Polysubstituted 3-acylamino-5-phenyl-1,4-benzodiazepin-2-one derivatives, process for their preparation and the pharmaceutical compositions containing them

Compounds of formula (I), in which R1 represents (C1-C4) alkyl; RII represents either a group RIIa which is indole optionally substituted on the nitrogen atom with a group W where W represents -(CH2)n-CO-R0 in which n represents 1 to 3 and R0 represents OR2 wherein R2 is H or (C1-C4) alkyl; or RII r...

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Hauptverfasser: FREHEL, DANIEL, DE COINTET, PAUL, DESPEYROUX, PIERRE, GULLY, DANIELE, BADORC, ALAIN
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creator FREHEL, DANIEL
DE COINTET, PAUL
DESPEYROUX, PIERRE
GULLY, DANIELE
BADORC, ALAIN
description Compounds of formula (I), in which R1 represents (C1-C4) alkyl; RII represents either a group RIIa which is indole optionally substituted on the nitrogen atom with a group W where W represents -(CH2)n-CO-R0 in which n represents 1 to 3 and R0 represents OR2 wherein R2 is H or (C1-C4) alkyl; or RII represents a group RIIb in which Y represents a halogen atom or a (C1-C3) alkyl group; X1, X2 and X3 are identical or different and represent a (C1-C4) alkyl or a (C1-C4) alkoxy group; X4 represents hydrogen or a (C1-C4) alkyl group; the stereoisomers thereof and the addition salts thereof.
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subjects BEER
BIOCHEMISTRY
CHEMISTRY
COMPOSITIONS THEREOF
CULTURE MEDIA
ENZYMOLOGY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
MICROBIOLOGY
MICROORGANISMS OR ENZYMES
MUTATION OR GENETIC ENGINEERING
ORGANIC CHEMISTRY
PEPTIDES
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
PROPAGATING, PRESERVING OR MAINTAINING MICROORGANISMS
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
SPIRITS
VINEGAR
WINE
title Polysubstituted 3-acylamino-5-phenyl-1,4-benzodiazepin-2-one derivatives, process for their preparation and the pharmaceutical compositions containing them
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