DERIVADOS DO ISOXAZOL E DE CROTONAMIDA E SUA UTILIZACAO COMO PRODUTOS FARMACEUTICOS E MEIOS DE DIAGNOSTICO

Anilide derivatives of formula (I) and their salts and pure stereoisomer forms are new. R1 = a group of formula (a) or (b); R2 = O(CH2)nCH=CH2, O(CH2)mCH2Y, NH2 or NHCOCHR3R4; R3 = halogen or NH2; R4 = H or the residue of an amino acid; Y = F, Cl, Br or I; m, n = 1 - 3. Also claimed are compounds of...

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Hauptverfasser: WILFRIED SCHWAB, BERND KIRSCHBAUM, STEFAN MULLNER
Format: Patent
Sprache:por
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Zusammenfassung:Anilide derivatives of formula (I) and their salts and pure stereoisomer forms are new. R1 = a group of formula (a) or (b); R2 = O(CH2)nCH=CH2, O(CH2)mCH2Y, NH2 or NHCOCHR3R4; R3 = halogen or NH2; R4 = H or the residue of an amino acid; Y = F, Cl, Br or I; m, n = 1 - 3. Also claimed are compounds of formula (IV). Q = O, NH, O(CH2)nCH2, NHCOCH(R') or O(CH2)nCH2, NHCOCH(R')NH; R' = as R4 or L; X = polymer or solid; L = a bridging group Q bonded via a spacer of formula NH(CH2)pS; p = 1-12.