FUNGICIDES
This invention relates to the use as plant fungicides of certain coumarin, quinolinone and benzothiinone derivatives and the corresponding thiones. It also relates to plant fungicidal compositions containing these compounds and to certain of the compounds themselves. The use as a plant fungicide of...
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| creator | MAY, LESLIE, FRANCIS DINH, PHI, MANH WORTHINGTON, PAUL, ANTHONY ASPINALL, MARY, BERNADETTE CLARKE, ERIC, DANIEL VALANCOGNE, INGRID, AURELIE WHITTINGHAM, WILLIAM, GUY |
| description | This invention relates to the use as plant fungicides of certain coumarin, quinolinone and benzothiinone derivatives and the corresponding thiones. It also relates to plant fungicidal compositions containing these compounds and to certain of the compounds themselves.
The use as a plant fungicide of a compound of the general formula (I): wherein M, L and K are independently O, S(O)n where n is 0, 1 or 2, NR5 or CHR6, provided that at least one is CHR6, that when two are O, L is CHR6 and that when two are NR5 or two or three are CHR6, the values of R5 and the values of R6 are the same or different; X is hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alkoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alkoxy, halo(C1-6)alkoxycarbonyloxy, C1-6 alkoxycarbonyl(phenyl)(C1-6)alkoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, heterocyclylcarbonyloxy, arylcarbonyl-(C1-6)alkoxy, aryl(C1-6)alkoxycarbonyl(C1-6)alkoxy, aminocarbonyloxy, mono- or di-(C1-6)alkyl-aminocarbonyloxy, C1-6 alkoxycarbonylcarbonyloxy, C1-6 alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, heterocyclylsulphonyloxy, di-(C1-4)alkoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alkoxy, carboxy(C1-6)alkoxy, carboxyhalo(C1-6)alkoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonylhalo(C1-6)alkoxy, aminocarbonyl-(C1-6)alkoxy, mono- or di-(C1-6)alkylaminocarbonyl(C1-6)alkoxy, hydrazinocarbonyl-(C1-6)alkoxy, amino, C1-6 alkylcarbonylamino, C1-6 alkoxycarbonylamino or C1-6 alkylsulphonylamino or X may be H when R4 is hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6 alkylcarbonylamino or C1-6 alkylsulphonylamino; Y is O, S or NR7; Z is O or S; R1, R2 and R3 are independently H, halo, hydroxy, C1-14alkyl, halo(C1-8)alkyl, hydroxy(C1-8)alkyl, C1-8alkoxy, halo(C1-8)alkoxy, C1-6 alkoxy(C1-6)alkoxy, C1-6alkoxy(C1-6)alkoxy(C1-6)alkoxy, cyclo(C3-6)alkyl, C1-4alkyl-cyclo(C3-6)alkyl, cyclo(C3-6)-alkoxy, C2-6alkenyl, C2-12alkenyloxy, C2-6alkynyl, C2-6 alkynyloxy, C1-6alkoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyl, C1-6alkoxy-carbonyl(C1-8)alkyl, C1-6alkoxycarbonyl(C1-8)alkoxy, carboxy(C1-6)alkoxy, cyano, nitro, aryl, heterocyclyl, aryloxy, heterocyclyloxy, aryl(C1-10)alkyl or heterocyclyl-(C1-4)alkyl, or R1 and R2 or R2 and R3 join to form optionally C1-6 alkyl substituted C2-4 alkylenedioxy; R4 and R6 are independently H, hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_WO0228183A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>WO0228183A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_WO0228183A13</originalsourceid><addsrcrecordid>eNrjZOByC_Vz93T2dHEN5mFgTUvMKU7lhdLcDApuriHOHrqpBfnxqcUFicmpeakl8eH-BkZGFoYWxo6GxkQoAQAn5BuM</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>FUNGICIDES</title><source>esp@cenet</source><creator>MAY, LESLIE, FRANCIS ; DINH, PHI, MANH ; WORTHINGTON, PAUL, ANTHONY ; ASPINALL, MARY, BERNADETTE ; CLARKE, ERIC, DANIEL ; VALANCOGNE, INGRID, AURELIE ; WHITTINGHAM, WILLIAM, GUY</creator><creatorcontrib>MAY, LESLIE, FRANCIS ; DINH, PHI, MANH ; WORTHINGTON, PAUL, ANTHONY ; ASPINALL, MARY, BERNADETTE ; CLARKE, ERIC, DANIEL ; VALANCOGNE, INGRID, AURELIE ; WHITTINGHAM, WILLIAM, GUY</creatorcontrib><description>This invention relates to the use as plant fungicides of certain coumarin, quinolinone and benzothiinone derivatives and the corresponding thiones. It also relates to plant fungicidal compositions containing these compounds and to certain of the compounds themselves.
