METHOD OF PREPARING 4-OXY-2H-NAPHTO 2,1-E-1,2-THIAZINE-3-CARBOXAMIDE-1,1-DIOXIDES OR SALTS THEREOF

METHOD OF PREPARING 4-OXY-2H-NAPHTO 2,1-E-1,2-THIAZINE-3-CARBOXAMIDE-1,1-DIOXIDES OR SALTS THEREOF

Compounds of the formula WHEREIN R1 is hydrogen, methyl or ethyl, and Ar is phenyl, 3-chlorophenyl, 3-bromophenyl, 2-fluorophenyl, 3-fluorophenyl, 4-fluorophenyl, 3-tolyl, 2-methoxyphenyl, 3-methoxyphenyl, 2-pyridyl, 4-methyl-2-pyridyl, 6-methyl-2-pyridyl, 3-hydroxy-2-pyridyl, 3-pyridyl, 4-pyridyl,...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: VALTER KHAARMANN,DT, GELMUT TOJFEL,DT, GYUNTER ENGELKHARDT,DT, GYUNTER TRUMMLITTS,DT, ERNST ZEEGER,DT, VOLFKHARD ENGEL,DT
Format: Patent
Sprache:eng
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:Compounds of the formula WHEREIN R1 is hydrogen, methyl or ethyl, and Ar is phenyl, 3-chlorophenyl, 3-bromophenyl, 2-fluorophenyl, 3-fluorophenyl, 4-fluorophenyl, 3-tolyl, 2-methoxyphenyl, 3-methoxyphenyl, 2-pyridyl, 4-methyl-2-pyridyl, 6-methyl-2-pyridyl, 3-hydroxy-2-pyridyl, 3-pyridyl, 4-pyridyl, 6-chloro-3-pyridazinyl, 2-pyrazinyl, 6-chloro-2-pyrazinyl, 6-chloro-4-pyrimidinyl, 2-thiazolyl, 4-methyl-2-thiazolyl, 4-ethyl-2-thiazolyl, 5-methyl-2-thiazolyl, 5-ethyl-2-thiazolyl, 4,5-dimethyl-2-thiazolyl, 4-ethyl-5-methyl-2-thiazolyl, 5-ethyl-4-methyl-2-thiazolyl, 2-benzothiazolyl, 4,5,6,7-tetrahydro-2-benzothiazolyl, 5,6-dihydro-7H-thiopyrano[4,3-d]thiazol-2-yl, 3-methyl-5-isothiazolyl, 1,3,4-thiadiazolyl, 5-methyl-1,3,4-thiadiazol-2-yl or 5-methyl-3-isoxazolyl, AND NON-TOXIC, PHARMACOLOGICALLY ACCEPTABLE SALTS THEREOF FORMED WITH AN INORGANIC OR ORGANIC BASE; THE COMPOUNDS AS WELL AS THEIR SALTS ARE USEFUL AS INHIBITORS OF PLATELET ADHESION AND AGGREGATION.