PHENYLACETIC ACID DERIVATIVES, THEIR INTERMEDIATES, AND AGENTS CONTAINING THEREOF
organic synthesis. SUBSTANCE: invention provides novel phenylacetic acid derivatives of general formula I: (I), in which X denotes NOCH3, CHOCH3 and CHCH2CH3; R1 hydrogen or C1-C4-alkyl; R2 halogen, C1-C4-alkyl, or C1- C4-alkoxy; m= 0 or 1; R3 denotes hydrogen, amino, halogen, C1-C4-alkyl, C1- C4-ha...
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creator | VASSILIOS GRAMMENOS RAJNKHARD KIRSTGEN AL'BREKHT KHARREUS GERBERT BAJER GIZELA LORENTS EHBERKHARD AMMERMANN KHUBERT ZAUTER FRANTS REL RUT MJULLER |
description | organic synthesis. SUBSTANCE: invention provides novel phenylacetic acid derivatives of general formula I: (I), in which X denotes NOCH3, CHOCH3 and CHCH2CH3; R1 hydrogen or C1-C4-alkyl; R2 halogen, C1-C4-alkyl, or C1- C4-alkoxy; m= 0 or 1; R3 denotes hydrogen, amino, halogen, C1-C4-alkyl, C1- C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-alkylamino, or di- C1- C4-alkylamino; R4 cyano, halogen, C1-C6-alkyl, C1-C6-alkoxy, C2-C6- alkenyl, C2-C6-alkenyloxy, or C2-C6-alkinyl; provided that hydrocarbon moieties of above-indicated groups can be partially or completely halogenated or can bear one to three substituents selected from cyano, C1- C6-alkoxy, C1-C6-alkoxycarbonyl, phenyl, and dioxan (cyclic radicals can be partially or completely halogenated), C3-C6-cycloalkyl, C3-C6-cycloalkenyl, aryl, isoxazolyl, pyridyl, dioxolanyl, benzoxazolyl, thienyl, oxazolyl, furyl, oxyranyl, pyrazolyl, thiazolyl, pyrimidyloxy or tetrahydropyranyl, provided that cyclic radicals can be partially or completely halogenated or can bear one to three substituents selected from nitro, C1-C6-alkyl, C1-C6- alkoxy, C1-C6-haloalkyl, C1-C6-alkylamino, di-C1-C6-alkylamino and aryl; R5 denotes hydrogen, C1-C10-alkyl, C2-C10-alkenyl, or C2-C10-alkinyl, provided that these radicals can be partially or completely halogenated or can bear one to three substituents selected from cyano, hydroxy, aminocarbonyl, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkoxycarbonyl, C1-C6- alkylamino, benzyl, aryl, aryloxy, thienyl, pyrrolyl, oxazolyl, furyl, thiazolyl, oxadiazolyl, and isoxazolyl, cyclic radicals themselves can be partially or completely halogenated or can bear one to three substituents selected from nitro, hydroxy, C1-C4-alkyl, C1-C4-haloakyl, and C3-C6- cycloalkyl; on condition that X cannot be NOCH3 and CHOCH3, when R4 is unsubstituted C1-C4-alkyl, unsubstituted C3-C6-cycloalkyl, substituted or unsubstituted phenyl, or unsubstituted thienyl; or X cannot be CHOCH3, when R3 is hydrogen and R5 is C1-C10-alkyl; as well as salts or above-indicated compounds. Compound I show fungicidal activity. EFFECT: extended choice of active fungicides. 8 cl, 16 tbl, 10 ex |
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fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_RU2165411C2</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>RU2165411C2</sourcerecordid><originalsourceid>FETCH-epo_espacenet_RU2165411C23</originalsourceid><addsrcrecordid>eNqNyj0KwkAQQOFtLES9wxxAi40__TA7yQ7oRDdjwCoEWSvRQLw_EvAAVg8e39xdzpH1dkRiEwIkCRA4SYsmLTdrsMiSQNQ4nTgI2jRRA2DFag1QrYaiotVEE9fl0s0e_XPMq18XDko2ips8vLs8Dv09v_KnS9fCH_Y776nY_kG-PqEu8A</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>PHENYLACETIC ACID DERIVATIVES, THEIR INTERMEDIATES, AND AGENTS CONTAINING THEREOF</title><source>esp@cenet</source><creator>VASSILIOS GRAMMENOS ; RAJNKHARD KIRSTGEN ; AL'BREKHT KHARREUS ; GERBERT BAJER ; GIZELA LORENTS ; EHBERKHARD AMMERMANN ; KHUBERT ZAUTER ; FRANTS REL ; RUT MJULLER</creator><creatorcontrib>VASSILIOS GRAMMENOS ; RAJNKHARD KIRSTGEN ; AL'BREKHT KHARREUS ; GERBERT BAJER ; GIZELA LORENTS ; EHBERKHARD AMMERMANN ; KHUBERT ZAUTER ; FRANTS REL ; RUT MJULLER</creatorcontrib><description>organic synthesis. SUBSTANCE: invention provides novel