Synephrine derivatives useful as anti-inflammatory agents
This invention provides compounds having the structural formula: wherein: R1 is an acyl or sulfonyl group, R2 is an acyl group selected from the group consisting of acyl groups derived from cycloaliphatic, aromatic or heterocyclic monocarboxylic acids, imidazolylcarbonyl and triazolylcarbonyl, and R...
Gespeichert in:
| Hauptverfasser: | , , , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | eng |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | CALENBERGH SERGE VAN HAEGEMAN GUY ARIAS RUBEN HOYA GERLO SARAH LACEY CARL JEFFREY GOSSYE VALERIE BERGHE WIM VANDEN BOSSCHER KAROLIEN DE |
| description | This invention provides compounds having the structural formula: wherein: R1 is an acyl or sulfonyl group, R2 is an acyl group selected from the group consisting of acyl groups derived from cycloaliphatic, aromatic or heterocyclic monocarboxylic acids, imidazolylcarbonyl and triazolylcarbonyl, and R3 is hydrogen or an amino-protecting group, a stereoisomer thereof, a solvate thereof, or a salt thereof, being useful as anti-inflammatory agents and anti-cancer agents. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_US2009029999A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>US2009029999A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_US2009029999A13</originalsourceid><addsrcrecordid>eNrjZLAMrsxLLcgoysxLVUhJLcosSyzJLEstVigtTk0rzVFILFZIzCvJ1M3MS8tJzM1NLMkvqlRITE_NKynmYWBNS8wpTuWF0twMym6uIc4euqkF-fGpxQWJyal5qSXxocFGBgaWBkaWQOBoaEycKgBYkTB3</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>Synephrine derivatives useful as anti-inflammatory agents</title><source>esp@cenet</source><creator>CALENBERGH SERGE VAN ; HAEGEMAN GUY ; ARIAS RUBEN HOYA ; GERLO SARAH ; LACEY CARL JEFFREY ; GOSSYE VALERIE ; BERGHE WIM VANDEN ; BOSSCHER KAROLIEN DE</creator><creatorcontrib>CALENBERGH SERGE VAN ; HAEGEMAN GUY ; ARIAS RUBEN HOYA ; GERLO SARAH ; LACEY CARL JEFFREY ; GOSSYE VALERIE ; BERGHE WIM VANDEN ; BOSSCHER KAROLIEN DE</creatorcontrib><description>This invention provides compounds having the structural formula: wherein: R1 is an acyl or sulfonyl group, R2 is an acyl group selected from the group consisting of acyl groups derived from cycloaliphatic, aromatic or heterocyclic monocarboxylic acids, imidazolylcarbonyl and triazolylcarbonyl, and R3 is hydrogen or an amino-protecting group, a stereoisomer thereof, a solvate thereof, or a salt thereof, being useful as anti-inflammatory agents and anti-cancer agents.</description><language>eng</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2009</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20090129&DB=EPODOC&CC=US&NR=2009029999A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20090129&DB=EPODOC&CC=US&NR=2009029999A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>CALENBERGH SERGE VAN</creatorcontrib><creatorcontrib>HAEGEMAN GUY</creatorcontrib><creatorcontrib>ARIAS RUBEN HOYA</creatorcontrib><creatorcontrib>GERLO SARAH</creatorcontrib><creatorcontrib>LACEY CARL JEFFREY</creatorcontrib><creatorcontrib>GOSSYE VALERIE</creatorcontrib><creatorcontrib>BERGHE WIM VANDEN</creatorcontrib><creatorcontrib>BOSSCHER KAROLIEN DE</creatorcontrib><title>Synephrine derivatives useful as anti-inflammatory agents</title><description>This invention provides compounds having the structural formula: wherein: R1 is an acyl or sulfonyl group, R2 is an acyl group selected from the group consisting of acyl groups derived from cycloaliphatic, aromatic or heterocyclic monocarboxylic acids, imidazolylcarbonyl and triazolylcarbonyl, and R3 is hydrogen or an amino-protecting group, a stereoisomer thereof, a solvate thereof, or a salt thereof, being useful as anti-inflammatory agents and anti-cancer agents.</description><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2009</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZLAMrsxLLcgoysxLVUhJLcosSyzJLEstVigtTk0rzVFILFZIzCvJ1M3MS8tJzM1NLMkvqlRITE_NKynmYWBNS8wpTuWF0twMym6uIc4euqkF-fGpxQWJyal5qSXxocFGBgaWBkaWQOBoaEycKgBYkTB3</recordid><startdate>20090129</startdate><enddate>20090129</enddate><creator>CALENBERGH SERGE VAN</creator><creator>HAEGEMAN GUY</creator><creator>ARIAS RUBEN HOYA</creator><creator>GERLO SARAH</creator><creator>LACEY CARL JEFFREY</creator><creator>GOSSYE VALERIE</creator><creator>BERGHE WIM VANDEN</creator><creator>BOSSCHER KAROLIEN DE</creator><scope>EVB</scope></search><sort><creationdate>20090129</creationdate><title>Synephrine derivatives useful as anti-inflammatory agents</title><author>CALENBERGH SERGE VAN ; HAEGEMAN GUY ; ARIAS RUBEN HOYA ; GERLO SARAH ; LACEY CARL JEFFREY ; GOSSYE VALERIE ; BERGHE WIM VANDEN ; BOSSCHER KAROLIEN DE</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_US2009029999A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>2009</creationdate><topic>ACYCLIC OR CARBOCYCLIC COMPOUNDS</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>CALENBERGH SERGE VAN</creatorcontrib><creatorcontrib>HAEGEMAN GUY</creatorcontrib><creatorcontrib>ARIAS RUBEN HOYA</creatorcontrib><creatorcontrib>GERLO SARAH</creatorcontrib><creatorcontrib>LACEY CARL JEFFREY</creatorcontrib><creatorcontrib>GOSSYE VALERIE</creatorcontrib><creatorcontrib>BERGHE WIM VANDEN</creatorcontrib><creatorcontrib>BOSSCHER KAROLIEN DE</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>CALENBERGH SERGE VAN</au><au>HAEGEMAN GUY</au><au>ARIAS RUBEN HOYA</au><au>GERLO SARAH</au><au>LACEY CARL JEFFREY</au><au>GOSSYE VALERIE</au><au>BERGHE WIM VANDEN</au><au>BOSSCHER KAROLIEN DE</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>Synephrine derivatives useful as anti-inflammatory agents</title><date>2009-01-29</date><risdate>2009</risdate><abstract>This invention provides compounds having the structural formula: wherein: R1 is an acyl or sulfonyl group, R2 is an acyl group selected from the group consisting of acyl groups derived from cycloaliphatic, aromatic or heterocyclic monocarboxylic acids, imidazolylcarbonyl and triazolylcarbonyl, and R3 is hydrogen or an amino-protecting group, a stereoisomer thereof, a solvate thereof, or a salt thereof, being useful as anti-inflammatory agents and anti-cancer agents.</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | eng |
| recordid | cdi_epo_espacenet_US2009029999A1 |
| source | esp@cenet |
| subjects | ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | Synephrine derivatives useful as anti-inflammatory agents |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-02T19%3A18%3A35IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=CALENBERGH%20SERGE%20VAN&rft.date=2009-01-29&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EUS2009029999A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |