachandra, KOMMULA, Narayanaswami, RANKIREDDI, Anand Ramesh
Format: Patent
Sprache:eng ; fre
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
container_end_page
container_issue
container_start_page
container_title
container_volume
creator MALHOTRA, Geena
PUPPALA, Ravikumar
GANGRADE, Manish Gopaldas
PATHI, Srinivas Laxminarayan
RAO, Dharmaraj Ramachandra
KOMMULA, Narayanaswami
RANKIREDDI, Anand Ramesh
description The present invention is directed to solid state forms of selexipag (Formula (I)), including an amorphous form of selexipag and a selexipag-containing premix, to methods for their preparation, to pharmaceutical compositions comprising them and to their use in medicine, particularly for the treatment of pulmonary arterial hypertension. (Formula (I)) La présente invention concerne des formes à l'état solide de selexipag (formule (I)), comprenant une forme amorphe du selexipag et un pré-mélange contenant du selexipag, des méthodes pour leur préparation, des compositions pharmaceutiques les comprenant et leur utilisation en médecine, en particulier pour le traitement de l'hypertension artérielle pulmonaire. (Formule (I))
format Patent
fullrecord <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_WO2018078383A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>WO2018078383A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_WO2018078383A13</originalsourceid><addsrcrecordid>eNrjZLAM8HAM8nV0dg0N8XR29FFw9vcN8A_2DPH09wOzgzyDPf3cFRx9_YMCPPxDgxWCXX1cIzwDHN15GFjTEnOKU3mhNDeDsptriLOHbmpBfnxqcUFicmpeakl8uL-RgaGFgbmFsYWxo6ExcaoAd68qUg</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>PHARMACEUTICAL COMPOSITION COMPRISING AMORPHOUS SELEXIPAG</title><source>esp@cenet</source><creator>MALHOTRA, Geena ; PUPPALA, Ravikumar ; GANGRADE, Manish Gopaldas ; PATHI, Srinivas Laxminarayan ; RAO, Dharmaraj Ramachandra ; KOMMULA, Narayanaswami ; RANKIREDDI, Anand Ramesh</creator><creatorcontrib>MALHOTRA, Geena ; PUPPALA, Ravikumar ; GANGRADE, Manish Gopaldas ; PATHI, Srinivas Laxminarayan ; RAO, Dharmaraj Ramachandra ; KOMMULA, Narayanaswami ; RANKIREDDI, Anand Ramesh</creatorcontrib><description>The present invention is directed to solid state forms of selexipag (Formula (I)), including an amorphous form of selexipag and a selexipag-containing premix, to methods for their preparation, to pharmaceutical compositions comprising them and to their use in medicine, particularly for the treatment of pulmonary arterial hypertension. (Formula (I)) La présente invention concerne des formes à l'état solide de selexipag (formule (I)), comprenant une forme amorphe du selexipag et un pré-mélange contenant du selexipag, des méthodes pour leur préparation, des compositions pharmaceutiques les comprenant et leur utilisation en médecine, en particulier pour le traitement de l'hypertension artérielle pulmonaire. (Formule (I))</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2018</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20180503&amp;DB=EPODOC&amp;CC=WO&amp;NR=2018078383A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,777,882,25545,76296</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20180503&amp;DB=EPODOC&amp;CC=WO&amp;NR=2018078383A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>MALHOTRA, Geena</creatorcontrib><creatorcontrib>PUPPALA, Ravikumar</creatorcontrib><creatorcontrib>GANGRADE, Manish Gopaldas</creatorcontrib><creatorcontrib>PATHI, Srinivas Laxminarayan</creatorcontrib><creatorcontrib>RAO, Dharmaraj Ramachandra</creatorcontrib><creatorcontrib>KOMMULA, Narayanaswami</creatorcontrib><creatorcontrib>RANKIREDDI, Anand Ramesh</creatorcontrib><title>PHARMACEUTICAL COMPOSITION COMPRISING AMORPHOUS SELEXIPAG</title><description>The present invention is directed to solid state forms of selexipag (Formula (I)), including an amorphous form of selexipag and a