SELECTIVE HYDROGENATION PRODUCTA OF C-076 COMPOUNDS AND DERIVATIVES THEREOF

The invention provide compounds having the formula: in which R1 is iso-propyl or sec-butyl; R2 is methoxy, hydroxy or loweralkanoyloxy; and R3 is hydrogen; lower alkanoyl; alpha -L-oleandrosyl; 4 min -(lower alkanoyl)- alpha -L- oleandrosyl; 4 min -( alpha -L- oleandrosyl)- alpha -L-oleandrosyl or 4...

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Hauptverfasser: CHABALA JOHN CLIFFORD, FISHER MICHAEL HERBERT
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creator CHABALA JOHN CLIFFORD
FISHER MICHAEL HERBERT
description The invention provide compounds having the formula: in which R1 is iso-propyl or sec-butyl; R2 is methoxy, hydroxy or loweralkanoyloxy; and R3 is hydrogen; lower alkanoyl; alpha -L-oleandrosyl; 4 min -(lower alkanoyl)- alpha -L- oleandrosyl; 4 min -( alpha -L- oleandrosyl)- alpha -L-oleandrosyl or 4Rx-(lower alkanoyl)-4 min -( alpha -L- oleandrosyl)- alpha -L- oleandrosyl. These compounds are derivatives of C-076 and are produced by catalytic reduction of the 22,23-position of the C-076 molecule. Further reaction of the reduced C-076 compounds is also possible. The compounds thus produced are used for their profound anthelmintic, insecticidal, ectoparasiticidal and acaracidal activity. Compositions containing the described C-076 derivatives as active ingredient are also disclosed.
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These compounds are derivatives of C-076 and are produced by catalytic reduction of the 22,23-position of the C-076 molecule. Further reaction of the reduced C-076 compounds is also possible. The compounds thus produced are used for their profound anthelmintic, insecticidal, ectoparasiticidal and acaracidal activity. 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These compounds are derivatives of C-076 and are produced by catalytic reduction of the 22,23-position of the C-076 molecule. Further reaction of the reduced C-076 compounds is also possible. The compounds thus produced are used for their profound anthelmintic, insecticidal, ectoparasiticidal and acaracidal activity. Compositions containing the described C-076 derivatives as active ingredient are also disclosed.</abstract><oa>free_for_read</oa></addata></record>
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subjects AGRICULTURE
ANIMAL HUSBANDRY
APPARATUS THEREFOR
BEER
BIOCHEMISTRY
BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES
CHEMISTRY
DERIVATIVES THEREOF
ENZYMOLOGY
FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIREDCHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERSFROM A RACEMIC MIXTURE
FISHING
FORESTRY
GENERAL METHODS OF ORGANIC CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HUNTING
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
MICROBIOLOGY
MUTATION OR GENETIC ENGINEERING
NUCLEIC ACIDS
NUCLEOSIDES
NUCLEOTIDES
ORGANIC CHEMISTRY
PEST REPELLANTS OR ATTRACTANTS
PLANT GROWTH REGULATORS
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
SPIRITS
SUGARS
TRAPPING
VINEGAR
WINE
title SELECTIVE HYDROGENATION PRODUCTA OF C-076 COMPOUNDS AND DERIVATIVES THEREOF
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