DERIVADOS DE PIPERIDINA/PIPERAZINA
REFERIDO A DERIVADOS DE PIPERIDINA/PIPERAZINA DE FORMULA (I): DONDE A ES CH, N; --- ES UN ENLACE OPCIONAL EN EL CASO QUE A SEA C; X ES -O-C(=O)-, -C(=O)-C(=O)-, -NRx-C(=O)-, ENTRE OTROS; Rx ES H, ALQUILO C1-C4; Y ES -C(=O)-NRx-, -NRx-C(=O)-; R1 ES ADAMANTANILO, CICLOALQUILO C3-C6, FENILO, NAFTALENO,...
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| creator | VAN LOMMEN GUY ROSALIA EUGEEN BRAEKEN MIRIELLE ROEVENS PETER WALTER MARIA BONGARTZ JEAN-PIERRE ANDRE MARC COESEMANS ERWIN DE WAEPENAERT KATHARINA ANTONIA GERMANIA J.M DAVIDENKO PETR VLADIMIRIVICH BUYCK CHRISTOPHE FRANCIS ROBERT NESTOR MEERPOEL LIEVEN LINDERS JOANNES THEODORUS MARIA BERWAER MONIQUE JENNY MARIE |
| description | REFERIDO A DERIVADOS DE PIPERIDINA/PIPERAZINA DE FORMULA (I): DONDE A ES CH, N; --- ES UN ENLACE OPCIONAL EN EL CASO QUE A SEA C; X ES -O-C(=O)-, -C(=O)-C(=O)-, -NRx-C(=O)-, ENTRE OTROS; Rx ES H, ALQUILO C1-C4; Y ES -C(=O)-NRx-, -NRx-C(=O)-; R1 ES ADAMANTANILO, CICLOALQUILO C3-C6, FENILO, NAFTALENO, ENTRE OTROS; R2 ES CICLOALQUILO C3-C6, FENILO, NAFTALENILO, ENTRE OTROS; R7 ES H, HALO, ALQUILO C1-C4, ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA Y A UN PROCESO DE PREPARACION. DICHO COMPUESTO TIENE ACTIVIDAD INHIBITORIA DE DGAT Y ES UTIL EN EL TRATAMIENTO DE ENFERMEDADES MEDIADAS POR DGAT1 COMO OBESIDAD, SINDROME DE RESISITENCIA A LA INSULINA
The invention relates to a DGAT inhibitor of formula (I), including any stereochemically isomeric form thereof, a N-oxide thereof, a pharmaceutically acceptable salt thereof or a solvate thereof, and methods for preparing such compounds, pharmaceutical compositions comprising said compounds as well as the use as a medicine, as a DGAT inhibitor, of said compounds. |
| format | Patent |
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The invention relates to a DGAT inhibitor of formula (I), including any stereochemically isomeric form thereof, a N-oxide thereof, a pharmaceutically acceptable salt thereof or a solvate thereof, and methods for preparing such compounds, pharmaceutical compositions comprising said compounds as well as the use as a medicine, as a DGAT inhibitor, of said compounds.</description><language>spa</language><subject>HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2009</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20090627&DB=EPODOC&CC=PE&NR=20090820A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20090627&DB=EPODOC&CC=PE&NR=20090820A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>VAN LOMMEN GUY ROSALIA EUGEEN</creatorcontrib><creatorcontrib>BRAEKEN MIRIELLE</creatorcontrib><creatorcontrib>ROEVENS PETER WALTER MARIA</creatorcontrib><creatorcontrib>BONGARTZ JEAN-PIERRE ANDRE MARC</creatorcontrib><creatorcontrib>COESEMANS ERWIN</creatorcontrib><creatorcontrib>DE WAEPENAERT KATHARINA ANTONIA GERMANIA J.M</creatorcontrib><creatorcontrib>DAVIDENKO PETR VLADIMIRIVICH</creatorcontrib><creatorcontrib>BUYCK CHRISTOPHE FRANCIS ROBERT NESTOR</creatorcontrib><creatorcontrib>MEERPOEL LIEVEN</creatorcontrib><creatorcontrib>LINDERS JOANNES THEODORUS MARIA</creatorcontrib><creatorcontrib>BERWAER MONIQUE JENNY MARIE</creatorcontrib><title>DERIVADOS DE PIPERIDINA/PIPERAZINA</title><description>REFERIDO A DERIVADOS DE PIPERIDINA/PIPERAZINA DE FORMULA (I): DONDE A ES CH, N; --- ES UN ENLACE OPCIONAL EN EL CASO QUE A SEA C; X ES -O-C(=O)-, -C(=O)-C(=O)-, -NRx-C(=O)-, ENTRE OTROS; Rx ES H, ALQUILO C1-C4; Y ES -C(=O)-NRx-, -NRx-C(=O)-; R1 ES ADAMANTANILO, CICLOALQUILO C3-C6, FENILO, NAFTALENO, ENTRE OTROS; R2 ES CICLOALQUILO C3-C6, FENILO, NAFTALENILO, ENTRE OTROS; R7 ES H, HALO, ALQUILO C1-C4, ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA Y A UN PROCESO DE PREPARACION. DICHO COMPUESTO TIENE ACTIVIDAD INHIBITORIA DE DGAT Y ES UTIL EN EL TRATAMIENTO DE ENFERMEDADES MEDIADAS POR DGAT1 COMO OBESIDAD, SINDROME DE RESISITENCIA A LA INSULINA