The use as a plant fungicide of a compound of the general formula (I): wherein M, L and K are independently O, S(O)n where n is 0, 1 or 2, NR5 or CHR6, provided that at least one is CHR6, that when two are O, L is CHR6 and that when two are NR5 or two or three are CHR6, the values of R5 and the values of R6 are the same or different; X is hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alkoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alkoxy, halo(C1-6)alkoxycarbonyloxy, C1-6 alkoxycarbonyl(phenyl)(C1-6)alkoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, heterocyclylcarbonyloxy, arylcarbonyl-(C1-6)alkoxy, aryl(C1-6)alkoxycarbonyl(C1-6)alkoxy, aminocarbonyloxy, mono- or di-(C1-6)alkyl-aminocarbonyloxy, C1-6 alkoxycarbonylcarbonyloxy, C1-6 alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, heterocyclylsulphonyloxy, di-(C1-4)alkoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alkoxy, carboxy(C1-6)alkoxy, carboxyhalo(C1-6)alkoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonylhalo(C1-6)alkoxy, aminocarbonyl-(C1-6)alkoxy, mono- or di-(C1-6)alkylaminocarbonyl(C1-6)alkoxy, hydrazinocarbonyl-(C1-6)alkoxy, amino, C1-6 alkylcarbonylamino, C1-6 alkoxycarbonylamino or C1-6 alkylsulphonylamino or X may be H when R4 is hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6 alkylcarbonylamino or C1-6 alkylsulphonylamino; Y is O, S or NR7; Z is O or S; R1, R2 and R3 are independently H, halo, hydroxy, C1-14alkyl, halo(C1-8)alkyl, hydroxy(C1-8)alkyl, C1-8alkoxy, halo(C1-8)alkoxy, C1-6 alkoxy(C1-6)alkoxy, C1-6alkoxy(C1-6)alkoxy(C1-6)alkoxy, cyclo(C3-6)alkyl, C1-4alkyl-cyclo(C3-6)alkyl, cyclo(C3-6)-alkoxy, C2-6alkenyl, C2-12alkenyloxy, C2-6alkynyl, C2-6 alkynyloxy, C1-6alkoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyl, C1-6alkoxy-carbonyl(C1-8)alkyl, C1-6alkoxycarbonyl(C1-8)alkoxy, carboxy(C1-6)alkoxy, cyano, nitro, aryl, heterocyclyl, aryloxy, heterocyclyloxy, aryl(C1-10)alkyl or heterocyclyl-(C1-4)alkyl, or R1 and R2 or R2 and R3 join to form optionally C1-6 alkyl substituted C2-4 alkylenedioxy; R4 and R6 are independently H, hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, C1-6alkylsulphonylamino, C1-6 alkyl, C1-6 alkoxy, C2-4 alkylenedioxy, cyclo(C3-6)alkyl, cyclo(C3-6)alkoxy, C2-6 alkenyl, C2-6 alkenyloxy, C2-6 alkynyl, C2-6 alkynyloxy, C1-4 alkylcarbonyloxy, aryl, heterocyclyl, aryloxy or heterocyclyloxy; and R5 and R7 are independently H, an acid addition salt, C1-6 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 alkylcarbonyl, C2-4 alkenylcarbonyl, aryl, aryl(C1-4)-alkyl, arylcarbonyl, C1-4alkylsulphonyl or arylsulphonyl; any of the foregoing aryl, heterocyclyl, cycloalkyl and cycloalkoxy groups or moieties being optionally substituted. The invention also includes a plant fungicidal composition containing the compound (I), a method of combating or controlling phytopathogenic fungi using compound (I) or a composition thereof and certain compounds per se.