phenylacetic acid derivatives of general formula I: (I), in which X denotes NOCH3, CHOCH3 and CHCH2CH3; R1 hydrogen or C1-C4-alkyl; R2 halogen, C1-C4-alkyl, or C1- C4-alkoxy; m= 0 or 1; R3 denotes hydrogen, amino, halogen, C1-C4-alkyl, C1- C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-alkylamino, or di- C1- C4-alkylamino; R4 cyano, halogen, C1-C6-alkyl, C1-C6-alkoxy, C2-C6- alkenyl, C2-C6-alkenyloxy, or C2-C6-alkinyl; provided that hydrocarbon moieties of above-indicated groups can be partially or completely halogenated or can bear one to three substituents selected from cyano, C1- C6-alkoxy, C1-C6-alkoxycarbonyl, phenyl, and dioxan (cyclic radicals can be partially or completely halogenated), C3-C6-cycloalkyl, C3-C6-cycloalkenyl, aryl, isoxazolyl, pyridyl, dioxolanyl, benzoxazolyl, thienyl, oxazolyl, furyl, oxyranyl, pyrazolyl, thiazolyl, pyrimidyloxy or tetrahydropyranyl, provided that cyclic radicals can be partially or completely halogenated or can bear one to three substituents selected from nitro, C1-C6-alkyl, C1-C6- alkoxy, C1-C6-haloalkyl, C1-C6-alkylamino, di-C1-C6-alkylamino and aryl; R5 denotes hydrogen, C1-C10-alkyl, C2-C10-alkenyl, or C2-C10-alkinyl, provided that these radicals can be partially or completely halogenated or can bear one to three substituents selected from cyano, hydroxy, aminocarbonyl, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkoxycarbonyl, C1-C6- alkylamino, benzyl, aryl, aryloxy, thienyl, pyrrolyl, oxazolyl, furyl, thiazolyl, oxadiazolyl, and isoxazolyl, cyclic radicals themselves can be partially or completely halogenated or can bear one to three substituents selected from nitro, hydroxy, C1-C4-alkyl, C1-C4-haloakyl, and C3-C6- cycloalkyl; on condition that X cannot be NOCH3 and CHOCH3, when R4 is unsubstituted C1-C4-alkyl, unsubstituted C3-C6-cycloalkyl, substituted or unsubstituted phenyl, or unsubstituted thienyl; or X cannot be CHOCH3, when R3 is hydrogen and R5 is C1-C10-alkyl; as well as salts or above-indicated compounds. Compound I show fungicidal activity. EFFECT: extended choice of active fungicides. 8 cl, 16 tbl, 10 ex</description><edition>7</edition><language>eng ; rus</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; AGRICULTURE ; ANIMAL HUSBANDRY ; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES ; CHEMISTRY ; FISHING ; FORESTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HUNTING ; METALLURGY ; ORGANIC CHEMISTRY ; PEST REPELLANTS OR ATTRACTANTS ; PLANT GROWTH REGULATORS ; PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF ; TRAPPING</subject><creationdate>2001</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20010420&DB=EPODOC&CC=RU&NR=2165411C2$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25563,76318</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20010420&DB=EPODOC&CC=RU&NR=2165411C2$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>VASSILIOS GRAMMENOS</creatorcontrib><creatorcontrib>RAJNKHARD KIRSTGEN</creatorcontrib><creatorcontrib>AL'BREKHT KHARREUS</creatorcontrib><creatorcontrib>GERBERT BAJER</creatorcontrib><creatorcontrib>GIZELA LORENTS</creatorcontrib><creatorcontrib>EHBERKHARD AMMERMANN</creatorcontrib><creatorcontrib>KHUBERT ZAUTER</creatorcontrib><creatorcontrib>FRANTS REL</creatorcontrib><creatorcontrib>RUT MJULLER</creatorcontrib><title>PHENYLACETIC ACID DERIVATIVES, THEIR INTERMEDIATES, AND AGENTS CONTAINING THEREOF</title><description>organic synthesis. SUBSTANCE: invention provides novel phenylacetic acid derivatives of general formula I: (I), in which X denotes NOCH3, CHOCH3 and CHCH2CH3; R1 hydrogen or C1-C4-alkyl; R2 halogen, C1-C4-alkyl, or C1- C4-alkoxy; m= 0 or 1; R3 denotes hydrogen, amino, halogen, C1-C4-alkyl, C1- C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-alkylamino, or di- C1- C4-alkylamino; R4 cyano, halogen, C1-C6-alkyl, C1-C6-alkoxy, C2-C6- alkenyl, C2-C6-alkenyloxy, or