INHIBITION OF INVERTEBRATES USING LIGANDS THAT MODULATE ECDYSONE RECEPTORS
The present invention relates to the use of N-substituted ?-methylene ?-lactams as non- steroidal ligands for modulating ecdysone receptors generally (resulting in controlled insect growth) and, in particular, ecdysone receptors of the Australian blowfly, Lucilia cuprina and the sheep body louse Bov...
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creator | LIEPA, ANDRIS JURIS TURNER, KATHLEEN ANNE JOHNSON, WYNONA MARGUERITE |
description | The present invention relates to the use of N-substituted ?-methylene ?-lactams as non- steroidal ligands for modulating ecdysone receptors generally (resulting in controlled insect growth) and, in particular, ecdysone receptors of the Australian blowfly, Lucilia cuprina and the sheep body louse Bovicola ovis. The present invention further relates to novel N-substituted ?-methylene ?-lactams. These compounds are useful as insecticides or as lead compounds for the development of insecticides. The compounds are also useful as effectors for ecdysone switches.
La présente invention concerne l'utilisation de ?-méthylène ?-lactames N-substituées en tant que ligands non stéroïdiens permettant de moduler les récepteurs de l'ecdysone en général (ce qui permet de contrôler la croissance des insectes), et en particulier les récepteurs de l'ecdysone de la calliphore australienne, Lucilia cuprina, et du pou du mouton, Bovicola ovis. L'invention a également trait à de nouvelles ?-méthylène ?-lactames N-substituées. Lesdits composés sont utiles en tant qu'insecticides ou en tant que têtes de série permettant l'élaboration d'insecticides. Les composés sont également utiles en tant qu'effecteurs pour les commutateurs de l'ecdysone. |
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La présente invention concerne l'utilisation de ?-méthylène ?-lactames N-substituées en tant que ligands non stéroïdiens permettant de moduler les récepteurs de l'ecdysone en général (ce qui permet de contrôler la croissance des insectes), et en particulier les récepteurs de l'ecdysone de la calliphore australienne, Lucilia cuprina, et du pou du mouton, Bovicola ovis. L'invention a également trait à de nouvelles ?-méthylène ?-lactames N-substituées. Lesdits composés sont utiles en tant qu'insecticides ou en tant que têtes de série permettant l'élaboration d'insecticides. Les composés sont également utiles en tant qu'effecteurs pour les commutateurs de l'ecdysone.</description><language>eng ; fre</language><subject>AGRICULTURE ; ANIMAL HUSBANDRY ; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES ; CHEMISTRY ; FISHING ; FORESTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HUNTING ; METALLURGY ; ORGANIC CHEMISTRY ; PEST REPELLANTS OR ATTRACTANTS ; PLANT GROWTH REGULATORS ; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF ; TRAPPING</subject><creationdate>2008</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20080619&DB=EPODOC&CC=WO&NR=2008070934A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76516</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20080619&DB=EPODOC&CC=WO&NR=2008070934A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>LIEPA, ANDRIS JURIS</creatorcontrib><creatorcontrib>TURNER, KATHLEEN ANNE</creatorcontrib><creatorcontrib>JOHNSON, WYNONA MARGUERITE</creatorcontrib><title>INHIBITION OF INVERTEBRATES USING LIGANDS THAT MODULATE ECDYSONE RECEPTORS</title><description>The present invention relates to the use of N-substituted ?-methylene ?-lactams as non- steroidal ligands for modulating ecdysone receptors generally (resulting in controlled insect growth) and, in particular, ecdysone receptors of the Australian blowfly, Lucilia cuprina and the sheep body louse Bovicola ovis. The present invention further relates to novel N-substituted ?-methylene ?-lactams. These compounds are useful as insecticides or as lead compounds for the development of insecticides. The compounds are also useful as effectors for ecdysone switches.
