Phthalazinone compound, and preparation method therefor and medical use thereof

Disclosed are a phthalazinone compound, and a preparation method therefor and the medical use thereof. In particular, disclosed are a compound as represented by formula (I), and a pharmacodynamically acceptable salt, and the use of the compound as an androgen receptor (AR) for degradation.

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Hauptverfasser: Lv, Yongcong, Xing, Weiqiang, Guo, Haibing, Lu, Hongfu, Qi, Baojian, Peng, Jianbiao
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creator Lv, Yongcong
Xing, Weiqiang
Guo, Haibing
Lu, Hongfu
Qi, Baojian
Peng, Jianbiao
description Disclosed are a phthalazinone compound, and a preparation method therefor and the medical use thereof. In particular, disclosed are a compound as represented by formula (I), and a pharmacodynamically acceptable salt, and the use of the compound as an androgen receptor (AR) for degradation.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Phthalazinone compound, and preparation method therefor and medical use thereof
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