C2-C6-alkinyl; provided that hydrocarbon moieties of above-indicated groups can be partially or completely halogenated or can bear one to three substituents selected from cyano, C1- C6-alkoxy, C1-C6-alkoxycarbonyl, phenyl, and dioxan (cyclic radicals can be partially or completely halogenated), C3-C6-cycloalkyl, C3-C6-cycloalkenyl, aryl, isoxazolyl, pyridyl, dioxolanyl, benzoxazolyl, thienyl, oxazolyl, furyl, oxyranyl, pyrazolyl, thiazolyl, pyrimidyloxy or tetrahydropyranyl, provided that cyclic radicals can be partially or completely halogenated or can bear one to three substituents selected from nitro, C1-C6-alkyl, C1-C6- alkoxy, C1-C6-haloalkyl, C1-C6-alkylamino, di-C1-C6-alkylamino and aryl; R5 denotes hydrogen, C1-C10-alkyl, C2-C10-alkenyl, or C2-C10-alkinyl, provided that these radicals can be partially or completely halogenated or can bear one to three substituents selected from cyano, hydroxy, aminocarbonyl, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkoxycarbonyl, C1-C6- alkylamino, benzyl, aryl, aryloxy, thienyl, pyrrolyl, oxazolyl, furyl, thiazolyl, oxadiazolyl, and isoxazolyl, cyclic radicals themselves can be partially or completely halogenated or can bear one to three substituents selected from nitro, hydroxy, C1-C4-alkyl, C1-C4-haloakyl, and C3-C6- cycloalkyl; on condition that X cannot be NOCH3 and CHOCH3, when R4 is unsubstituted C1-C4-alkyl, unsubstituted C3-C6-cycloalkyl, substituted or unsubstituted phenyl, or unsubstituted thienyl; or X cannot be CHOCH3, when R3 is hydrogen and R5 is C1-C10-alkyl; as well as salts or above-indicated compounds. Compound I show fungicidal activity. EFFECT: extended choice of active fungicides. 8 cl, 16 tbl, 10 ex</description><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS</subject><subject>AGRICULTURE</subject><subject>ANIMAL HUSBANDRY</subject><subject>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</subject><subject>CHEMISTRY</subject><subject>FISHING</subject><subject>FORESTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HUNTING</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PEST REPELLANTS OR ATTRACTANTS</subject><subject>PLANT GROWTH REGULATORS</subject><subject>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</subject><subject>TRAPPING</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2001</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNyj0KwkAQQOFtLES9wxxAi40__TA7yQ7oRDdjwCoEWSvRQLw_EvAAVg8e39xdzpH1dkRiEwIkCRA4SYsmLTdrsMiSQNQ4nTgI2jRRA2DFag1QrYaiotVEE9fl0s0e_XPMq18XDko2ips8vLs8Dv09v_KnS9fCH_Y776nY_kG-PqEu8A</recordid><startdate>20010420</startdate><enddate>20010420</enddate><creator>VASSILIOS GRAMMENOS</creator><creator>RAJNKHARD KIRSTGEN</creator><creator>AL'BREKHT KHARREUS</creator><creator>GERBERT BAJER</creator><creator>GIZELA LORENTS</creator><creator>EHBERKHARD AMMERMANN</creator><creator>KHUBERT ZAUTER</creator><creator>FRANTS REL</creator><creator>RUT MJULLER</creator><scope>EVB</scope></search><sort><creationdate>20010420</creationdate><title>PHENYLACETIC ACID DERIVATIVES, THEIR INTERMEDIATES, AND AGENTS CONTAINING THEREOF</title><author>VASSILIOS GRAMMENOS ; RAJNKHARD KIRSTGEN ; AL'BREKHT KHARREUS ; GERBERT BAJER ; GIZELA LORENTS ; EHBERKHARD AMMERMANN ; KHUBERT ZAUTER ; FRANTS REL ; RUT MJULLER</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_RU2165411C23</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; rus</language><creationdate>2001</creationdate><topic>ACYCLIC OR CARBOCYCLIC COMPOUNDS</topic><topic>AGRICULTURE</topic><topic>ANIMAL HUSBANDRY</topic><topic>BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES</topic><topic>CHEMISTRY</topic><topic>FISHING</topic><topic>FORESTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HUNTING</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PEST REPELLANTS OR ATTRACTANTS</topic><topic>PLANT