PYRIDINYLAMINES

Described are pyridinylamines and pharmaceutically acceptable salts thereof, the use of these pyridinylamines for the prophylaxis and/or treatment of various diseases such as infectious diseases, including opportunistic infections, prion diseases, immunological diseases, autoimmune diseases, bipolar...

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Hauptverfasser: SAVIC, VLADIMIR, EICKHOFF, JAN, EIKE, LE, JOELLE, COTTON, MATTHEW, SHERBORNE, BRAD, ZECH, BIRGIT, HARRIS, JOHN, SCHWAB, WILFRIED, KLEBL, BERT, MATTHIAS, HAFENBRADL, DORIS, MUELLER, STEFAN, MACRITCHIE, JACKIE
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creator SAVIC, VLADIMIR
EICKHOFF, JAN, EIKE
LE, JOELLE
COTTON, MATTHEW
SHERBORNE, BRAD
ZECH, BIRGIT
HARRIS, JOHN
SCHWAB, WILFRIED
KLEBL, BERT, MATTHIAS
HAFENBRADL, DORIS
MUELLER, STEFAN
MACRITCHIE, JACKIE
description Described are pyridinylamines and pharmaceutically acceptable salts thereof, the use of these pyridinylamines for the prophylaxis and/or treatment of various diseases such as infectious diseases, including opportunistic infections, prion diseases, immunological diseases, autoimmune diseases, bipolar and clinical disorders, cardiovascular diseases, cell proliferative diseases, diabetes, inflammation, transplant rejections, erectile dysfunction, neurodegenerative diseases and stroke, as well as pharmaceutical compositions containing at least one pyridinylamine and/or pharmaceutically acceptable salts thereof. Furthermore, reaction procedures for the synthesis of the pyridinylamines are disclosed. La présente invention a trait à des pyridinylamines et leurs sels pharmaceutiquement acceptables, l'utilisation de ces pyridinylamines pour la prophylaxie et/ou le traitement de diverses maladies telles que des maladies infectieuses, comprenant des infections opportunistes, des maladies à prion, des maladies immunologiques, des maladies auto-immunes, des troubles bipolaires et cliniques, des maladies cardio-vasculaires, des maladies de prolifération cellulaire, le diabète, l'inflammation, les rejets de transplantation, le dysfonctionnement érectile, les maladies neurodégénératives et l'accident vasculaire cérébral, ainsi qu'à des compositions pharmaceutiques contenant au moins une pyridinylamine et/ou des sels acceptable de celle-ci. L'invention a également trait à des procédés de réaction pour la synthèse des pyridinylamines.
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Furthermore, reaction procedures for the synthesis of the pyridinylamines are disclosed. La présente invention a trait à des pyridinylamines et leurs sels pharmaceutiquement acceptables, l'utilisation de ces pyridinylamines pour la prophylaxie et/ou le traitement de diverses maladies telles que des maladies infectieuses, comprenant des infections opportunistes, des maladies à prion, des maladies immunologiques, des maladies auto-immunes, des troubles bipolaires et cliniques, des maladies cardio-vasculaires, des maladies de prolifération cellulaire, le diabète, l'inflammation, les rejets de transplantation, le dysfonctionnement érectile, les maladies neurodégénératives et l'accident vasculaire cérébral, ainsi qu'à des compositions pharmaceutiques contenant au moins une pyridinylamine et/ou des sels acceptable de celle-ci. 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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
title PYRIDINYLAMINES
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