5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONE DERIVATIVES, COMPOSITION BASED THEREON AND METHOD FOR CONTROLLING FUNGAL DISEASES
FIELD: agriculture.SUBSTANCE: invention relates to agriculture. Fungicidally active compound of formula I:formula I, wherein Rrepresents: C-C-alkyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkenyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkynyl, optionally...
Gespeichert in:
| Hauptverfasser: | , , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | eng ; rus |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | OUEN U Dzhon YAO Chenlin BEBEL Timoti A SALLENBERGER Majkl T LORSBAKH Bet VEBSTER Dzheffri D GELLIFORD Kris V |
| description | FIELD: agriculture.SUBSTANCE: invention relates to agriculture. Fungicidally active compound of formula I:formula I, wherein Rrepresents: C-C-alkyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkenyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkynyl, optionally having as substitutes from 1 to 3 radicals R; phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms, and each ring can optionally contain as substitutes from 1 to 3 radicals R, -(CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; or -C(=S)N(R)R; where m is an integer from 1 to 3; Rrepresents: H; or C-C-alkyl, optionally having as substitutes radical R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, amino, halogenthio, C-C-alkylamino, C-C-alkoxycarbonyl, C-C-alkylcarbonyl, C-C-alkylaminocarbonyl, hydroxyl, C-C-trialkylsilyl, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, halogenthio, amino, C-C-alkylamino, C-C-dialkylamino, C-C-alkoxycarbonyl, C-C-alkylsulphonyl or C-C-alkylcarbonyl, nitro, hydroxyl or cyano; Rrepresents H, C-C-alkyl, C-C-alkoxy, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alk |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_RU2613451C2</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>RU2613451C2</sourcerecordid><originalsourceid>FETCH-epo_espacenet_RU2613451C23</originalsourceid><addsrcrecordid>eNqNyz2KAkEQhuFJNljcvUOFClYwf-bjVI1dMNMl3dWCkYi00bIruCfxxE7gAYw-Xni-z-LR4jAmDYoNyiRescZlTNtoYsmYVlivGyRxRwq6P4bZkHiscFm6FapnIA5y6EwOHNfQ67TXKCbqYdtFJjDHgefqPMHE5pRg0DBDb0HHUfwOhuR33QgkkedL_Co-ruefe_5-7aKAga13mG9_p3y_nS_5N_-fQqo2Zd20ZV_Vb5Anx2BAIA</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONE DERIVATIVES, COMPOSITION BASED THEREON AND METHOD FOR CONTROLLING FUNGAL DISEASES</title><source>esp@cenet</source><creator>OUEN U Dzhon ; YAO Chenlin ; BEBEL Timoti A ; SALLENBERGER Majkl T ; LORSBAKH Bet ; VEBSTER Dzheffri D ; GELLIFORD Kris V</creator><creatorcontrib>OUEN U Dzhon ; YAO Chenlin ; BEBEL Timoti A ; SALLENBERGER Majkl T ; LORSBAKH Bet ; VEBSTER Dzheffri D ; GELLIFORD Kris V</creatorcontrib><description>FIELD: agriculture.SUBSTANCE: invention relates to agriculture. Fungicidally active compound of formula I:formula I, wherein Rrepresents: C-C-alkyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkenyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkynyl, optionally having as substitutes from 1 to 3 radicals R; phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms, and each ring can optionally contain as substitutes from 1 to 3 radicals R, -(CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; or -C(=S)N(R)R; where m is an integer from 1 to 3; Rrepresents: H; or C-C-alkyl, optionally having as substitutes radical R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, amino, halogenthio, C-C-alkylamino, C-C-alkoxycarbonyl, C-C-alkylcarbonyl, C-C-alkylaminocarbonyl, hydroxyl, C-C-trialkylsilyl, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, halogenthio, amino, C-C-alkylamino, C-C-dialkylamino, C-C-alkoxycarbonyl, C-C-alkylsulphonyl or C-C-alkylcarbonyl, nitro, hydroxyl or cyano; Rrepresents H, C-C-alkyl, C-C-alkoxy, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; and Rrepresents H, C-C-alkyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, or benzyl, wherein benzyl can optionally contain as substitutes from 1 to 3 radicals R; alternatively, Rand Rcan together form a 5- or 6-member saturated or unsaturated ring containing from 1 to 3 heteroatoms, each ring can optionally contain as substitutes from 1 to 3 radicals R.EFFECT: higher efficiency of controlling plant fungal diseases.17 cl, 2 tbl, 5 ex
