Lactams as CBL-B inhibitors selective over C-CBL

A compound, of formula (I):suitable for treating a cancer wherein the cancer is susceptible to inhibition of Cbl-B.

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Hauptverfasser: Barton, Lisa Marie, Zbieg, Jason Robert, Broccatelli, Fabio, Jakalian, Araz, Larouche-Gauthier, Robin, Ung, Man Un, Liang, Jun, Huestis, Malcolm, Wang, Xiaojing, Yadav, Arun, Castanedo, Georgette Marie, Lambrecht, Michael John, Zhu, Bing-Yan
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creator Barton, Lisa Marie
Zbieg, Jason Robert
Broccatelli, Fabio
Jakalian, Araz
Larouche-Gauthier, Robin
Ung, Man Un
Liang, Jun
Huestis, Malcolm
Wang, Xiaojing
Yadav, Arun
Castanedo, Georgette Marie
Lambrecht, Michael John
Zhu, Bing-Yan
description A compound, of formula (I):suitable for treating a cancer wherein the cancer is susceptible to inhibition of Cbl-B.
format Patent
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Lactams as CBL-B inhibitors selective over C-CBL
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