DERIVATIVES OF 2-PYRIDIN-2-YL-PYRAZOL-3(2H)-ONE, PREPARATION AND THERAPEUTIC USE THEREOF

DERIVATIVES OF 2-PYRIDIN-2-YL-PYRAZOL-3(2H)-ONE, PREPARATION AND THERAPEUTIC USE THEREOF

593797 Disclosed are substituted dihydropyrazolone derivatives of formula (I), wherein the substituents are as described within the specification. An examples of compounds of formula (I) is 2-[5-(piperidin-1-ylsulfonyl)pyridine-2-yl]-1,2,4,5,6,7-hexahydro-3H-indazol-3-one. Further disclosed is a pro...

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Hauptverfasser: FOSSEY, VALERIE, ILLIANO, STEPHANE, MANETTE, GERALDINE, ALTENBURGER, JEAN-MICHEL
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Sprache:eng
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CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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creator FOSSEY, VALERIE
ILLIANO, STEPHANE
MANETTE, GERALDINE
ALTENBURGER, JEAN-MICHEL
description 593797 Disclosed are substituted dihydropyrazolone derivatives of formula (I), wherein the substituents are as described within the specification. An examples of compounds of formula (I) is 2-[5-(piperidin-1-ylsulfonyl)pyridine-2-yl]-1,2,4,5,6,7-hexahydro-3H-indazol-3-one. Further disclosed is a process for preparing a compound of formula (I), a pharmaceutical composition comprising formula (I), and the use of a compound of formula (I) in the manufacture of a medicament for the treatment/prophylaxis of cardiovascular diseases, glaucoma, neurodegenerative diseases, etc.
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An examples of compounds of formula (I) is 2-[5-(piperidin-1-ylsulfonyl)pyridine-2-yl]-1,2,4,5,6,7-hexahydro-3H-indazol-3-one. 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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title DERIVATIVES OF 2-PYRIDIN-2-YL-PYRAZOL-3(2H)-ONE, PREPARATION AND THERAPEUTIC USE THEREOF
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