Изобретение относится к сельскому хозяйству. Фунгицидоактивное соединение формулы I:в которой Rпредставляет собой: C-C-алкил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; C-C-алкенил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; C-C-алкинил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; фенил или бензил, причем каждый фенил или бензил может необязательно содержать в качестве заместителей от 1 до 3 радикалов R, или систему из 5- или 6-членных насыщенных или ненасыщенных колец, или конденсированную систему из 5- и 6-членных колец, или конденсированную систему из 6-6-членных колец, причем каждая система содержит от 1 до 3 гетероатомов, и каждое кольцо может необязательно содержать в качестве заместителей от 1 до 3 радикалов R, - (CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; или -C(=S)N(R)R; в которой m представляет собой целое число от 1 до 3; Rпредставляет собой: Н; или C-C-алкил, необязательно содержащий в качестве заместителя радикал R; Rнезависимо представляет собой галоген, C-C-алкил, C-C-галогеналкил, C-C-алкокси, C-C-галогеналкокси, C-C-алкилтио, C-C-галогеналкилтио, амино, галогентио, C-C-алкиламино, C-C-алкоксикарбонил, C-C-алкилкарбонил, C-C-алкиламинокарбонил, гидроксил, C-C-триалкилсилил, или систему из 5- или 6-членных насыщенных или ненасыщенных колец, или конденсированную систему из 5- и 6-членных колец, или конденсированную систему из 6-6-членных колец, причем каждая система содержит от 1 до 3 гетероатомов и каждое кольцо может необязательно содержать в качестве заместителей от 1 до 3 радикалов R; Rнезависимо представляет собой галоген, C-C-алкил, C-C-галогеналкил, C-C-алкокси, C-C-галогеналкокси, C-C-алкилтио, C-C-галогеналкилтио, галогентио, амино, C-C-алкиламино, C-C-диалкиламино, C-C-алкоксикарбонил,</description><language>eng ; rus</language><subject>AGRICULTURE ; ANIMAL HUSBANDRY ; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES ; FISHING ; FORESTRY ; HUMAN NECESSITIES ; HUNTING ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; PEST REPELLANTS OR ATTRACTANTS ; PLANT GROWTH REGULATORS ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF ; TRAPPING</subject><creationdate>2017</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20170316&DB=EPODOC&CC=RU&NR=2613451C2$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25563,76418</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20170316&DB=EPODOC&CC=RU&NR=2613451C2$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>OUEN U Dzhon</creatorcontrib><creatorcontrib>YAO Chenlin</creatorcontrib><creatorcontrib>BEBEL Timoti A</creatorcontrib><creatorcontrib>SALLENBERGER Majkl T</creatorcontrib><creatorcontrib>LORSBAKH Bet</creatorcontrib><creatorcontrib>VEBSTER Dzheffri D</creatorcontrib><creatorcontrib>GELLIFORD Kris V</creatorcontrib><title>5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONE DERIVATIVES, COMPOSITION BASED THEREON AND METHOD FOR CONTROLLING FUNGAL DISEASES</title><description>FIELD: agriculture.SUBSTANCE: invention relates to agriculture. Fungicidally active compound of formula I:formula I, wherein Rrepresents: C-C-alkyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkenyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkynyl, optionally having as substitutes from 1 to 3 radicals R; phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms, and each ring can optionally contain as substitutes from 1 to 3 radicals R, -(CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; or -C(=S)N(R)R; where m is an integer from 1 to 3; Rrepresents: H; or C-C-alkyl, optionally having as substitutes radical R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, amino, halogenthio, C-C-alkylamino, C-C-alkoxycarbonyl, C-C-alkylcarbonyl, C-C-alkylaminocarbonyl, hydroxyl, C-C-trialkylsilyl, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, halogenthio, amino, C-C-alkylamino, C-C-dialkylamino, C-C-alkoxycarbonyl, C-C-alkylsulphonyl or C-C-alkylcarbonyl, nitro, hydroxyl or cyano; Rrepresents H, C-C-alkyl, C-C-alkoxy, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; and Rrepresents H, C-C-alkyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, or benzyl, wherein benzyl can optionally contain as substitutes from 1 to 3 radicals R; alternatively, Rand Rcan together form a 5- or 6-member saturated or unsaturated ring containing from 1 to 3 heteroatoms, each ring can optionally contain as substitutes from 1 to 3 radicals R.EFFECT: higher efficiency of controlling plant fungal diseases.17 cl, 2 tbl, 5 ex