GROWTH REGULATORS</topic><topic>PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF</topic><topic>TRAPPING</topic><toplevel>online_resources</toplevel><creatorcontrib>VASSILIOS GRAMMENOS</creatorcontrib><creatorcontrib>RAJNKHARD KIRSTGEN</creatorcontrib><creatorcontrib>AL'BREKHT KHARREUS</creatorcontrib><creatorcontrib>GERBERT BAJER</creatorcontrib><creatorcontrib>GIZELA LORENTS</creatorcontrib><creatorcontrib>EHBERKHARD AMMERMANN</creatorcontrib><creatorcontrib>KHUBERT ZAUTER</creatorcontrib><creatorcontrib>FRANTS REL</creatorcontrib><creatorcontrib>RUT MJULLER</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>VASSILIOS GRAMMENOS</au><au>RAJNKHARD KIRSTGEN</au><au>AL'BREKHT KHARREUS</au><au>GERBERT BAJER</au><au>GIZELA LORENTS</au><au>EHBERKHARD AMMERMANN</au><au>KHUBERT ZAUTER</au><au>FRANTS REL</au><au>RUT MJULLER</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>PHENYLACETIC ACID DERIVATIVES, THEIR INTERMEDIATES, AND AGENTS CONTAINING THEREOF</title><date>2001-04-20</date><risdate>2001</risdate><abstract>organic synthesis. SUBSTANCE: invention provides novel phenylacetic acid derivatives of general formula I: (I), in which X denotes NOCH3, CHOCH3 and CHCH2CH3; R1 hydrogen or C1-C4-alkyl; R2 halogen, C1-C4-alkyl, or C1- C4-alkoxy; m= 0 or 1; R3 denotes hydrogen, amino, halogen, C1-C4-alkyl, C1- C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-alkylamino, or di- C1- C4-alkylamino; R4 cyano, halogen, C1-C6-alkyl, C1-C6-alkoxy, C2-C6- alkenyl, C2-C6-alkenyloxy, or C2-C6-alkinyl; provided that hydrocarbon moieties of above-indicated groups can be partially or completely halogenated or can bear one to three substituents selected from cyano, C1- C6-alkoxy, C1-C6-alkoxycarbonyl, phenyl, and dioxan (cyclic radicals can be partially or completely halogenated), C3-C6-cycloalkyl, C3-C6-cycloalkenyl, aryl, isoxazolyl, pyridyl, dioxolanyl, benzoxazolyl, thienyl, oxazolyl, furyl, oxyranyl, pyrazolyl, thiazolyl, pyrimidyloxy or tetrahydropyranyl, provided that cyclic radicals can be partially or completely halogenated or can bear one to three substituents selected from nitro, C1-C6-alkyl, C1-C6- alkoxy, C1-C6-haloalkyl, C1-C6-alkylamino, di-C1-C6-alkylamino and aryl; R5 denotes hydrogen, C1-C10-alkyl, C2-C10-alkenyl, or C2-C10-alkinyl, provided that these radicals can be partially or completely halogenated or can bear one to three substituents selected from cyano, hydroxy, aminocarbonyl, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkoxycarbonyl, C1-C6- alkylamino, benzyl, aryl, aryloxy, thienyl, pyrrolyl, oxazolyl, furyl, thiazolyl, oxadiazolyl, and isoxazolyl, cyclic radicals themselves can be partially or completely halogenated or can bear one to three substituents selected from nitro, hydroxy, C1-C4-alkyl, C1-C4-haloakyl, and C3-C6- cycloalkyl; on condition that X cannot be NOCH3 and CHOCH3, when R4 is unsubstituted C1-C4-alkyl, unsubstituted C3-C6-cycloalkyl, substituted or unsubstituted phenyl, or unsubstituted thienyl; or X cannot be CHOCH3, when R3 is hydrogen and R5 is C1-C10-alkyl; as well as salts or above-indicated compounds. Compound I show fungicidal activity. EFFECT: extended choice of active fungicides. 8 cl, 16 tbl, 10 ex</abstract><edition>7</edition><oa>free_for_read</oa></addata></record> |
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subjects | ACYCLIC OR CARBOCYCLIC COMPOUNDS AGRICULTURE ANIMAL HUSBANDRY BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES CHEMISTRY FISHING FORESTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HUNTING METALLURGY ORGANIC CHEMISTRY PEST REPELLANTS OR ATTRACTANTS PLANT GROWTH REGULATORS PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF TRAPPING |
title | PHENYLACETIC ACID DERIVATIVES, THEIR INTERMEDIATES, AND AGENTS CONTAINING THEREOF |
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