L'invention concerne l'utilisation comme fongicide pour plante d'un composé représenté par la formule générale (I). Dans ladite formule, M, L et K sont indépendamment O, S(O)n, n valant 0, 1 ou 2, NR5 ou CHR6, à condition qu'au moins l'un d'entre eux soit CHR6, que lorsque deux d'entre eux sont O, L soit CHR6, et que lorsque deux d'entre eux sont NR5 ou bien deux ou trois d'entre eux sont CHR6, les valeurs de R5 et celles de R6 soient identiques ou différentes; X est hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alcoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alcoxy, halo(C1-6)alcoxycarbonyloxy, C1-6 alcoxycarbonyl(phényl)(C1-6)alcoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, hétérocyclylcarbonyloxy, arylcarbonyl-(C1-6)alcoxy, aryl(C1-6)alcoxycarbonyl(C1-6)alcoxy, aminocarbonyloxy, mono- ou di-(C1-6)alkyl-aminocarbonyloxy, C1-6alkoxycarbonylcarbonyloxy, C1-6alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, hétérocyclylsulphonyloxy, di-(C1-4)alcoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alcoxy, carboxy(C1-6)alcoxy, carboxyhalo(C1-6)alcoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alcoxycarbonyl(C1-6)alcoxy, C1-6 alcoxycarbonylhalo(C1-6) alcoxy, aminocarbonyl-(C1-6) alkoxy, mono- ou di-(C1-6) alkylaminocarbonyl(C1-6)alcoxy, hydrazinocarbonyl-(C1-6)alcoxy, amino, C1-6 alkylcarbonylamino, C1-6alcoxycarbonylamino ou C1-6alkylsulphonylamino ou X peut être H lorsque R4 est hydroxy, oxo, hydroximino, amino, mono-ou-di-(C1-6)alkylamino, C1-6alkylcarbonylamino ou C1-6alkylsulphonylamino; Y est O, S ou NR7; Z est O ou S; R1, R2 et R3 sont indépendamment H, halo, hydroxy, C1-14alkyle, halo(C1-8)alkyle, hydroxy(C1-8)alkyle, C1-8alcoxy, halo(C1-8) alcoxy, C1-6 alkoxy(C1-6)alcoxy, C1-6alcoxy(C1-6)alcoxy(C1-6)alcoxy, cyclo(C3-6)alkyle, C1-4alkyl-cyclo(C3-6)alkyle, cyclo(C3-6)-alcoxy, C2-6alcényle, C2-12alcényloxy, C2-6alkynyle, C2-6 alkynyloxy, C1-6alcoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyle, C1-6alcoxy-carbonyl(C1-8)alkyle, C1-6alcoxycarbonyl(C1-8)alcoxy, carboxy(C1-6)alcoxy, cyano, nitro, aryle, hétérocyclyle, aryloxy, hétérocyclyloxy, aryl(C1-10)alkyle ou hétérocyclyl-(C1-4)alkyle, ou R1 et R2 ou R2 et R3 s'unissent pour former éventuellement C2-4alkylènedioxy à substitution C1-6; R4 et R6 sont indépendamment H, hydroxy, oxo, hydroximino, amino, mono-ou-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, C1-6alkylsulphonylamino, C1-6alkyle, C1-6 alcoxy, C2-4 alkylènedioxy, cyclo(C3-6)alkyle, cyclo(C3-6)alcoxy, C2-6 alcényle, C2-6 alcényloxy, C2-6 e, C2-6 alkynyloxy, C1-4 alkylcarbonyloxy, aryle hétérocyclyle, aryloxy ou hétérocyclyloxy; et R5 et R7 sont indépendamment H, un sel d'addition acide, C1-6alkyle, C2-4 alcényle, C2-4 alkynyle, C1-4 alkylcarbonyle, C2-4 alcénylcarbonyle, aryle, aryl(C1-4)-alkyle, arylcarbonyle, C1-4alkylsulphonyle ou arylsulphonyle; l'un ou l'une quelconque des groupes ou fractions aryle, hétérocyclyle, cycloalkyle et cycloalkoxy sont à substitution éventuelle. L'invention concerne également une composition fongicide pour plante renfermant le composé (I), un procédé visant à combattre ou à contrôler les champignons phythopathogènes en utilisant le composé (I) ou une composition de ce composé et certains composés per se.</description><edition>7</edition><language>eng ; fre</language><subject>AGRICULTURE ; ANIMAL HUSBANDRY ; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES ; FISHING ; FORESTRY ; HUMAN NECESSITIES ; HUNTING ; PEST REPELLANTS OR ATTRACTANTS ; PLANT GROWTH REGULATORS ; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF ; TRAPPING</subject><creationdate>2002</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20020411&DB=EPODOC&CC=WO&NR=0228183A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,778,883,25547,76298</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20020411&DB=EPODOC&CC=WO&NR=0228183A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>MAY, LESLIE, FRANCIS</creatorcontrib><creatorcontrib>DINH, PHI, MANH</creatorcontrib><creatorcontrib>WORTHINGTON, PAUL, ANTHONY</creatorcontrib><creatorcontrib>ASPINALL, MARY, BERNADETTE</creatorcontrib><creatorcontrib>CLARKE, ERIC, DANIEL</creatorcontrib><creatorcontrib>VALANCOGNE, INGRID, AURELIE</creatorcontrib><creatorcontrib>WHITTINGHAM, WILLIAM, GUY</creatorcontrib><title>FUNGICIDES</title><description>This invention relates to the use as plant fungicides of certain coumarin, quinolinone and benzothiinone derivatives and the corresponding thiones. It also relates to plant fungicidal compositions containing these compounds and to certain of the compounds themselves.