Изобретение относится к сельскому хозяйству. Фунгицидоактивное соединение формулы I:в которой Rпредставляет собой: C-C-алкил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; C-C-алкенил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; C-C-алкинил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; фенил или бензил, причем каждый фенил или бензил может необязательно содержать в качестве заместителей от 1 до 3 радикалов R, или систему из 5- или 6-членных насыщенных или ненасыщенных колец, или конденсированную систему из 5- и 6-членных колец, или конденсированную систему из 6-6-членных колец, причем каждая система содержит от 1 до 3 гетероатомов, и каждое кольцо может необязательно содержать в качестве заместителей от 1 до 3 радикалов R, - (CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; или -C(=S)N(R)R; в которой m представляет собой целое число от 1 до 3; Rпредставляет собой: Н; или C-C-алкил, необязательно содержащий в качестве заместителя радикал R; Rнезависимо представляет собой галоген, C-C-алкил, C-C-галогеналкил, C-C-алкокси, C-C-галогеналкокси, C-C-алкилтио, C-C-галогеналкилтио, амино, галогентио, C-C-алкиламино, C-C-алкоксикарбонил, C-C-алкилкарбонил, C-C-алкиламинокарбонил, гидроксил, C-C-триалкилсилил, или систему из 5- или 6-членных насыщенных или ненасыщенных колец, или конденсированную систему из 5- и 6-членных колец, или конденсированную систему из 6-6-членных колец, причем каждая система содержит от 1 до 3 гетероатомов и каждое кольцо может необязательно содержать в качестве заместителей от 1 до 3 радикалов R; Rнезависимо представляет собой галоген, C-C-алкил, C-C-галогеналкил, C-C-алкокси, C-C-галогеналкокси, C-C-алкилтио, C-C-галогеналкилтио, галогентио, амино, C-C-алкиламино, C-C-диалкиламино, C-C-алкоксикарбонил,</description><subject>AGRICULTURE</subject><subject>ANIMAL HUSBANDRY</subject><subject>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</subject><subject>FISHING</subject><subject>FORESTRY</subject><subject>HUMAN NECESSITIES</subject><subject>HUNTING</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>PEST REPELLANTS OR ATTRACTANTS</subject><subject>PLANT GROWTH REGULATORS</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</subject><subject>TRAPPING</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2017</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNyz2KAkEQhuFJNljcvUOFClYwf-bjVI1dMNMl3dWCkYi00bIruCfxxE7gAYw-Xni-z-LR4jAmDYoNyiRescZlTNtoYsmYVlivGyRxRwq6P4bZkHiscFm6FapnIA5y6EwOHNfQ67TXKCbqYdtFJjDHgefqPMHE5pRg0DBDb0HHUfwOhuR33QgkkedL_Co-ruefe_5-7aKAga13mG9_p3y_nS_5N_-fQqo2Zd20ZV_Vb5Anx2BAIA</recordid><startdate>20170316</startdate><enddate>20170316</enddate><creator>OUEN U Dzhon</creator><creator>YAO Chenlin</creator><creator>BEBEL Timoti A</creator><creator>SALLENBERGER Majkl T</creator><creator>LORSBAKH Bet</creator><creator>VEBSTER Dzheffri D</creator><creator>GELLIFORD Kris V</creator><scope>EVB</scope></search><sort><creationdate>20170316</creationdate><title>5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONE DERIVATIVES, COMPOSITION BASED THEREON AND METHOD FOR CONTROLLING FUNGAL DISEASES</title><author>OUEN U Dzhon ; YAO Chenlin ; BEBEL Timoti A ; SALLENBERGER Majkl T ; LORSBAKH Bet ; VEBSTER Dzheffri D ; GELLIFORD Kris V</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_RU2613451C23</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; rus</language><creationdate>2017</creationdate><topic>AGRICULTURE</topic><topic>ANIMAL HUSBANDRY</topic><topic>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</topic><topic>FISHING</topic><topic>FORESTRY</topic><topic>HUMAN NECESSITIES</topic><topic>HUNTING</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>PEST REPELLANTS OR ATTRACTANTS</topic><topic>PLANT GROWTH REGULATORS</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</topic><topic>TRAPPING</topic><toplevel>online_resources</toplevel><creatorcontrib>OUEN U Dzhon</creatorcontrib><creatorcontrib>YAO Chenlin</creatorcontrib><creatorcontrib>BEBEL Timoti A</creatorcontrib><creatorcontrib>SALLENBERGER Majkl T</creatorcontrib><creatorcontrib>LORSBAKH Bet</creatorcontrib><creatorcontrib>VEBSTER Dzheffri D</creatorcontrib><creatorcontrib>GELLIFORD Kris V</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>OUEN U Dzhon</au><au>YAO Chenlin</au><au>BEBEL Timoti A</au><au>SALLENBERGER Majkl T</au><au>LORSBAKH Bet</au><au>VEBSTER Dzheffri D</au><au>GELLIFORD Kris V</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONE DERIVATIVES, COMPOSITION BASED THEREON AND METHOD FOR CONTROLLING FUNGAL DISEASES</title><date>2017-03-16</date><risdate>2017</risdate><abstract>FIELD: agriculture.SUBSTANCE: invention relates to agriculture. Fungicidally active compound of formula I:formula I, wherein Rrepresents: C-C-alkyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkenyl, optionally having as substitutes from 1 to 3 radicals R; C-C-alkynyl, optionally having as substitutes from 1 to 3 radicals R; phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms, and