NAPHT-2-YLACETIC ACID DERIVATIVES TO TREAT AIDS
The invention provides compounds of formula (I): or a salt thereof as described herein. The invention also provides pharmaceutical compositions comprising a compound of formula I, processes for preparing compounds of formula (I), intermediates useful for preparing compounds of formula I and therapeu...
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creator | LIANHONG XU JAMES TAYLOR MICHAEL L. MITCHELL HONGYAN GUO PAUL A. ROETHLE JAMES D. TRENKLE RANDALL W. VIVIAN RANDALL L. HALCOMB KERIM BABAOGLU JOHN O. LINK RYAN MCFADDEN KYLA BJORNSON HONGTAO LIU PAUL HRVATIN ELIZABETH BACON |
description | The invention provides compounds of formula (I): or a salt thereof as described herein. The invention also provides pharmaceutical compositions comprising a compound of formula I, processes for preparing compounds of formula (I), intermediates useful for preparing compounds of formula I and therapeutic methods for treating the proliferation of the HIV virus, treating AIDS or delaying the onset of AIDS or ARC symptoms in a mammal using compounds of formula (I). |
format | Patent |
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LINK ; RYAN MCFADDEN ; KYLA BJORNSON ; HONGTAO LIU ; PAUL HRVATIN ; ELIZABETH BACON</creator><creatorcontrib>LIANHONG XU ; JAMES TAYLOR ; MICHAEL L. MITCHELL ; HONGYAN GUO ; PAUL A. ROETHLE ; JAMES D. TRENKLE ; RANDALL W. VIVIAN ; RANDALL L. HALCOMB ; KERIM BABAOGLU ; JOHN O. LINK ; RYAN MCFADDEN ; KYLA BJORNSON ; HONGTAO LIU ; PAUL HRVATIN ; ELIZABETH BACON</creatorcontrib><description>The invention provides compounds of formula (I): or a salt thereof as described herein. The invention also provides pharmaceutical compositions comprising a compound of formula I, processes for preparing compounds of formula (I), intermediates useful for preparing compounds of formula I and therapeutic methods for treating the proliferation of the HIV virus, treating AIDS or delaying the onset of AIDS or ARC symptoms in a mammal using compounds of formula (I).</description><language>eng ; por</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2017</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20170803&DB=EPODOC&CC=PT&NR=2588450T$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76290</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20170803&DB=EPODOC&CC=PT&NR=2588450T$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>LIANHONG XU</creatorcontrib><creatorcontrib>JAMES TAYLOR</creatorcontrib><creatorcontrib>MICHAEL L. MITCHELL</creatorcontrib><creatorcontrib>HONGYAN GUO</creatorcontrib><creatorcontrib>PAUL A. ROETHLE</creatorcontrib><creatorcontrib>JAMES D. TRENKLE</creatorcontrib><creatorcontrib>RANDALL W. VIVIAN</creatorcontrib><creatorcontrib>RANDALL L. HALCOMB</creatorcontrib><creatorcontrib>KERIM BABAOGLU</creatorcontrib><creatorcontrib>JOHN O. LINK</creatorcontrib><creatorcontrib>RYAN MCFADDEN</creatorcontrib><creatorcontrib>KYLA BJORNSON</creatorcontrib><creatorcontrib>HONGTAO LIU</creatorcontrib><creatorcontrib>PAUL HRVATIN</creatorcontrib><creatorcontrib>ELIZABETH BACON</creatorcontrib><title>NAPHT-2-YLACETIC ACID DERIVATIVES TO TREAT AIDS</title><description>The invention provides compounds of formula (I): or a salt thereof as described herein. The invention also provides pharmaceutical compositions comprising a compound of formula I, processes for preparing compounds of formula (I), intermediates useful for preparing compounds of formula I and therapeutic methods for treating the proliferation of the HIV virus, treating AIDS or delaying the onset of AIDS or ARC symptoms in a mammal using compounds of formula (I).</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2017</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZND3cwzwCNE10o30cXR2DfF0VnB09nRRcHEN8gxzDPEMcw1WCPFXCAlydQxRcPR0CeZhYE1LzClO5YXS3AwKbq4hzh66qQX58anFBYnJqXmpJfEBIUamFhYmpgYhIcZEKAEApQcl2A</recordid><startdate>20170803</startdate><enddate>20170803</enddate><creator>LIANHONG XU</creator><creator>JAMES TAYLOR</creator><creator>MICHAEL L. 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VIVIAN</creatorcontrib><creatorcontrib>RANDALL L. HALCOMB</creatorcontrib><creatorcontrib>KERIM BABAOGLU</creatorcontrib><creatorcontrib>JOHN O. LINK</creatorcontrib><creatorcontrib>RYAN MCFADDEN</creatorcontrib><creatorcontrib>KYLA BJORNSON</creatorcontrib><creatorcontrib>HONGTAO LIU</creatorcontrib><creatorcontrib>PAUL HRVATIN</creatorcontrib><creatorcontrib>ELIZABETH BACON</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>LIANHONG XU</au><au>JAMES TAYLOR</au><au>MICHAEL L. MITCHELL</au><au>HONGYAN GUO</au><au>PAUL A. ROETHLE</au><au>JAMES D. TRENKLE</au><au>RANDALL W. VIVIAN</au><au>RANDALL L. HALCOMB</au><au>KERIM BABAOGLU</au><au>JOHN O. LINK</au><au>RYAN MCFADDEN</au><au>KYLA BJORNSON</au><au>HONGTAO LIU</au><au>PAUL HRVATIN</au><au>ELIZABETH BACON</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>NAPHT-2-YLACETIC ACID DERIVATIVES TO TREAT AIDS</title><date>2017-08-03</date><risdate>2017</risdate><abstract>The invention provides compounds of formula (I): or a salt thereof as described herein. The invention also provides pharmaceutical compositions comprising a compound of formula I, processes for preparing compounds of formula (I), intermediates useful for preparing compounds of formula I and therapeutic methods for treating the proliferation of the HIV virus, treating AIDS or delaying the onset of AIDS or ARC symptoms in a mammal using compounds of formula (I).</abstract><oa>free_for_read</oa></addata></record> |
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subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
title | NAPHT-2-YLACETIC ACID DERIVATIVES TO TREAT AIDS |
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