The use as a plant fungicide of a compound of the general formula (I): wherein M, L and K are independently O, S(O)n where n is 0, 1 or 2, NR5 or CHR6, provided that at least one is CHR6, that when two are O, L is CHR6 and that when two are NR5 or two or three are CHR6, the values of R5 and the values of R6 are the same or different; X is hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alkoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alkoxy, halo(C1-6)alkoxycarbonyloxy, C1-6 alkoxycarbonyl(phenyl)(C1-6)alkoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, heterocyclylcarbonyloxy, arylcarbonyl-(C1-6)alkoxy, aryl(C1-6)alkoxycarbonyl(C1-6)alkoxy, aminocarbonyloxy, mono- or di-(C1-6)alkyl-aminocarbonyloxy, C1-6 alkoxycarbonylcarbonyloxy, C1-6 alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, heterocyclylsulphonyloxy, di-(C1-4)alkoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alkoxy, carboxy(C1-6)alkoxy, carboxyhalo(C1-6)alkoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonylhalo(C1-6)alkoxy, aminocarbonyl-(C1-6)alkoxy, mono- or di-(C1-6)alkylaminocarbonyl(C1-6)alkoxy, hydrazinocarbonyl-(C1-6)alkoxy, amino, C1-6 alkylcarbonylamino, C1-6 alkoxycarbonylamino or C1-6 alkylsulphonylamino or X may be H when R4 is hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6 alkylcarbonylamino or C1-6 alkylsulphonylamino; Y is O, S or NR7; Z is O or S; R1, R2 and R3 are independently H, halo, hydroxy, C1-14alkyl, halo(C1-8)alkyl, hydroxy(C1-8)alkyl, C1-8alkoxy, halo(C1-8)alkoxy, C1-6 alkoxy(C1-6)alkoxy, C1-6alkoxy(C1-6)alkoxy(C1-6)alkoxy, cyclo(C3-6)alkyl, C1-4alkyl-cyclo(C3-6)alkyl, cyclo(C3-6)-alkoxy, C2-6alkenyl, C2-12alkenyloxy, C2-6alkynyl, C2-6 alkynyloxy, C1-6alkoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyl, C1-6alkoxy-carbonyl(C1-8)alkyl, C1-6alkoxycarbonyl(C1-8)alkoxy, carboxy(C1-6)alkoxy, cyano, nitro, aryl, heterocyclyl, aryloxy, heterocyclyloxy, aryl(C1-10)alkyl or heterocyclyl-(C1-4)alkyl, or R1 and R2 or R2 and R3 join to form optionally C1-6 alkyl substituted C2-4 alkylenedioxy; R4 and R6 are independently H, hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, C1-6alkylsulphonylamino, C1-6 alkyl, C1-6 alkoxy, C2-4 alkylenedioxy, cyclo(C3-6)alkyl, cyclo(C3-6)alkoxy, C2-6 alkenyl, C2-6 alkenyloxy, C2-6 alkynyl, C2-6 alkynyloxy, C1-4 alkylcarbonyloxy, aryl, heterocyclyl, aryloxy or heterocyclyloxy; and R5 and R7 are independently H, an acid addition salt, C1-6 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 alkylcarbonyl, C2-4 alkenylcarbonyl, aryl, aryl(C1-4)-alkyl, arylcarbonyl, C1-4alkylsulphonyl or arylsulphonyl; any of the foregoing aryl, heterocyclyl, cycloalkyl and cycloalkoxy groups or moieties being optionally substituted. The invention also includes a plant fungicidal composition containing the compound (I), a method of combating or controlling phytopathogenic fungi using compound (I) or a composition thereof and certain compounds per se.