each ring can optionally contain as substitutes from 1 to 3 radicals R, -(CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; or -C(=S)N(R)R; where m is an integer from 1 to 3; Rrepresents: H; or C-C-alkyl, optionally having as substitutes radical R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, amino, halogenthio, C-C-alkylamino, C-C-alkoxycarbonyl, C-C-alkylcarbonyl, C-C-alkylaminocarbonyl, hydroxyl, C-C-trialkylsilyl, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R; Rindependently represents a halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-halogenalkoxy, C-C-alkylthio, C-C-halogenalkylthio, halogenthio, amino, C-C-alkylamino, C-C-dialkylamino, C-C-alkoxycarbonyl, C-C-alkylsulphonyl or C-C-alkylcarbonyl, nitro, hydroxyl or cyano; Rrepresents H, C-C-alkyl, C-C-alkoxy, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-haloalkyl, C-C-alkoxyalkyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; Rrepresents H, C-C-alkyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally contain as substitutes from 1 to 3 radicals R, or a system of 5- or 6-member saturated or unsaturated rings, or condensed system consisting of 5- and 6-member rings, or condensed system of 6-6-member rings, each system includes from 1 to 3 heteroatoms and each ring can optionally contain as substitutes from 1 to 3 radicals R, biphenyl or naphthyl, optionally having as substitutes from 1 to 3 radicals R; and Rrepresents H, C-C-alkyl, C-C-haloalkyl, C-C-alkoxyalkyl, C-C-alkylcarbonyl, or benzyl, wherein benzyl can optionally contain as substitutes from 1 to 3 radicals R; alternatively, Rand Rcan together form a 5- or 6-member saturated or unsaturated ring containing from 1 to 3 heteroatoms, each ring can optionally contain as substitutes from 1 to 3 radicals R.EFFECT: higher efficiency of controlling plant fungal diseases.17 cl, 2 tbl, 5 ex
Изобретение относится к сельскому хозяйству. Фунгицидоактивное соединение формулы I:в которой Rпредставляет собой: C-C-алкил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; C-C-алкенил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; C-C-алкинил, необязательно содержащий в качестве заместителей от 1 до 3 радикалов R; фенил или бензил, причем каждый фенил или бензил может необязательно содержать в качестве заместителей от 1 до 3 радикалов R, или систему из 5- или 6-членных насыщенных или ненасыщенных колец, или конденсированную систему из 5- и 6-членных колец, или конденсированную систему из 6-6-членных колец, причем каждая система содержит от 1 до 3 гетероатомов, и каждое кольцо может необязательно содержать в качестве заместителей от 1 до 3 радикалов R, - (CHR)OR; -C(=O)R; -C(=S)R; -C(=O)OR; -C(=S)OR; -S(O)R; -(CHR)N(R)R; -C(=O)N(R)R; или -C(=S)N(R)R; в которой m представляет собой целое число от 1 до 3; Rпредставляет собой: Н; или C-C-алкил, необязательно содержащий в качестве заместителя радикал R; Rнезависимо представляет собой галоген, C-C-алкил, C-C-галогеналкил, C-C-алкокси, C-C-галогеналкокси, C-C-алкилтио, C-C-галогеналкилтио, амино, галогентио, C-C-алкиламино, C-C-алкоксикарбонил, C-C-алкилкарбонил, C-C-алкиламинокарбонил, гидроксил, C-C-триалкилсилил, или систему из 5- или 6-членных насыщенных или ненасыщенных колец, или конденсированную систему из 5- и 6-членных колец, или конденсированную систему из 6-6-членных колец, причем каждая система содержит от 1 до 3 гетероатомов и каждое кольцо может необязательно содержать в качестве заместителей от 1 до 3 радикалов R; Rнезависимо представляет собой галоген, C-C-алкил, C-C-галогеналкил, C-C-алкокси, C-C-галогеналкокси, C-C-алкилтио, C-C-галогеналкилтио, галогентио, амино, C-C-алкиламино, C-C-диалкиламино, C-C-алкоксикарбонил,</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | eng ; rus |
| recordid | cdi_epo_espacenet_RU2613451C2 |
| source | esp@cenet |
| subjects | AGRICULTURE ANIMAL HUSBANDRY BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES FISHING FORESTRY HUMAN NECESSITIES HUNTING HYGIENE MEDICAL OR VETERINARY SCIENCE PEST REPELLANTS OR ATTRACTANTS PLANT GROWTH REGULATORS PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF TRAPPING |
| title | 5-FLUORO-4-IMINO-3-(SUBSTITUTED)-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONE DERIVATIVES, COMPOSITION BASED THEREON AND METHOD FOR CONTROLLING FUNGAL DISEASES |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-08T07%3A43%3A40IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=OUEN%20U%20Dzhon&rft.date=2017-03-16&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3ERU2613451C2%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |