AUGMENTING MOIETIES FOR ANTI-INFLAMMATORY COMPOUNDS
Augmented or synergized anti-inflammatory constructs are disclosed including terpenes covalently conjugated with other anti-inflammatory molecules such as nonsteroidal anti-inflammatory drugs, vanilloids, amino acids and polyamines; and anti-inflammatory molecules covalently conjugated with specific...
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| creator | HECK, DIANE, E LASKIN, JEFFREY, D LACEY, CARL, JEFFREY HEINDEL, NED, D YOUNG, SHERRI, C |
| description | Augmented or synergized anti-inflammatory constructs are disclosed including terpenes covalently conjugated with other anti-inflammatory molecules such as nonsteroidal anti-inflammatory drugs, vanilloids, amino acids and polyamines; and anti-inflammatory molecules covalently conjugated with specific amino acids. For the latter, further conjugation with a choline bioisostere further augments the anti-inflammatory activity.
L'invention concerne des constructions anti-inflammatoires augmentées ou synergétiques, notamment des terpènes conjugués de manière covalente à d'autres molécules anti-inflammatoires, comme des médicaments anti-inflammatoires non stéroïdiens, des vanilloïdes, des acides aminés et des polyamines ; ainsi que des molécules anti-inflammatoires conjuguées de manière covalente à des acides aminés spécifiques. Dans ce dernier cas, une conjugaison supplémentaire avec un bioisostère de la choline augmente davantage l'activité anti-inflammatoire. |
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L'invention concerne des constructions anti-inflammatoires augmentées ou synergétiques, notamment des terpènes conjugués de manière covalente à d'autres molécules anti-inflammatoires, comme des médicaments anti-inflammatoires non stéroïdiens, des vanilloïdes, des acides aminés et des polyamines ; ainsi que des molécules anti-inflammatoires conjuguées de manière covalente à des acides aminés spécifiques. Dans ce dernier cas, une conjugaison supplémentaire avec un bioisostère de la choline augmente davantage l'activité anti-inflammatoire.</description><language>eng ; fre</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><creationdate>2014</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20140918&DB=EPODOC&CC=WO&NR=2014144073A2$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20140918&DB=EPODOC&CC=WO&NR=2014144073A2$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>HECK, DIANE, E</creatorcontrib><creatorcontrib>LASKIN, JEFFREY, D</creatorcontrib><creatorcontrib>LACEY, CARL, JEFFREY</creatorcontrib><creatorcontrib>HEINDEL, NED, D</creatorcontrib><creatorcontrib>YOUNG, SHERRI, C</creatorcontrib><title>AUGMENTING MOIETIES FOR ANTI-INFLAMMATORY COMPOUNDS</title><description>Augmented or synergized anti-inflammatory constructs are disclosed including terpenes covalently conjugated with other anti-inflammatory molecules such as nonsteroidal anti-inflammatory drugs, vanilloids, amino acids and polyamines; and anti-inflammatory molecules covalently conjugated with specific amino acids. For the latter, further conjugation with a choline bioisostere further augments the anti-inflammatory activity.
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L'invention concerne des constructions anti-inflammatoires augmentées ou synergétiques, notamment des terpènes conjugués de manière covalente à d'autres molécules anti-inflammatoires, comme des médicaments anti-inflammatoires non stéroïdiens, des vanilloïdes, des acides aminés et des polyamines ; ainsi que des molécules anti-inflammatoires conjuguées de manière covalente à des acides aminés spécifiques. Dans ce dernier cas, une conjugaison supplémentaire avec un bioisostère de la choline augmente davantage l'activité anti-inflammatoire.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES |
| title | AUGMENTING MOIETIES FOR ANTI-INFLAMMATORY COMPOUNDS |
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