L'invention concerne l'utilisation comme fongicide pour plante d'un composé représenté par la formule générale (I). Dans ladite formule, M, L et K sont indépendamment O, S(O)n, n valant 0, 1 ou 2, NR5 ou CHR6, à condition qu'au moins l'un d'entre eux soit CHR6, que lorsque deux d'entre eux sont O, L soit CHR6, et que lorsque deux d'entre eux sont NR5 ou bien deux ou trois d'entre eux sont CHR6, les valeurs de R5 et celles de R6 soient identiques ou différentes; X est hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alcoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alcoxy, halo(C1-6)alcoxycarbonyloxy, C1-6 alcoxycarbonyl(phényl)(C1-6)alcoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, hétérocyclylcarbonyloxy, arylcarbonyl-(C1-6)alcoxy, aryl(C1-6)alcoxycarbonyl(C1-6)alcoxy, aminocarbonyloxy, mono- ou di-(C1-6)alkyl-aminocarbonyloxy, C1-6alkoxycarbonylcarbonyloxy, C1-6alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, hétérocyclylsulphonyloxy, di-(C1-4)alcoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alcoxy, carboxy(C1-6)alcoxy, carboxyhalo(C1-6)alcoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alcoxycarbonyl(C1-6)alcoxy, C1-6 alcoxycarbonylhalo(C1-6) alcoxy, aminocarbonyl-(C1-6) alkoxy, mono- ou di-(C1-6) alkylaminocarbonyl(C1-6)alcoxy, hydrazinocarbonyl-(C1-6)alcoxy, amino, C1-6 alkylcarbonylamino, C1-6alcoxycarbonylamino ou C1-6alkylsulphonylamino ou X peut être H lorsque R4 est hydroxy, oxo, hydroximino, amino, mono-ou-di-(C1-6)alkylamino, C1-6alkylcarbonylamino ou C1-6alkylsulphonylamino; Y est O, S ou NR7; Z est O ou S; R1, R2 et R3 sont indépendamment H, halo, hydroxy, C1-14alkyle, halo(C1-8)alkyle, hydroxy(C1-8)alkyle, C1-8alcoxy, halo(C1-8) alcoxy, C1-6 alkoxy(C1-6)alcoxy, C1-6alcoxy(C1-6)alcoxy(C1-6)alcoxy, cyclo(C3-6)alkyle, C1-4alkyl-cyclo(C3-6)alkyle, cyclo(C3-6)-alcoxy, C2-6alcényle, C2-12alcényloxy, C2-6alkynyle, C2-6 alkynyloxy, C1-6alcoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyle, C1-6alcoxy-carbonyl(C1-8)alkyle, C1-6alcoxycarbonyl(C1-8)alcoxy, carboxy(C1-6)alcoxy, cyano, nitro, aryle, hétérocyclyle, aryloxy, hétérocyclyloxy, aryl(C1-10)alkyle ou hétérocyclyl-(C1-4)alkyle, ou R1 et R2 ou R2 et R3 s'unissent pour former éventuellement C2-4alkylènedioxy à substitution C1-6; R4 et R6 sont indépendamment H, hydroxy, oxo, hydroximino, amino, mono-ou-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, C1-6alkylsulphonylamino, C1-6alkyle, C1-6 alcoxy, C2-4 alkylènedioxy, cyclo(C3-6)alkyle, cyclo(C3-6)alcoxy, C2-6 alcényle, C2-6 alcényloxy, C2-6 e, C2-6 alkynyloxy, C1-4 alkylcarbonyloxy, aryle hétérocyclyle, aryloxy ou hétérocyclyloxy; et R5 et R7 sont indépendamment H, un sel d'addition acide, C1-6alkyle, C2-4 alcényle, C2-4 alkynyle, C1-4 alkylcarbonyle, C2-4 alcénylcarbonyle, aryle, aryl(C1-4)-alkyle, arylcarbonyle, C1-4alkylsulphonyle ou arylsulphonyle; l'un ou l'une quelconque des groupes ou fractions aryle, hétérocyclyle, cycloalkyle et cycloalkoxy sont à substitution éventuelle. L'invention concerne également une composition fongicide pour plante renfermant le composé (I), un procédé visant à combattre ou à contrôler les champignons phythopathogènes en utilisant le composé (I) ou une composition de ce composé et certains composés per se.