Process for preparing combinatorial amide alcohol libraries

Combinatorial chemical libraries of the Formula [S]-C(O)-L'-Z containing dihyroxy amides and hydroxyphosphonate amides are disclosed, in which [S] represents a solid support and -L'-Z is a linker/ligand residue. In these libraries, Z isand Y is -P(O)(OR6)(OR7), -CH(OH)-COR8, -CH,CH=CH2-CH2...

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Hauptverfasser:	SHIMSHOCK YVONNE CLASS, CAVALLARO CULLEN LEE, HERPIN TIMOTHEE FELIX, DOLLE, III ROLAND ELLWOOD
Format:	Patent
Sprache:	eng
Schlagworte:	ACYCLIC OR CARBOCYCLIC COMPOUNDS APPARATUS THEREFOR CHEMISTRY COMBINATORIAL CHEMISTRY GENERAL METHODS OF ORGANIC CHEMISTRY LIBRARIES, e.g. CHEMICAL LIBRARIES, IN SILICOLIBRARIES METALLURGY ORGANIC CHEMISTRY
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creator	SHIMSHOCK YVONNE CLASS CAVALLARO CULLEN LEE HERPIN TIMOTHEE FELIX DOLLE, III ROLAND ELLWOOD
description	Combinatorial chemical libraries of the Formula [S]-C(O)-L'-Z containing dihyroxy amides and hydroxyphosphonate amides are disclosed, in which [S] represents a solid support and -L'-Z is a linker/ligand residue. In these libraries, Z isand Y is -P(O)(OR6)(OR7), -CH(OH)-COR8, -CH,CH=CH2-CH2CH(OH)CH2OH, -CH2CHO, -CH2CH2OH, -CH2CH2OC(O)NHR26, -CH2CH2NR27R28, orThe combinatorial libraries are optionally encoded with tags. The use of these libraries in assays to discover biologically active compounds is also disclosed.
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subjects	ACYCLIC OR CARBOCYCLIC COMPOUNDS APPARATUS THEREFOR CHEMISTRY COMBINATORIAL CHEMISTRY GENERAL METHODS OF ORGANIC CHEMISTRY LIBRARIES, e.g. CHEMICAL LIBRARIES, IN SILICOLIBRARIES METALLURGY ORGANIC CHEMISTRY
title	Process for preparing combinatorial amide alcohol libraries
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