Compounds antagonizing A3 adenosine receptor, method for preparing them, and medical-use thereof
The present disclosure provides compounds useful in the amelioration, prevention or treatment of A3 adenosine receptor mediated diseases, such as glaucoma and glaucoma-related ocular disorders, having the structure of Formula I as defined in the detailed description; pharmaceutical compositions comp...
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| creator | Kim, Do-Ran Ahn, Koo-Hyeon Lee, Jin-Hwa Lee, Gwi-Bin Kim, Doo-Seop Hwang, Hyun-Sook Kim, Seung-Yong |
| description | The present disclosure provides compounds useful in the amelioration, prevention or treatment of A3 adenosine receptor mediated diseases, such as glaucoma and glaucoma-related ocular disorders, having the structure of Formula I as defined in the detailed description; pharmaceutical compositions comprising at least one of the compounds; and methods for ameliorating, preventing or treating A3 adenosine receptor mediated diseases using the compound. |
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Hwang, Hyun-Sook ; Kim, Seung-Yong</creatorcontrib><description>The present disclosure provides compounds useful in the amelioration, prevention or treatment of A3 adenosine receptor mediated diseases, such as glaucoma and glaucoma-related ocular disorders, having the structure of Formula I as defined in the detailed description; pharmaceutical compositions comprising at least one of the compounds; and methods for ameliorating, preventing or treating A3 adenosine receptor mediated diseases using the compound.</description><language>eng</language><subject>AGRICULTURE ; ANIMAL HUSBANDRY ; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES ; CHEMISTRY ; FISHING ; FORESTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HUNTING ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PEST REPELLANTS OR ATTRACTANTS ; PLANT GROWTH REGULATORS ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF ; 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pharmaceutical compositions comprising at least one of the compounds; and methods for ameliorating, preventing or treating A3 adenosine receptor mediated diseases using the compound.</description><subject>AGRICULTURE</subject><subject>ANIMAL HUSBANDRY</subject><subject>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</subject><subject>CHEMISTRY</subject><subject>FISHING</subject><subject>FORESTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HUNTING</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PEST REPELLANTS OR ATTRACTANTS</subject><subject>PLANT GROWTH REGULATORS</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</subject><subject>TRAPPING</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2019</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNi8EKgkAURd20iOofXnuFTBBclhTtq7U9nKsO6HvDzLjp60voA1pdOOfcdfKqdXI6iwnEErlXsW8rPZ0KYgPRYAXk0cJF9SlNiIMa6tST83DslzYOmNLv3Xy1sS2P2RywUA_ttsmq4zFg99tNsr9eHvUtg9MGwXELQWye9_yQV2VRledj8U_zAal9PS8</recordid><startdate>20190205</startdate><enddate>20190205</enddate><creator>Kim, Do-Ran</creator><creator>Ahn, Koo-Hyeon</creator><creator>Lee, Jin-Hwa</creator><creator>Lee, Gwi-Bin</creator><creator>Kim, Doo-Seop</creator><creator>Hwang, Hyun-Sook</creator><creator>Kim, Seung-Yong</creator><scope>EVB</scope></search><sort><creationdate>20190205</creationdate><title>Compounds antagonizing A3 adenosine receptor, method for preparing them, and medical-use thereof</title><author>Kim, Do-Ran ; Ahn, Koo-Hyeon ; Lee, Jin-Hwa ; Lee, Gwi-Bin ; Kim, Doo-Seop ; Hwang, Hyun-Sook ; Kim, Seung-Yong</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_US10196396B23</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>2019</creationdate><topic>AGRICULTURE</topic><topic>ANIMAL HUSBANDRY</topic><topic>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</topic><topic>CHEMISTRY</topic><topic>FISHING</topic><topic>FORESTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HUNTING</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PEST REPELLANTS OR ATTRACTANTS</topic><topic>PLANT GROWTH REGULATORS</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</topic><topic>TRAPPING</topic><toplevel>online_resources</toplevel><creatorcontrib>Kim, Do-Ran</creatorcontrib><creatorcontrib>Ahn, Koo-Hyeon</creatorcontrib><creatorcontrib>Lee, Jin-Hwa</creatorcontrib><creatorcontrib>Lee, Gwi-Bin</creatorcontrib><creatorcontrib>Kim, Doo-Seop</creatorcontrib><creatorcontrib>Hwang, Hyun-Sook</creatorcontrib><creatorcontrib>Kim, Seung-Yong</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>Kim, Do-Ran</au><au>Ahn, Koo-Hyeon</au><au>Lee, Jin-Hwa</au><au>Lee, Gwi-Bin</au><au>Kim, Doo-Seop</au><au>Hwang, Hyun-Sook</au><au>Kim, Seung-Yong</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>Compounds antagonizing A3 adenosine receptor, method for preparing them, and medical-use thereof</title><date>2019-02-05</date><risdate>2019</risdate><abstract>The present disclosure provides compounds useful in the amelioration, prevention or treatment of A3 adenosine receptor mediated diseases, such as glaucoma and glaucoma-related ocular disorders, having the structure of Formula I as defined in the detailed description; pharmaceutical compositions comprising at least one of the compounds; and methods for ameliorating, preventing or treating A3 adenosine receptor mediated diseases using the compound.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | AGRICULTURE ANIMAL HUSBANDRY BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES CHEMISTRY FISHING FORESTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HUNTING HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PEST REPELLANTS OR ATTRACTANTS PLANT GROWTH REGULATORS PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF TRAPPING |
| title | Compounds antagonizing A3 adenosine receptor, method for preparing them, and medical-use thereof |
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