SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS
The invention provides compounds of Formula (I): and pharmaceutically acceptable salts thereof. The compounds of Formula (I) inhibit protein kinase activity thereby making them useful as anticancer agents. L'invention concerne des composés de formule (I) et leurs sels pharmaceutiquement accepta...
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| creator | LIU, PEIYING REDDY, BANDREDDY SUBBA PEARCE, BRADLEY C BORA, RAJESH ONKARDAS KUMARAVEL, SELVAKUMAR DASGUPTA, BIRESHWAR NAGALAKSHMI, PULICHARLA MULLICK, DIBAKAR NAIR, JALATHI SURENDRAN JANAKIRAMAN, SAKTHI KUMARAN RAO, METTU MALLIKARJUNA ARAUJO, ERIKA M.V WITTMAN, MARK D RACHAMREDDY, CHANDRASEKHAR REDDY KARUPPIAH, ARUL MOZHI SELVAN SUBBIAH MAHESHWARAPPA, SHILPA HOLEHATTI SISTLA, RAMESH VELAPARTHI, UPENDER DARNE, CHETAN PADMAKAR |
| description | The invention provides compounds of Formula (I): and pharmaceutically acceptable salts thereof. The compounds of Formula (I) inhibit protein kinase activity thereby making them useful as anticancer agents.
L'invention concerne des composés de formule (I) et leurs sels pharmaceutiquement acceptables. Les composés de formule (I) inhibent l'activité protéine kinase, ce qui leur permet d'être utilisés comme agents anticancéreux. |
| format | Patent |
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L'invention concerne des composés de formule (I) et leurs sels pharmaceutiquement acceptables. Les composés de formule (I) inhibent l'activité protéine kinase, ce qui leur permet d'être utilisés comme agents anticancéreux.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2015</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20150521&DB=EPODOC&CC=WO&NR=2015073763A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25543,76293</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20150521&DB=EPODOC&CC=WO&NR=2015073763A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>LIU, PEIYING</creatorcontrib><creatorcontrib>REDDY, BANDREDDY SUBBA</creatorcontrib><creatorcontrib>PEARCE, BRADLEY C</creatorcontrib><creatorcontrib>BORA, RAJESH ONKARDAS</creatorcontrib><creatorcontrib>KUMARAVEL, SELVAKUMAR</creatorcontrib><creatorcontrib>DASGUPTA, BIRESHWAR</creatorcontrib><creatorcontrib>NAGALAKSHMI, PULICHARLA</creatorcontrib><creatorcontrib>MULLICK, DIBAKAR</creatorcontrib><creatorcontrib>NAIR, JALATHI SURENDRAN</creatorcontrib><creatorcontrib>JANAKIRAMAN, SAKTHI KUMARAN</creatorcontrib><creatorcontrib>RAO, METTU MALLIKARJUNA</creatorcontrib><creatorcontrib>ARAUJO, ERIKA M.V</creatorcontrib><creatorcontrib>WITTMAN, MARK D</creatorcontrib><creatorcontrib>RACHAMREDDY, CHANDRASEKHAR REDDY</creatorcontrib><creatorcontrib>KARUPPIAH, ARUL MOZHI SELVAN SUBBIAH</creatorcontrib><creatorcontrib>MAHESHWARAPPA, SHILPA HOLEHATTI</creatorcontrib><creatorcontrib>SISTLA, RAMESH</creatorcontrib><creatorcontrib>VELAPARTHI, UPENDER</creatorcontrib><creatorcontrib>DARNE, CHETAN PADMAKAR</creatorcontrib><title>SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS</title><description>The invention provides compounds of Formula (I): and pharmaceutically acceptable salts thereof. The compounds of Formula (I) inhibit protein kinase activity thereby making them useful as anticancer agents.