selexipag-containing premix, to methods for their preparation, to pharmaceutical compositions comprising them and to their use in medicine, particularly for the treatment of pulmonary arterial hypertension. (Formula (I)) La présente invention concerne des formes à l'état solide de selexipag (formule (I)), comprenant une forme amorphe du selexipag et un pré-mélange contenant du selexipag, des méthodes pour leur préparation, des compositions pharmaceutiques les comprenant et leur utilisation en médecine, en particulier pour le traitement de l'hypertension artérielle pulmonaire. (Formule (I))</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2018</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZLAM8HAM8nV0dg0N8XR29FFw9vcN8A_2DPH09wOzgzyDPf3cFRx9_YMCPPxDgxWCXX1cIzwDHN15GFjTEnOKU3mhNDeDsptriLOHbmpBfnxqcUFicmpeakl8uL-RgaGFgbmFsYWxo6ExcaoAd68qUg</recordid><startdate>20180503</startdate><enddate>20180503</enddate><creator>MALHOTRA, Geena</creator><creator>PUPPALA, Ravikumar</creator><creator>GANGRADE, Manish Gopaldas</creator><creator>PATHI, Srinivas Laxminarayan</creator><creator>RAO, Dharmaraj Ramachandra</creator><creator>KOMMULA, Narayanaswami</creator><creator>RANKIREDDI, Anand Ramesh</creator><scope>EVB</scope></search><sort><creationdate>20180503</creationdate><title>PHARMACEUTICAL COMPOSITION COMPRISING AMORPHOUS SELEXIPAG</title><author>MALHOTRA, Geena ; PUPPALA, Ravikumar ; GANGRADE, Manish Gopaldas ; PATHI, Srinivas Laxminarayan ; RAO, Dharmaraj Ramachandra ; KOMMULA, Narayanaswami ; RANKIREDDI, Anand Ramesh</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2018078383A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2018</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>MALHOTRA, Geena</creatorcontrib><creatorcontrib>PUPPALA, Ravikumar</creatorcontrib><creatorcontrib>GANGRADE, Manish Gopaldas</creatorcontrib><creatorcontrib>PATHI, Srinivas Laxminarayan</creatorcontrib><creatorcontrib>RAO, Dharmaraj Ramachandra</creatorcontrib><creatorcontrib>KOMMULA, Narayanaswami</creatorcontrib><creatorcontrib>RANKIREDDI, Anand Ramesh</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>MALHOTRA, Geena</au><au>PUPPALA, Ravikumar</au><au>GANGRADE, Manish Gopaldas</au><au>PATHI, Srinivas Laxminarayan</au><au>RAO, Dharmaraj Ramachandra</au><au>KOMMULA, Narayanaswami</au><au>RANKIREDDI, Anand Ramesh</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>PHARMACEUTICAL COMPOSITION COMPRISING AMORPHOUS SELEXIPAG</title><date>2018-05-03</date><risdate>2018</risdate><abstract>The present invention is directed to solid state forms of selexipag (Formula (I)), including an amorphous form of selexipag and a selexipag-containing premix, to methods for their preparation, to pharmaceutical compositions comprising them and to their use in medicine, particularly for the treatment of pulmonary arterial hypertension. (Formula (I)) La présente invention concerne des formes à l'état solide de selexipag (formule (I)), comprenant une forme amorphe du selexipag et un pré-mélange contenant du selexipag, des méthodes pour leur préparation, des compositions pharmaceutiques les comprenant et leur utilisation en médecine, en particulier pour le traitement de l'hypertension artérielle pulmonaire. (Formule (I))</abstract><oa>free_for_read</oa></addata></record>
fulltext fulltext_linktorsrc
identifier
ispartof
issn
language eng ; fre
recordid cdi_epo_espacenet_WO2018078383A1
source esp@cenet
subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title PHARMACEUTICAL COMPOSITION COMPRISING AMORPHOUS SELEXIPAG
url https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-17T16%3A12%3A41IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=MALHOTRA,%20Geena&rft.date=2018-05-03&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EWO2018078383A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true