NOVEL AZAPEPTIDE OR AZAPEPTIDOMIMETIC COMPOUNDS INHIBITING BCRP AND/OR P-GP

The present invention relates to azapeptide or azapeptidomimetic compounds of formula (I): where R1, R2, R3, X1, X2, X2, X4 and Y are as defined in claim 1, to the pharmaceutical compositions containing said compounds and to such compounds as adjuvants for anti-cancer or anti-infective drugs. La pré...

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Hauptverfasser: DI PIETRO, ATILLIO, ARNAUD, OPHELIE, FALSON, PIERRE, PARIS, JOELLE, MILLION, MARIE-EMMANUELLE
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creator DI PIETRO, ATILLIO
ARNAUD, OPHELIE
FALSON, PIERRE
PARIS, JOELLE
MILLION, MARIE-EMMANUELLE
description The present invention relates to azapeptide or azapeptidomimetic compounds of formula (I): where R1, R2, R3, X1, X2, X2, X4 and Y are as defined in claim 1, to the pharmaceutical compositions containing said compounds and to such compounds as adjuvants for anti-cancer or anti-infective drugs. La présente invention concerne composés de type azapeptide ou azapeptidomimétique de formule (I) : dans laquelle R1, R2, R3, X1, X2, X2, X4 et Y sont tels que définis à la revendication 1, les compositions pharmaceutiques les contenant et de tels composés en tant qu'adjuvant d'un médicament anti-cancéreux ou anti¬ infectieux.
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subjects ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
title NOVEL AZAPEPTIDE OR AZAPEPTIDOMIMETIC COMPOUNDS INHIBITING BCRP AND/OR P-GP
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