L'invention concerne des composés de formule (I) et leurs sels pharmaceutiquement acceptables. Les composés de formule (I) inhibent l'activité protéine kinase, ce qui leur permet d'être utilisés comme agents anticancéreux.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2015</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNisEKgkAUAL10iOofHnRdyc3U8-q-8FG4sfs0LEJEtlOUUP9PEX1Ap5mBmQaDq3PHxDWjho1IRCqykJGtKlttzaG16mT25ixFEqrLN6lC0GipUUwNOlAOCuWQKthR9RGQoFcIVJWUExvr5sHk2t-efvHjLFhukYsy9OOj88-xH_zdv7qjWUcyibI4S2Ml4_-uN984NQE</recordid><startdate>20150521</startdate><enddate>20150521</enddate><creator>LIU, PEIYING</creator><creator>REDDY, BANDREDDY SUBBA</creator><creator>PEARCE, BRADLEY C</creator><creator>BORA, RAJESH ONKARDAS</creator><creator>KUMARAVEL, SELVAKUMAR</creator><creator>DASGUPTA, BIRESHWAR</creator><creator>NAGALAKSHMI, PULICHARLA</creator><creator>MULLICK, DIBAKAR</creator><creator>NAIR, JALATHI SURENDRAN</creator><creator>JANAKIRAMAN, SAKTHI KUMARAN</creator><creator>RAO, METTU MALLIKARJUNA</creator><creator>ARAUJO, ERIKA M.V</creator><creator>WITTMAN, MARK D</creator><creator>RACHAMREDDY, CHANDRASEKHAR REDDY</creator><creator>KARUPPIAH, ARUL MOZHI SELVAN SUBBIAH</creator><creator>MAHESHWARAPPA, SHILPA HOLEHATTI</creator><creator>SISTLA, RAMESH</creator><creator>VELAPARTHI, UPENDER</creator><creator>DARNE, CHETAN PADMAKAR</creator><scope>EVB</scope></search><sort><creationdate>20150521</creationdate><title>SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS</title><author>LIU, PEIYING ; REDDY, BANDREDDY SUBBA ; PEARCE, BRADLEY C ; BORA, RAJESH ONKARDAS ; KUMARAVEL, SELVAKUMAR ; DASGUPTA, BIRESHWAR ; NAGALAKSHMI, PULICHARLA ; MULLICK, DIBAKAR ; NAIR, JALATHI SURENDRAN ; JANAKIRAMAN, SAKTHI KUMARAN ; RAO, METTU MALLIKARJUNA ; ARAUJO, ERIKA M.V ; WITTMAN, MARK D ; RACHAMREDDY, CHANDRASEKHAR REDDY ; KARUPPIAH, ARUL MOZHI SELVAN SUBBIAH ; MAHESHWARAPPA, SHILPA HOLEHATTI ; SISTLA, RAMESH ; VELAPARTHI, UPENDER ; DARNE, CHETAN PADMAKAR</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2015073763A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2015</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>LIU, PEIYING</creatorcontrib><creatorcontrib>REDDY, BANDREDDY SUBBA</creatorcontrib><creatorcontrib>PEARCE, BRADLEY C</creatorcontrib><creatorcontrib>BORA, RAJESH ONKARDAS</creatorcontrib><creatorcontrib>KUMARAVEL, SELVAKUMAR</creatorcontrib><creatorcontrib>DASGUPTA, BIRESHWAR</creatorcontrib><creatorcontrib>NAGALAKSHMI, PULICHARLA</creatorcontrib><creatorcontrib>MULLICK, DIBAKAR</creatorcontrib><creatorcontrib>NAIR, JALATHI SURENDRAN</creatorcontrib><creatorcontrib>JANAKIRAMAN, SAKTHI KUMARAN</creatorcontrib><creatorcontrib>RAO, METTU MALLIKARJUNA</creatorcontrib><creatorcontrib>ARAUJO, ERIKA M.V</creatorcontrib><creatorcontrib>WITTMAN, MARK D</creatorcontrib><creatorcontrib>RACHAMREDDY, CHANDRASEKHAR REDDY</creatorcontrib><creatorcontrib>KARUPPIAH, ARUL MOZHI SELVAN SUBBIAH</creatorcontrib><creatorcontrib>MAHESHWARAPPA, SHILPA HOLEHATTI</creatorcontrib><creatorcontrib>SISTLA, RAMESH</creatorcontrib><creatorcontrib>VELAPARTHI, UPENDER</creatorcontrib><creatorcontrib>DARNE, CHETAN PADMAKAR</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>LIU, PEIYING</au><au>REDDY, BANDREDDY SUBBA</au><au>PEARCE, BRADLEY C</au><au>BORA, RAJESH ONKARDAS</au><au>KUMARAVEL, SELVAKUMAR</au><au>DASGUPTA, BIRESHWAR</au><au>NAGALAKSHMI, PULICHARLA</au><au>MULLICK, DIBAKAR</au><au>NAIR, JALATHI SURENDRAN</au><au>JANAKIRAMAN, SAKTHI KUMARAN</au><au>RAO, METTU MALLIKARJUNA</au><au>ARAUJO, ERIKA M.V</au><au>WITTMAN, MARK D</au><au>RACHAMREDDY, CHANDRASEKHAR REDDY</au><au>KARUPPIAH, ARUL MOZHI SELVAN SUBBIAH</au><au>MAHESHWARAPPA, SHILPA HOLEHATTI</au><au>SISTLA, RAMESH</au><au>VELAPARTHI, UPENDER</au><au>DARNE, CHETAN PADMAKAR</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS</title><date>2015-05-21</date><risdate>2015</risdate><abstract>The invention provides compounds of Formula (I): and pharmaceutically acceptable salts thereof. The compounds of Formula (I) inhibit protein kinase activity thereby making them useful as anticancer agents.
L'invention concerne des composés de formule (I) et leurs sels pharmaceutiquement acceptables. Les composés de formule (I) inhibent l'activité protéine kinase, ce qui leur permet d'être utilisés comme agents anticancéreux.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS |
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