(1-METHYLPIPERIDIN-4-YL)-2-PROPYL PENTANOATE HYDROCHLORIDE, HAVING CHOLINOLYTIC AND ANTICONVULSANT ACTIVITY
FIELD: chemistry.SUBSTANCE: invention relates to 1-methylpiperidin-4-yl 2-propyl pentanoate hydrochloride of formula I, having cholinolytic and anticonvulsant activity.(I)EFFECT: claimed agent provides considerable reduction of intensity and reduced duration of toxic convulsive syndrome, as well as...
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| creator | Melekhova Aleksandra Sergeevna Kozlov Viktor Konstantinovich Belskaya Alisa Vladimirovna Petrov Aleksandr Nikolaevich Melnikova Margarita Viktorovna Prokopenko Lyubov Ivanovna Gorchakova Tatyana Leonidovna Zajtseva Mariya Anatolevna Ivanov Maksim Borisovich Bespalov Aleksandr Yakovlevich |
| description | FIELD: chemistry.SUBSTANCE: invention relates to 1-methylpiperidin-4-yl 2-propyl pentanoate hydrochloride of formula I, having cholinolytic and anticonvulsant activity.(I)EFFECT: claimed agent provides considerable reduction of intensity and reduced duration of toxic convulsive syndrome, as well as reduced mortality in acute poisoning with cholinesterase inhibitors, particularly carbamates, by using the claimed substance as a specific antidote.1 cl, 3 tbl, 5 ex
Изобретение относится к 1-метилпиперидин-4-ил 2-пропилпентаноата гидрохлориду формулы I, обладающему холинолитической и противосудорожной активностью. Заявляемое средство обеспечивает значительное уменьшение выраженности и сокращение продолжительности токсического судорожного синдрома, а также снижение летальности при острых отравлениях ингибиторами холинэстеразы, в частности карбаматами, путем использования заявляемого вещества как специфического антидота. 3 табл., 5 пр. |
| format | Patent |
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Изобретение относится к 1-метилпиперидин-4-ил 2-пропилпентаноата гидрохлориду формулы I, обладающему холинолитической и противосудорожной активностью. Заявляемое средство обеспечивает значительное уменьшение выраженности и сокращение продолжительности токсического судорожного синдрома, а также снижение летальности при острых отравлениях ингибиторами холинэстеразы, в частности карбаматами, путем использования заявляемого вещества как специфического антидота. 3 табл., 5 пр.</description><language>eng ; rus</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2020</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20200212&DB=EPODOC&CC=RU&NR=2714135C1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20200212&DB=EPODOC&CC=RU&NR=2714135C1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>Melekhova Aleksandra Sergeevna</creatorcontrib><creatorcontrib>Kozlov Viktor Konstantinovich</creatorcontrib><creatorcontrib>Belskaya Alisa Vladimirovna</creatorcontrib><creatorcontrib>Petrov Aleksandr Nikolaevich</creatorcontrib><creatorcontrib>Melnikova Margarita Viktorovna</creatorcontrib><creatorcontrib>Prokopenko Lyubov Ivanovna</creatorcontrib><creatorcontrib>Gorchakova Tatyana Leonidovna</creatorcontrib><creatorcontrib>Zajtseva Mariya Anatolevna</creatorcontrib><creatorcontrib>Ivanov Maksim Borisovich</creatorcontrib><creatorcontrib>Bespalov Aleksandr Yakovlevich</creatorcontrib><title>(1-METHYLPIPERIDIN-4-YL)-2-PROPYL PENTANOATE HYDROCHLORIDE, HAVING CHOLINOLYTIC AND ANTICONVULSANT ACTIVITY</title><description>FIELD: chemistry.SUBSTANCE: invention relates to 1-methylpiperidin-4-yl 2-propyl pentanoate hydrochloride of formula I, having cholinolytic and anticonvulsant activity.(I)EFFECT: claimed agent provides considerable reduction of intensity and reduced duration of toxic convulsive syndrome, as well as reduced mortality in acute poisoning with cholinesterase inhibitors, particularly carbamates, by using the claimed substance as a specific antidote.1 cl, 3 tbl, 5 ex
