PYRAZOLYL DERIVATIVES USEFUL AS ANTI-CANCER AGENTS

The present invention provides a compound of formula (I) or a stereoisomer thereof, or an atropisomer thereof, or a pharmaceutically acceptable salt thereof, or a pharmaceutically acceptable salt of a stereoisomer thereof, or a pharmaceutically acceptable salt of an atropisomer thereof;a method for...

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Hauptverfasser: MAH, ROBERT, RIGOLLIER, PASCAL, WILCKEN, RAINER, LEBLANC, CATHERINE, VAUPEL, ANDREA, COTESTA, SIMONA, MURA, CHRISTOPHE, GERSPACHER, MARC, WARIN, NICOLAS, MACHAUER, RAINER, SCHNEIDER, NADINE, STUTZ, STEFAN, LORTHIOIS, EDWIGE, LILIANE, JEANNE, LIU, BO
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creator MAH, ROBERT
RIGOLLIER, PASCAL
WILCKEN, RAINER
LEBLANC, CATHERINE
VAUPEL, ANDREA
COTESTA, SIMONA
MURA, CHRISTOPHE
GERSPACHER, MARC
WARIN, NICOLAS
MACHAUER, RAINER
SCHNEIDER, NADINE
STUTZ, STEFAN
LORTHIOIS, EDWIGE, LILIANE, JEANNE
LIU, BO
description The present invention provides a compound of formula (I) or a stereoisomer thereof, or an atropisomer thereof, or a pharmaceutically acceptable salt thereof, or a pharmaceutically acceptable salt of a stereoisomer thereof, or a pharmaceutically acceptable salt of an atropisomer thereof;a method for manufacturing said compound, and its therapeutic uses. The present invention further provides a combination of pharmacologically active agents and a pharmaceutical composition comprising said compound.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title PYRAZOLYL DERIVATIVES USEFUL AS ANTI-CANCER AGENTS
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