La présente invention concerne l'utilisation de ?-méthylène ?-lactames N-substituées en tant que ligands non stéroïdiens permettant de moduler les récepteurs de l'ecdysone en général (ce qui permet de contrôler la croissance des insectes), et en particulier les récepteurs de l'ecdysone de la calliphore australienne, Lucilia cuprina, et du pou du mouton, Bovicola ovis. L'invention a également trait à de nouvelles ?-méthylène ?-lactames N-substituées. Lesdits composés sont utiles en tant qu'insecticides ou en tant que têtes de série permettant l'élaboration d'insecticides. Les composés sont également utiles en tant qu'effecteurs pour les commutateurs de l'ecdysone.</description><subject>AGRICULTURE</subject><subject>ANIMAL HUSBANDRY</subject><subject>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</subject><subject>CHEMISTRY</subject><subject>FISHING</subject><subject>FORESTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HUNTING</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PEST REPELLANTS OR ATTRACTANTS</subject><subject>PLANT GROWTH REGULATORS</subject><subject>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</subject><subject>TRAPPING</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2008</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZPDy9PPwdPIM8fT3U_B3U_D0C3MNCnF1CnIMcQ1WCA329HNX8PF0d_RzCVYI8XAMUfD1dwn1AUoquDq7RAb7-7kqBLk6uwaE-AcF8zCwpiXmFKfyQmluBmU31xBnD93Ugvz41OKCxOTUvNSS-HB_IwMDCwNzA0tjE0dDY-JUAQA9py6o</recordid><startdate>20080619</startdate><enddate>20080619</enddate><creator>LIEPA, ANDRIS JURIS</creator><creator>TURNER, KATHLEEN ANNE</creator><creator>JOHNSON, WYNONA MARGUERITE</creator><scope>EVB</scope></search><sort><creationdate>20080619</creationdate><title>INHIBITION OF INVERTEBRATES USING LIGANDS THAT MODULATE ECDYSONE RECEPTORS</title><author>LIEPA, ANDRIS JURIS ; TURNER, KATHLEEN ANNE ; JOHNSON, WYNONA MARGUERITE</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2008070934A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2008</creationdate><topic>AGRICULTURE</topic><topic>ANIMAL HUSBANDRY</topic><topic>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</topic><topic>CHEMISTRY</topic><topic>FISHING</topic><topic>FORESTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HUNTING</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PEST REPELLANTS OR ATTRACTANTS</topic><topic>PLANT GROWTH REGULATORS</topic><topic>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</topic><topic>TRAPPING</topic><toplevel>online_resources</toplevel><creatorcontrib>LIEPA, ANDRIS JURIS</creatorcontrib><creatorcontrib>TURNER, KATHLEEN ANNE</creatorcontrib><creatorcontrib>JOHNSON, WYNONA MARGUERITE</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>LIEPA, ANDRIS JURIS</au><au>TURNER, KATHLEEN ANNE</au><au>JOHNSON, WYNONA MARGUERITE</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>INHIBITION OF INVERTEBRATES USING LIGANDS THAT MODULATE ECDYSONE RECEPTORS</title><date>2008-06-19</date><risdate>2008</risdate><abstract>The present invention relates to the use of N-substituted ?-methylene ?-lactams as non- steroidal ligands for modulating ecdysone receptors generally (resulting in controlled insect growth) and, in particular, ecdysone receptors of the Australian blowfly, Lucilia cuprina and the sheep body louse Bovicola ovis. The present invention further relates to novel N-substituted ?-methylene ?-lactams. These compounds are useful as insecticides or as lead compounds for the development of insecticides. The compounds are also useful as effectors for ecdysone switches.
La présente invention concerne l'utilisation de ?-méthylène ?-lactames N-substituées en tant que ligands non stéroïdiens permettant de moduler les récepteurs de l'ecdysone en général (ce qui permet de contrôler la croissance des insectes), et en particulier les récepteurs de l'ecdysone de la calliphore australienne, Lucilia cuprina, et du pou du mouton, Bovicola ovis. L'invention a également trait à de nouvelles ?-méthylène ?-lactames N-substituées. Lesdits composés sont utiles en tant qu'insecticides ou en tant que têtes de série permettant l'élaboration d'insecticides. Les composés sont également utiles en tant qu'effecteurs pour les commutateurs de l'ecdysone.</abstract><oa>free_for_read</oa></addata></record> |
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subjects | AGRICULTURE ANIMAL HUSBANDRY BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES CHEMISTRY FISHING FORESTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HUNTING METALLURGY ORGANIC CHEMISTRY PEST REPELLANTS OR ATTRACTANTS PLANT GROWTH REGULATORS PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF TRAPPING |
title | INHIBITION OF INVERTEBRATES USING LIGANDS THAT MODULATE ECDYSONE RECEPTORS |
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