</description><subject>AGRICULTURE</subject><subject>ANIMAL HUSBANDRY</subject><subject>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</subject><subject>FISHING</subject><subject>FORESTRY</subject><subject>HUMAN NECESSITIES</subject><subject>HUNTING</subject><subject>PEST REPELLANTS OR ATTRACTANTS</subject><subject>PLANT GROWTH REGULATORS</subject><subject>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</subject><subject>TRAPPING</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2002</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZOByC_Vz93T2dHEN5mFgTUvMKU7lhdLcDApuriHOHrqpBfnxqcUFicmpeakl8eH-BkZGFoYWxo6GxkQoAQAn5BuM</recordid><startdate>20020411</startdate><enddate>20020411</enddate><creator>MAY, LESLIE, FRANCIS</creator><creator>DINH, PHI, MANH</creator><creator>WORTHINGTON, PAUL, ANTHONY</creator><creator>ASPINALL, MARY, BERNADETTE</creator><creator>CLARKE, ERIC, DANIEL</creator><creator>VALANCOGNE, INGRID, AURELIE</creator><creator>WHITTINGHAM, WILLIAM, GUY</creator><scope>EVB</scope></search><sort><creationdate>20020411</creationdate><title>FUNGICIDES</title><author>MAY, LESLIE, FRANCIS ; DINH, PHI, MANH ; WORTHINGTON, PAUL, ANTHONY ; ASPINALL, MARY, BERNADETTE ; CLARKE, ERIC, DANIEL ; VALANCOGNE, INGRID, AURELIE ; WHITTINGHAM, WILLIAM, GUY</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO0228183A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2002</creationdate><topic>AGRICULTURE</topic><topic>ANIMAL HUSBANDRY</topic><topic>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</topic><topic>FISHING</topic><topic>FORESTRY</topic><topic>HUMAN NECESSITIES</topic><topic>HUNTING</topic><topic>PEST REPELLANTS OR ATTRACTANTS</topic><topic>PLANT GROWTH REGULATORS</topic><topic>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</topic><topic>TRAPPING</topic><toplevel>online_resources</toplevel><creatorcontrib>MAY, LESLIE, FRANCIS</creatorcontrib><creatorcontrib>DINH, PHI, MANH</creatorcontrib><creatorcontrib>WORTHINGTON, PAUL, ANTHONY</creatorcontrib><creatorcontrib>ASPINALL, MARY, BERNADETTE</creatorcontrib><creatorcontrib>CLARKE, ERIC, DANIEL</creatorcontrib><creatorcontrib>VALANCOGNE, INGRID, AURELIE</creatorcontrib><creatorcontrib>WHITTINGHAM, WILLIAM, GUY</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>MAY, LESLIE, FRANCIS</au><au>DINH, PHI, MANH</au><au>WORTHINGTON, PAUL, ANTHONY</au><au>ASPINALL, MARY, BERNADETTE</au><au>CLARKE, ERIC, DANIEL</au><au>VALANCOGNE, INGRID, AURELIE</au><au>WHITTINGHAM, WILLIAM, GUY</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>FUNGICIDES</title><date>2002-04-11</date><risdate>2002</risdate><abstract>This invention relates to the use as plant fungicides of certain coumarin, quinolinone and benzothiinone derivatives and the corresponding thiones. It also relates to plant fungicidal compositions containing these compounds and to certain of the compounds themselves.
