NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA-2 RECEPTORS
The present invention relates to named compounds of the formula (I) having both M3 receptor antagonist and ß2 agonist activity; compositions comprising such compounds; the use of such compounds in therapy (such as respiratory tract disorders); and a method of treating a patient with such compounds....
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| creator | ROUSSEL, FABIEN SUTTON, JONATHAN, MARK ALCARAZ, LILIAN VAN DEN HEUVEL, MARCO RAY, NICHOLAS, CHARLES |
| description | The present invention relates to named compounds of the formula (I) having both M3 receptor antagonist and ß2 agonist activity; compositions comprising such compounds; the use of such compounds in therapy (such as respiratory tract disorders); and a method of treating a patient with such compounds.
La présente invention porte sur les composés cités représentés par la formule (I) ayant à la fois une activité d'antagoniste des récepteurs M3 et une activité d'agoniste des récepteurs ß2 ; sur des compositions comprenant de tels composés ; sur l'utilisation de tels composés en thérapie (telle que pour des troubles des voies respiratoires) ; et sur une méthode de traitement d'un patient avec de tels composés. |
| format | Patent |
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La présente invention porte sur les composés cités représentés par la formule (I) ayant à la fois une activité d'antagoniste des récepteurs M3 et une activité d'agoniste des récepteurs ß2 ; sur des compositions comprenant de tels composés ; sur l'utilisation de tels composés en thérapie (telle que pour des troubles des voies respiratoires) ; et sur une méthode de traitement d'un patient avec de tels composés.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2010</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20100211&DB=EPODOC&CC=WO&NR=2010015792A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25562,76317</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20100211&DB=EPODOC&CC=WO&NR=2010015792A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>ROUSSEL, FABIEN</creatorcontrib><creatorcontrib>SUTTON, JONATHAN, MARK</creatorcontrib><creatorcontrib>ALCARAZ, LILIAN</creatorcontrib><creatorcontrib>VAN DEN HEUVEL, MARCO</creatorcontrib><creatorcontrib>RAY, NICHOLAS, CHARLES</creatorcontrib><title>NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA-2 RECEPTORS</title><description>The present invention relates to named compounds of the formula (I) having both M3 receptor antagonist and ß2 agonist activity; compositions comprising such compounds; the use of such compounds in therapy (such as respiratory tract disorders); and a method of treating a patient with such compounds.
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA-2 RECEPTORS |
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