Изобретение относится к 1-метилпиперидин-4-ил 2-пропилпентаноата гидрохлориду формулы I, обладающему холинолитической и противосудорожной активностью. Заявляемое средство обеспечивает значительное уменьшение выраженности и сокращение продолжительности токсического судорожного синдрома, а также снижение летальности при острых отравлениях ингибиторами холинэстеразы, в частности карбаматами, путем использования заявляемого вещества как специфического антидота. 3 табл., 5 пр.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2020</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNirEKwjAUALs4iPoPGRXMkLbiHNJoHjzzQkwDmUqRuChaqP-PGfwAh-NuuGX12Ap-0cEkdOC0hw4sb3nCHa-58-QSMqdtkJZk0MykzpMySGXUe2ZkBHtmyhCCJUwBFJO2K5QiG3u8lmRSBYgQ0rpa3MfnnDc_ryp20kEZnqf3kOdpvOVX_gy-r4-iFc1BieaP5QtmxTZt</recordid><startdate>20200212</startdate><enddate>20200212</enddate><creator>Melekhova Aleksandra Sergeevna</creator><creator>Kozlov Viktor Konstantinovich</creator><creator>Belskaya Alisa Vladimirovna</creator><creator>Petrov Aleksandr Nikolaevich</creator><creator>Melnikova Margarita Viktorovna</creator><creator>Prokopenko Lyubov Ivanovna</creator><creator>Gorchakova Tatyana Leonidovna</creator><creator>Zajtseva Mariya Anatolevna</creator><creator>Ivanov Maksim Borisovich</creator><creator>Bespalov Aleksandr Yakovlevich</creator><scope>EVB</scope></search><sort><creationdate>20200212</creationdate><title>(1-METHYLPIPERIDIN-4-YL)-2-PROPYL PENTANOATE HYDROCHLORIDE, HAVING CHOLINOLYTIC AND ANTICONVULSANT ACTIVITY</title><author>Melekhova Aleksandra Sergeevna ; Kozlov Viktor Konstantinovich ; Belskaya Alisa Vladimirovna ; Petrov Aleksandr Nikolaevich ; Melnikova Margarita Viktorovna ; Prokopenko Lyubov Ivanovna ; Gorchakova Tatyana Leonidovna ; Zajtseva Mariya Anatolevna ; Ivanov Maksim Borisovich ; Bespalov Aleksandr Yakovlevich</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_RU2714135C13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; rus</language><creationdate>2020</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>Melekhova Aleksandra Sergeevna</creatorcontrib><creatorcontrib>Kozlov Viktor Konstantinovich</creatorcontrib><creatorcontrib>Belskaya Alisa Vladimirovna</creatorcontrib><creatorcontrib>Petrov Aleksandr Nikolaevich</creatorcontrib><creatorcontrib>Melnikova Margarita Viktorovna</creatorcontrib><creatorcontrib>Prokopenko Lyubov Ivanovna</creatorcontrib><creatorcontrib>Gorchakova Tatyana Leonidovna</creatorcontrib><creatorcontrib>Zajtseva Mariya Anatolevna</creatorcontrib><creatorcontrib>Ivanov Maksim Borisovich</creatorcontrib><creatorcontrib>Bespalov Aleksandr Yakovlevich</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>Melekhova Aleksandra Sergeevna</au><au>Kozlov Viktor Konstantinovich</au><au>Belskaya Alisa Vladimirovna</au><au>Petrov Aleksandr Nikolaevich</au><au>Melnikova Margarita Viktorovna</au><au>Prokopenko Lyubov Ivanovna</au><au>Gorchakova Tatyana Leonidovna</au><au>Zajtseva Mariya Anatolevna</au><au>Ivanov Maksim Borisovich</au><au>Bespalov Aleksandr Yakovlevich</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>(1-METHYLPIPERIDIN-4-YL)-2-PROPYL PENTANOATE HYDROCHLORIDE, HAVING CHOLINOLYTIC AND ANTICONVULSANT ACTIVITY</title><date>2020-02-12</date><risdate>2020</risdate><abstract>FIELD: chemistry.SUBSTANCE: invention relates to 1-methylpiperidin-4-yl 2-propyl pentanoate hydrochloride of formula I, having cholinolytic and anticonvulsant activity.(I)EFFECT: claimed agent provides considerable reduction of intensity and reduced duration of toxic convulsive syndrome, as well as reduced mortality in acute poisoning with cholinesterase inhibitors, particularly carbamates, by using the claimed substance as a specific antidote.1 cl, 3 tbl, 5 ex
Изобретение относится к 1-метилпиперидин-4-ил 2-пропилпентаноата гидрохлориду формулы I, обладающему холинолитической и противосудорожной активностью. Заявляемое средство обеспечивает значительное уменьшение выраженности и сокращение продолжительности токсического судорожного синдрома, а также снижение летальности при острых отравлениях ингибиторами холинэстеразы, в частности карбаматами, путем использования заявляемого вещества как специфического антидота. 3 табл., 5 пр.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | (1-METHYLPIPERIDIN-4-YL)-2-PROPYL PENTANOATE HYDROCHLORIDE, HAVING CHOLINOLYTIC AND ANTICONVULSANT ACTIVITY |
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