The use as a plant fungicide of a compound of the general formula (I): wherein M, L and K are independently O, S(O)n where n is 0, 1 or 2, NR5 or CHR6, provided that at least one is CHR6, that when two are O, L is CHR6 and that when two are NR5 or two or three are CHR6, the values of R5 and the values of R6 are the same or different; X is hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alkoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alkoxy, halo(C1-6)alkoxycarbonyloxy, C1-6 alkoxycarbonyl(phenyl)(C1-6)alkoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, heterocyclylcarbonyloxy, arylcarbonyl-(C1-6)alkoxy, aryl(C1-6)alkoxycarbonyl(C1-6)alkoxy, aminocarbonyloxy, mono- or di-(C1-6)alkyl-aminocarbonyloxy, C1-6 alkoxycarbonylcarbonyloxy, C1-6 alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, heterocyclylsulphonyloxy, di-(C1-4)alkoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alkoxy, carboxy(C1-6)alkoxy, carboxyhalo(C1-6)alkoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonyl(C1-6)alkoxy, C1-6 alkoxycarbonylhalo(C1-6)alkoxy, aminocarbonyl-(C1-6)alkoxy, mono- or di-(C1-6)alkylaminocarbonyl(C1-6)alkoxy, hydrazinocarbonyl-(C1-6)alkoxy, amino, C1-6 alkylcarbonylamino, C1-6 alkoxycarbonylamino or C1-6 alkylsulphonylamino or X may be H when R4 is hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6 alkylcarbonylamino or C1-6 alkylsulphonylamino; Y is O, S or NR7; Z is O or S; R1, R2 and R3 are independently H, halo, hydroxy, C1-14alkyl, halo(C1-8)alkyl, hydroxy(C1-8)alkyl, C1-8alkoxy, halo(C1-8)alkoxy, C1-6 alkoxy(C1-6)alkoxy, C1-6alkoxy(C1-6)alkoxy(C1-6)alkoxy, cyclo(C3-6)alkyl, C1-4alkyl-cyclo(C3-6)alkyl, cyclo(C3-6)-alkoxy, C2-6alkenyl, C2-12alkenyloxy, C2-6alkynyl, C2-6 alkynyloxy, C1-6alkoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyl, C1-6alkoxy-carbonyl(C1-8)alkyl, C1-6alkoxycarbonyl(C1-8)alkoxy, carboxy(C1-6)alkoxy, cyano, nitro, aryl, heterocyclyl, aryloxy, heterocyclyloxy, aryl(C1-10)alkyl or heterocyclyl-(C1-4)alkyl, or R1 and R2 or R2 and R3 join to form optionally C1-6 alkyl substituted C2-4 alkylenedioxy; R4 and R6 are independently H, hydroxy, oxo, hydroximino, amino, mono-or-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, C1-6alkylsulphonylamino, C1-6 alkyl, C1-6 alkoxy, C2-4 alkylenedioxy, cyclo(C3-6)alkyl, cyclo(C3-6)alkoxy, C2-6 alkenyl, C2-6 alkenyloxy, C2-6 alkynyl, C2-6 alkynyloxy, C1-4 alkylcarbonyloxy, aryl, heterocyclyl, aryloxy or heterocyclyloxy; and R5 and R7 are independently H, an acid addition salt, C1-6 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 alkylcarbonyl, C2-4 alkenylcarbonyl, aryl, aryl(C1-4)-alkyl, arylcarbonyl, C1-4alkylsulphonyl or arylsulphonyl; any of the foregoing aryl, heterocyclyl, cycloalkyl and cycloalkoxy groups or moieties being optionally substituted. The invention also includes a plant fungicidal composition containing the compound (I), a method of combating or controlling phytopathogenic fungi using compound (I) or a composition thereof and certain compounds per se.