The invention relates to a DGAT inhibitor of formula (I), including any stereochemically isomeric form thereof, a N-oxide thereof, a pharmaceutically acceptable salt thereof or a solvate thereof, and methods for preparing such compounds, pharmaceutical compositions comprising said compounds as well as the use as a medicine, as a DGAT inhibitor, of said compounds.</description><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2009</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZFBycQ3yDHN08Q9WcHFVCPAMAHJdPP0c9cFMxyggk4eBNS0xpziVF0pzMyi6uYY4e-imFuTHpxYXJCan5qWWxAe4GhkYWBpYGBk4GhoTowYAOkcibg</recordid><startdate>20090627</startdate><enddate>20090627</enddate><creator>VAN LOMMEN GUY ROSALIA EUGEEN</creator><creator>BRAEKEN MIRIELLE</creator><creator>ROEVENS PETER WALTER MARIA</creator><creator>BONGARTZ JEAN-PIERRE ANDRE MARC</creator><creator>COESEMANS ERWIN</creator><creator>DE WAEPENAERT KATHARINA ANTONIA GERMANIA J.M</creator><creator>DAVIDENKO PETR VLADIMIRIVICH</creator><creator>BUYCK CHRISTOPHE FRANCIS ROBERT NESTOR</creator><creator>MEERPOEL LIEVEN</creator><creator>LINDERS JOANNES THEODORUS MARIA</creator><creator>BERWAER MONIQUE JENNY MARIE</creator><scope>EVB</scope></search><sort><creationdate>20090627</creationdate><title>DERIVADOS DE PIPERIDINA/PIPERAZINA</title><author>VAN LOMMEN GUY ROSALIA EUGEEN ; BRAEKEN MIRIELLE ; ROEVENS PETER WALTER MARIA ; BONGARTZ JEAN-PIERRE ANDRE MARC ; COESEMANS ERWIN ; DE WAEPENAERT KATHARINA ANTONIA GERMANIA J.M ; DAVIDENKO PETR VLADIMIRIVICH ; BUYCK CHRISTOPHE FRANCIS ROBERT NESTOR ; MEERPOEL LIEVEN ; LINDERS JOANNES THEODORUS MARIA ; BERWAER MONIQUE JENNY MARIE</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_PE20090820A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>spa</language><creationdate>2009</creationdate><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>VAN LOMMEN GUY ROSALIA EUGEEN</creatorcontrib><creatorcontrib>BRAEKEN MIRIELLE</creatorcontrib><creatorcontrib>ROEVENS PETER WALTER MARIA</creatorcontrib><creatorcontrib>BONGARTZ JEAN-PIERRE ANDRE MARC</creatorcontrib><creatorcontrib>COESEMANS ERWIN</creatorcontrib><creatorcontrib>DE WAEPENAERT KATHARINA ANTONIA GERMANIA J.M</creatorcontrib><creatorcontrib>DAVIDENKO PETR VLADIMIRIVICH</creatorcontrib><creatorcontrib>BUYCK CHRISTOPHE FRANCIS ROBERT NESTOR</creatorcontrib><creatorcontrib>MEERPOEL LIEVEN</creatorcontrib><creatorcontrib>LINDERS JOANNES THEODORUS MARIA</creatorcontrib><creatorcontrib>BERWAER MONIQUE JENNY MARIE</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>VAN LOMMEN GUY ROSALIA EUGEEN</au><au>BRAEKEN MIRIELLE</au><au>ROEVENS PETER WALTER MARIA</au><au>BONGARTZ JEAN-PIERRE ANDRE MARC</au><au>COESEMANS ERWIN</au><au>DE WAEPENAERT KATHARINA ANTONIA GERMANIA J.M</au><au>DAVIDENKO PETR VLADIMIRIVICH</au><au>BUYCK CHRISTOPHE FRANCIS ROBERT NESTOR</au><au>MEERPOEL LIEVEN</au><au>LINDERS JOANNES THEODORUS MARIA</au><au>BERWAER MONIQUE JENNY MARIE</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>DERIVADOS DE PIPERIDINA/PIPERAZINA</title><date>2009-06-27</date><risdate>2009</risdate><abstract>REFERIDO A DERIVADOS DE PIPERIDINA/PIPERAZINA DE FORMULA (I): DONDE A ES CH, N; --- ES UN ENLACE OPCIONAL EN EL CASO QUE A SEA C; X ES -O-C(=O)-, -C(=O)-C(=O)-, -NRx-C(=O)-, ENTRE OTROS; Rx ES H, ALQUILO C1-C4; Y ES -C(=O)-NRx-, -NRx-C(=O)-; R1 ES ADAMANTANILO, CICLOALQUILO C3-C6, FENILO, NAFTALENO, ENTRE OTROS; R2 ES CICLOALQUILO C3-C6, FENILO, NAFTALENILO, ENTRE OTROS; R7 ES H, HALO, ALQUILO C1-C4, ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA Y A UN PROCESO DE PREPARACION. DICHO COMPUESTO TIENE ACTIVIDAD INHIBITORIA DE DGAT Y ES UTIL EN EL TRATAMIENTO DE ENFERMEDADES MEDIADAS POR DGAT1 COMO OBESIDAD, SINDROME DE RESISITENCIA A LA INSULINA
The invention relates to a DGAT inhibitor of formula (I), including any stereochemically isomeric form thereof, a N-oxide thereof, a pharmaceutically acceptable salt thereof or a solvate thereof, and methods for preparing such compounds, pharmaceutical compositions comprising said compounds as well as the use as a medicine, as a DGAT inhibitor, of said compounds.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | DERIVADOS DE PIPERIDINA/PIPERAZINA |
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