A PROCESS FOR THE PREPARATION OF EZETIMIBE VIA A NOVEL INTERMEDIATE

The present invention relates to a process for the preparation of Ezetimibe via a novel intermediate. Trans-3(R)-(3-[2-oxo-4(S)-(4-benzyloxyphenyl)-1-(4-fluorophenyl)-azetidinyl]propanoic acid is converted to trans-N-methoxy-N-methyl-3(R)-3-[2-oxo-4(S)-(4-benzyloxyphenyl)-1-(4-fluorophenyl)-azetidin...

Ausführliche Beschreibung

Bibliographische Detailangaben

Hauptverfasser:	SHRIGADI, NILESH, BALKRISHNA, PRABHAVALKAR, TIRTHA, SURESH, THORAT, AMOL, NARAYAN, RAMAKRISHNAN, ARUL
Format:	Patent
Sprache:	eng ; fre
Schlagworte:	CHEMISTRY HETEROCYCLIC COMPOUNDS METALLURGY ORGANIC CHEMISTRY
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