L'invention concerne l'utilisation comme fongicide pour plante d'un composé représenté par la formule générale (I). Dans ladite formule, M, L et K sont indépendamment O, S(O)n, n valant 0, 1 ou 2, NR5 ou CHR6, à condition qu'au moins l'un d'entre eux soit CHR6, que lorsque deux d'entre eux sont O, L soit CHR6, et que lorsque deux d'entre eux sont NR5 ou bien deux ou trois d'entre eux sont CHR6, les valeurs de R5 et celles de R6 soient identiques ou différentes; X est hydroxy, cyclohexanon-2-yloxy, C1-6 alkylcarbonyloxy, halo (C1-6)-alkylcarbonyloxy, C1-6 alcoxycarbonyloxy, C1-6 alkoxycarbonyl (C1-6) alcoxy, halo(C1-6)alcoxycarbonyloxy, C1-6 alcoxycarbonyl(phényl)(C1-6)alcoxy, cyclo(C3-6)-alkylcarbonyloxy, arylcarbonyloxy, hétérocyclylcarbonyloxy, arylcarbonyl-(C1-6)alcoxy, aryl(C1-6)alcoxycarbonyl(C1-6)alcoxy, aminocarbonyloxy, mono- ou di-(C1-6)alkyl-aminocarbonyloxy, C1-6alkoxycarbonylcarbonyloxy, C1-6alkyl-sulphonyloxy, haloalkylsulphonyloxy, arylsulphonyloxy, hétérocyclylsulphonyloxy, di-(C1-4)alcoxyphosphonyloxy, dihydroxyphosphonyloxy, cyano(C1-6)alcoxy, carboxy(C1-6)alcoxy, carboxyhalo(C1-6)alcoxy, C1-6alkylcarbonyl(C1-6)alkoxy, C1-6 alcoxycarbonyl(C1-6)alcoxy, C1-6 alcoxycarbonylhalo(C1-6) alcoxy, aminocarbonyl-(C1-6) alkoxy, mono- ou di-(C1-6) alkylaminocarbonyl(C1-6)alcoxy, hydrazinocarbonyl-(C1-6)alcoxy, amino, C1-6 alkylcarbonylamino, C1-6alcoxycarbonylamino ou C1-6alkylsulphonylamino ou X peut être H lorsque R4 est hydroxy, oxo, hydroximino, amino, mono-ou-di-(C1-6)alkylamino, C1-6alkylcarbonylamino ou C1-6alkylsulphonylamino; Y est O, S ou NR7; Z est O ou S; R1, R2 et R3 sont indépendamment H, halo, hydroxy, C1-14alkyle, halo(C1-8)alkyle, hydroxy(C1-8)alkyle, C1-8alcoxy, halo(C1-8) alcoxy, C1-6 alkoxy(C1-6)alcoxy, C1-6alcoxy(C1-6)alcoxy(C1-6)alcoxy, cyclo(C3-6)alkyle, C1-4alkyl-cyclo(C3-6)alkyle, cyclo(C3-6)-alcoxy, C2-6alcényle, C2-12alcényloxy, C2-6alkynyle, C2-6 alkynyloxy, C1-6alcoxycarbonyl, C1-6alkylcarbonyloxy(C1-8)alkyle, C1-6alcoxy-carbonyl(C1-8)alkyle, C1-6alcoxycarbonyl(C1-8)alcoxy, carboxy(C1-6)alcoxy, cyano, nitro, aryle, hétérocyclyle, aryloxy, hétérocyclyloxy, aryl(C1-10)alkyle ou hétérocyclyl-(C1-4)alkyle, ou R1 et R2 ou R2 et R3 s'unissent pour former éventuellement C2-4alkylènedioxy à substitution C1-6; R4 et R6 sont indépendamment H, hydroxy, oxo, hydroximino, amino, mono-ou-di-(C1-6)alkylamino, C1-6alkylcarbonylamino, C1-6alkylsulphonylamino, C1-6alkyle, C1-6 alcoxy, C2-4 alkylènedioxy, cyclo(C3-6)alkyle, cyclo(C3-6)alcoxy, C2-6 alcényle, C2-6 alcényloxy, C2-6 e, C2-6 alkynyloxy, C1-4 alkylcarbonyloxy, aryle hétérocyclyle, aryloxy ou hétérocyclyloxy; et R5 et R7 sont indépendamment H, un sel d'addition acide, C1-6alkyle, C2-4 alcényle, C2-4 alkynyle, C1-4 alkylcarbonyle, C2-4 alcénylcarbonyle, aryle, aryl(C1-4)-alkyle, arylcarbonyle, C1-4alkylsulphonyle ou arylsulphonyle; l'un ou l'une quelconque des groupes ou fractions aryle, hétérocyclyle, cycloalkyle et cycloalkoxy sont à substitution éventuelle. L'invention concerne également une composition fongicide pour plante renfermant le composé (I), un procédé visant à combattre ou à contrôler les champignons phythopathogènes en utilisant le composé (I) ou une composition de ce composé et certains composés per se.</abstract><edition>7</edition><oa>free_for_read</oa></addata></record> |
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| language | eng ; fre |
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| subjects | AGRICULTURE ANIMAL HUSBANDRY BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES FISHING FORESTRY HUMAN NECESSITIES HUNTING PEST REPELLANTS OR ATTRACTANTS PLANT GROWTH REGULATORS PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF TRAPPING |
| title | FUNGICIDES |
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