Benzimidazole derivatives and their use as protein kinases inhibitors

The invention provides compounds of the formula (1): The compounds have activity against cyclin depdenent kinases, glycogen synthase kinase and Auroa kinases and are therefore useful to treat cancer and viral diseases.

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: TREWARTHA GARY, NAVARRO EVA F, HOWARD STEVEN, WOOLFORD ALISON J, GILL ADRIAN L, EARLY THERESA R, WYATT PAUL, O'BRIEN MICHAEL A, CARR MARIA G, BERDINI VALERIO, WOODHEAD ANDREW J
Format: Patent
Sprache:eng
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
container_end_page
container_issue
container_start_page
container_title
container_volume
creator TREWARTHA GARY
NAVARRO EVA F
HOWARD STEVEN
WOOLFORD ALISON J
GILL ADRIAN L
EARLY THERESA R
WYATT PAUL
O'BRIEN MICHAEL A
CARR MARIA G
BERDINI VALERIO
WOODHEAD ANDREW J
description The invention provides compounds of the formula (1): The compounds have activity against cyclin depdenent kinases, glycogen synthase kinase and Auroa kinases and are therefore useful to treat cancer and viral diseases.
format Patent
fullrecord <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_US2007135477A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>US2007135477A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_US2007135477A13</originalsourceid><addsrcrecordid>eNqNyjEKwkAQBdBtLES9w4C1kBhla5WIvVqH0XzJYJxddtYUOb0WHsDqNW_q6j10lJe0PIYe1CLJwFkGGLG2lDtIoreB2CimkCFKT1G2bxDt5CY5JJu7yYN7w-LnzC2P9eVwWiGGBhb5DkVurud1Ufiy2m6835XVf-sDBZk0tQ</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>Benzimidazole derivatives and their use as protein kinases inhibitors</title><source>esp@cenet</source><creator>TREWARTHA GARY ; NAVARRO EVA F ; HOWARD STEVEN ; WOOLFORD ALISON J ; GILL ADRIAN L ; EARLY THERESA R ; WYATT PAUL ; O'BRIEN MICHAEL A ; CARR MARIA G ; BERDINI VALERIO ; WOODHEAD ANDREW J</creator><creatorcontrib>TREWARTHA GARY ; NAVARRO EVA F ; HOWARD STEVEN ; WOOLFORD ALISON J ; GILL ADRIAN L ; EARLY THERESA R ; WYATT PAUL ; O'BRIEN MICHAEL A ; CARR MARIA G ; BERDINI VALERIO ; WOODHEAD ANDREW J</creatorcontrib><description>The invention provides compounds of the formula (1): The compounds have activity against cyclin depdenent kinases, glycogen synthase kinase and Auroa kinases and are therefore useful to treat cancer and viral diseases.</description><language>eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2007</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20070614&amp;DB=EPODOC&amp;CC=US&amp;NR=2007135477A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76516</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20070614&amp;DB=EPODOC&amp;CC=US&amp;NR=2007135477A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>TREWARTHA GARY</creatorcontrib><creatorcontrib>NAVARRO EVA F</creatorcontrib><creatorcontrib>HOWARD STEVEN</creatorcontrib><creatorcontrib>WOOLFORD ALISON J</creatorcontrib><creatorcontrib>GILL ADRIAN L</creatorcontrib><creatorcontrib>EARLY THERESA R</creatorcontrib><creatorcontrib>WYATT PAUL</creatorcontrib><creatorcontrib>O'BRIEN MICHAEL A</creatorcontrib><creatorcontrib>CARR MARIA G</creatorcontrib><creatorcontrib>BERDINI VALERIO</creatorcontrib><creatorcontrib>WOODHEAD ANDREW J</creatorcontrib><title>Benzimidazole derivatives and their use as protein kinases inhibitors</title><description>The invention provides compounds of the formula (1): The compounds have activity against cyclin depdenent kinases, glycogen synthase kinase and Auroa kinases and are therefore useful to treat cancer and viral diseases.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2007</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNyjEKwkAQBdBtLES9w4C1kBhla5WIvVqH0XzJYJxddtYUOb0WHsDqNW_q6j10lJe0PIYe1CLJwFkGGLG2lDtIoreB2CimkCFKT1G2bxDt5CY5JJu7yYN7w-LnzC2P9eVwWiGGBhb5DkVurud1Ufiy2m6835XVf-sDBZk0tQ</recordid><startdate>20070614</startdate><enddate>20070614</enddate><creator>TREWARTHA GARY</creator><creator>NAVARRO EVA F</creator><creator>HOWARD STEVEN</creator><creator>WOOLFORD ALISON J</creator><creator>GILL ADRIAN L</creator><creator>EARLY THERESA R</creator><creator>WYATT PAUL</creator><creator>O'BRIEN MICHAEL A</creator><creator>CARR MARIA G</creator><creator>BERDINI VALERIO</creator><creator>WOODHEAD ANDREW J</creator><scope>EVB</scope></search><sort><creationdate>20070614</creationdate><title>Benzimidazole derivatives and their use as protein kinases inhibitors</title><author>TREWARTHA GARY ; NAVARRO EVA F ; HOWARD STEVEN ; WOOLFORD ALISON J ; GILL ADRIAN L ; EARLY THERESA R ; WYATT PAUL ; O'BRIEN MICHAEL A ; CARR MARIA G ; BERDINI VALERIO ; WOODHEAD ANDREW J</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_US2007135477A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>2007</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>TREWARTHA GARY</creatorcontrib><creatorcontrib>NAVARRO EVA F</creatorcontrib><creatorcontrib>HOWARD STEVEN</creatorcontrib><creatorcontrib>WOOLFORD ALISON J</creatorcontrib><creatorcontrib>GILL ADRIAN L</creatorcontrib><creatorcontrib>EARLY THERESA R</creatorcontrib><creatorcontrib>WYATT PAUL</creatorcontrib><creatorcontrib>O'BRIEN MICHAEL A</creatorcontrib><creatorcontrib>CARR MARIA G</creatorcontrib><creatorcontrib>BERDINI VALERIO</creatorcontrib><creatorcontrib>WOODHEAD ANDREW J</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>TREWARTHA GARY</au><au>NAVARRO EVA F</au><au>HOWARD STEVEN</au><au>WOOLFORD ALISON J</au><au>GILL ADRIAN L</au><au>EARLY THERESA R</au><au>WYATT PAUL</au><au>O'BRIEN MICHAEL A</au><au>CARR MARIA G</au><au>BERDINI VALERIO</au><au>WOODHEAD ANDREW J</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>Benzimidazole derivatives and their use as protein kinases inhibitors</title><date>2007-06-14</date><risdate>2007</risdate><abstract>The invention provides compounds of the formula (1): The compounds have activity against cyclin depdenent kinases, glycogen synthase kinase and Auroa kinases and are therefore useful to treat cancer and viral diseases.</abstract><oa>free_for_read</oa></addata></record>
fulltext fulltext_linktorsrc
identifier
ispartof
issn
language eng
recordid cdi_epo_espacenet_US2007135477A1
source esp@cenet
subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Benzimidazole derivatives and their use as protein kinases inhibitors
url https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-14T22%3A08%3A40IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=TREWARTHA%20GARY&rft.date=2007-06-14&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EUS2007135477A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true