Tricyclic inhibitors of the BCL6 BTB domain protein-protein interaction and uses thereof

The present application relates to compounds of Formula (I) or pharmaceutically acceptable salts, solvates and/or prodrugs thereof, to compositions comprising these compounds or pharmaceutically acceptable salts, solvates and/or prodrugs thereof, and various uses in the treatment of diseases, disord...

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Hauptverfasser: Wilson, Brian, Watson, Iain, Subramanian, Pandiaraju, Isaac, Methvin, Poda, Gennady, Uehling, David, Al-awar, Rima, Mamai, Ahmed, Chau, Anh My
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creator Wilson, Brian
Watson, Iain
Subramanian, Pandiaraju
Isaac, Methvin
Poda, Gennady
Uehling, David
Al-awar, Rima
Mamai, Ahmed
Chau, Anh My
description The present application relates to compounds of Formula (I) or pharmaceutically acceptable salts, solvates and/or prodrugs thereof, to compositions comprising these compounds or pharmaceutically acceptable salts, solvates and/or prodrugs thereof, and various uses in the treatment of diseases, disorders or conditions that are treatable by inhibiting interactions with BCL6 BTB, such as cancer.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Tricyclic inhibitors of the BCL6 BTB domain protein-protein interaction and uses thereof
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