A CRYSTALLINE FORM OF A SALT OF A MORPHOLINO SULFONYL INDOLE DERIVATIVE AND A PROCESS FOR ITS PREPARATION
The present invention relates to a crystalline form of a pharmaceutically acceptable salt of a morpholino sulphonyl indole derivative, that is capable of inhibiting, modulating and/or regulating Insulin-Like-Growth Factor I Receptor and Insulin Receptor. The present invention also relates to a proce...
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creator | CHENNAMSETTY, SUNEEL, MANOHAR, BABU JOSHI, KISHOR HULAWALE, YOGESH CHINCHWADE, YOGESH HARIHARAN, SIVARAMAKRISHNAN SIVAKUMAR, MEENAKSHI PARAMASIVAN, SELVAM |
description | The present invention relates to a crystalline form of a pharmaceutically acceptable salt of a morpholino sulphonyl indole derivative, that is capable of inhibiting, modulating and/or regulating Insulin-Like-Growth Factor I Receptor and Insulin Receptor. The present invention also relates to a process for the preparation of the crystalline form of said compound. Formula (I):
La présente invention concerne une forme cristalline d'un sel pharmaceutiquement acceptable d'un dérivé de morpholinosulfonylindole, qui peut inhiber, moduler et/ou réguler le récepteur du facteur de croissance analogue à l'insuline I et le récepteur de l'insuline. La présente invention concerne également un procédé de préparation de la forme cristalline dudit composé. Formule (I) : |
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La présente invention concerne une forme cristalline d'un sel pharmaceutiquement acceptable d'un dérivé de morpholinosulfonylindole, qui peut inhiber, moduler et/ou réguler le récepteur du facteur de croissance analogue à l'insuline I et le récepteur de l'insuline. La présente invention concerne également un procédé de préparation de la forme cristalline dudit composé. Formule (I) :</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2012</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20121026&DB=EPODOC&CC=WO&NR=2012143879A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76516</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20121026&DB=EPODOC&CC=WO&NR=2012143879A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>CHENNAMSETTY, SUNEEL, MANOHAR, BABU</creatorcontrib><creatorcontrib>JOSHI, KISHOR</creatorcontrib><creatorcontrib>HULAWALE, YOGESH</creatorcontrib><creatorcontrib>CHINCHWADE, YOGESH</creatorcontrib><creatorcontrib>HARIHARAN, SIVARAMAKRISHNAN</creatorcontrib><creatorcontrib>SIVAKUMAR, MEENAKSHI</creatorcontrib><creatorcontrib>PARAMASIVAN, SELVAM</creatorcontrib><title>A CRYSTALLINE FORM OF A SALT OF A MORPHOLINO SULFONYL INDOLE DERIVATIVE AND A PROCESS FOR ITS PREPARATION</title><description>The present invention relates to a crystalline form of a pharmaceutically acceptable salt of a morpholino sulphonyl indole derivative, that is capable of inhibiting, modulating and/or regulating Insulin-Like-Growth Factor I Receptor and Insulin Receptor. The present invention also relates to a process for the preparation of the crystalline form of said compound. Formula (I):
La présente invention concerne une forme cristalline d'un sel pharmaceutiquement acceptable d'un dérivé de morpholinosulfonylindole, qui peut inhiber, moduler et/ou réguler le récepteur du facteur de croissance analogue à l'insuline I et le récepteur de l'insuline. La présente invention concerne également un procédé de préparation de la forme cristalline dudit composé. Formule (I) :</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2012</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNjMEKwjAQRHvxIOo_LHgWbCuox6XZ0ECaDUms9FSKRBBEC_X_MaIf4GlmeI-ZZzeEynU-oNbKEEh2DbAEBI86fFvDztacMIM_acmm06CMYE0gyKkWg2oJ0IjkWscVef_5ARV82mTRJYPNMptdh_sUV79cZGtJoao3cXz2cRqHS3zEV3_mYpsX-a487I-Yl_9Zb_N7Nok</recordid><startdate>20121026</startdate><enddate>20121026</enddate><creator>CHENNAMSETTY, SUNEEL, MANOHAR, BABU</creator><creator>JOSHI, KISHOR</creator><creator>HULAWALE, YOGESH</creator><creator>CHINCHWADE, YOGESH</creator><creator>HARIHARAN, SIVARAMAKRISHNAN</creator><creator>SIVAKUMAR, MEENAKSHI</creator><creator>PARAMASIVAN, SELVAM</creator><scope>EVB</scope></search><sort><creationdate>20121026</creationdate><title>A CRYSTALLINE FORM OF A SALT OF A MORPHOLINO SULFONYL INDOLE DERIVATIVE AND A PROCESS FOR ITS PREPARATION</title><author>CHENNAMSETTY, SUNEEL, MANOHAR, BABU ; JOSHI, KISHOR ; HULAWALE, YOGESH ; CHINCHWADE, YOGESH ; HARIHARAN, SIVARAMAKRISHNAN ; SIVAKUMAR, MEENAKSHI ; PARAMASIVAN, SELVAM</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2012143879A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2012</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>CHENNAMSETTY, SUNEEL, MANOHAR, BABU</creatorcontrib><creatorcontrib>JOSHI, KISHOR</creatorcontrib><creatorcontrib>HULAWALE, YOGESH</creatorcontrib><creatorcontrib>CHINCHWADE, YOGESH</creatorcontrib><creatorcontrib>HARIHARAN, SIVARAMAKRISHNAN</creatorcontrib><creatorcontrib>SIVAKUMAR, MEENAKSHI</creatorcontrib><creatorcontrib>PARAMASIVAN, SELVAM</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>CHENNAMSETTY, SUNEEL, MANOHAR, BABU</au><au>JOSHI, KISHOR</au><au>HULAWALE, YOGESH</au><au>CHINCHWADE, YOGESH</au><au>HARIHARAN, SIVARAMAKRISHNAN</au><au>SIVAKUMAR, MEENAKSHI</au><au>PARAMASIVAN, SELVAM</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>A CRYSTALLINE FORM OF A SALT OF A MORPHOLINO SULFONYL INDOLE DERIVATIVE AND A PROCESS FOR ITS PREPARATION</title><date>2012-10-26</date><risdate>2012</risdate><abstract>The present invention relates to a crystalline form of a pharmaceutically acceptable salt of a morpholino sulphonyl indole derivative, that is capable of inhibiting, modulating and/or regulating Insulin-Like-Growth Factor I Receptor and Insulin Receptor. The present invention also relates to a process for the preparation of the crystalline form of said compound. Formula (I):
La présente invention concerne une forme cristalline d'un sel pharmaceutiquement acceptable d'un dérivé de morpholinosulfonylindole, qui peut inhiber, moduler et/ou réguler le récepteur du facteur de croissance analogue à l'insuline I et le récepteur de l'insuline. La présente invention concerne également un procédé de préparation de la forme cristalline dudit composé. Formule (I) :</abstract><oa>free_for_read</oa></addata></record> |
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subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
title | A CRYSTALLINE FORM OF A SALT OF A MORPHOLINO SULFONYL INDOLE DERIVATIVE AND A PROCESS FOR ITS PREPARATION |
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