PYRAZINE COMPOUNDS FOR USE IN THE TREATMENT OF PARASITIC PROTOZOAL INFECTIONS

The present invention relates to compounds of Formula (I) having pharmacological activity, processes for its preparation, pharmaceutical compositions and their use in the treatment of certain parasitic certain parasiticprotozoalinfections such as malaria, in particular infection by Plasmodium falcip...

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Hauptverfasser: GARCIA MARTIN, Mercedes, CASTELLOTE ALVARO, Maria Isabel
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creator GARCIA MARTIN, Mercedes
CASTELLOTE ALVARO, Maria Isabel
description The present invention relates to compounds of Formula (I) having pharmacological activity, processes for its preparation, pharmaceutical compositions and their use in the treatment of certain parasitic certain parasiticprotozoalinfections such as malaria, in particular infection by Plasmodium falciparum. Formula (I), wherein R is methyl or fluoro. La présente invention concerne des composés de formule (I) présentant une activité pharmacologique, des procédés pour leur préparation, des compositions pharmaceutiques et leur utilisation dans le traitement de certaines infections causées par des protozoaires parasites telles que la malaria, en particulier une infection par Plasmodium falciparum. Formule (I), dans laquelle R est un méthyle ou un fluoro.
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Formula (I), wherein R is methyl or fluoro. La présente invention concerne des composés de formule (I) présentant une activité pharmacologique, des procédés pour leur préparation, des compositions pharmaceutiques et leur utilisation dans le traitement de certaines infections causées par des protozoaires parasites telles que la malaria, en particulier une infection par Plasmodium falciparum. 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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title PYRAZINE COMPOUNDS FOR USE IN THE TREATMENT OF PARASITIC PROTOZOAL INFECTIONS
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