PIPERAZINYL PYRIDINES AND PIPERINYL-IMIDAZOLES AND PHARMACEUTICAL COMPOSITIONS; INTERMEDIATES
A compound of the formula: or a pharmaceutically acceptable salt thereof, wherein is selected from (a) a 3- or 4-pyridinyl group optionally substituted by one or two substituents each independently selected from C1-C4 alkyl and amino, (b) a 2-pyridinyl group substituted by an amino group, (c) a 2-i...
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| creator | DICKINSON, R.P CROSS, P.E |
| description | A compound of the formula:
or a pharmaceutically acceptable salt thereof, wherein is selected from (a) a 3- or 4-pyridinyl group optionally substituted by one or two substituents each independently selected from C1-C4 alkyl and amino, (b) a 2-pyridinyl group substituted by an amino group, (c) a 2-imidazolyl group optionally substituted by one or two C1-C4 alkyl groups and (d) a 2-, 3- or 4-pyridinyl group substituted by a nitro group, or an N-oxide thereof, or a 2-, 3- or 4-pyridinyl group substituted by a group of the formula -NHCOO(C1-C4 alkyl);
R is selected from (a) -NHSO2R where R is C1-C4 alkyl, C3-C7 cycloalkyl or -NR R where R and R are each independently M or C1-C4 alkyl, (b) -SO2NR R where R and R are as defined above, (c) nitro, (d) amino and (e) acetamido;
and X is a group of the formula -(CH2)m- where m is an integer of from 1 to 4, -CO(CH2)n- or -CH(OH)(CH2)n- where n is 1, 2 or 3. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_NZ219193A</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>NZ219193A</sourcerecordid><originalsourceid>FETCH-epo_espacenet_NZ219193A3</originalsourceid><addsrcrecordid>eNqFirEKwjAUALM4iPoLkh_oUDsVp0fypA-Sl5DEoYFSisRJtFD_H1F0djq4u7UYPHkMkIl7I30fSBNjlMBafsrbV2RJQ3bmFzoIFhSeEykwUjnrXaREjuNREicMFjVBwrgVq-t0W8ruy43YnzCprirzYyzLPF3KvTxHzoe6rdsGmr_DCzJgMl8</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>PIPERAZINYL PYRIDINES AND PIPERINYL-IMIDAZOLES AND PHARMACEUTICAL COMPOSITIONS; INTERMEDIATES</title><source>esp@cenet</source><creator>DICKINSON, R.P ; CROSS, P.E</creator><creatorcontrib>DICKINSON, R.P ; CROSS, P.E</creatorcontrib><description>A compound of the formula:
or a pharmaceutically acceptable salt thereof, wherein <> is selected from (a) a 3- or 4-pyridinyl group optionally substituted by one or two substituents each independently selected from C1-C4 alkyl and amino, (b) a 2-pyridinyl group substituted by an amino group, (c) a 2-imidazolyl group optionally substituted by one or two C1-C4 alkyl groups and (d) a 2-, 3- or 4-pyridinyl group substituted by a nitro group, or an N-oxide thereof, or a 2-, 3- or 4-pyridinyl group substituted by a group of the formula -NHCOO(C1-C4 alkyl);
R is selected from (a) -NHSO2R where R is C1-C4 alkyl, C3-C7 cycloalkyl or -NR R where R and R are each independently M or C1-C4 alkyl, (b) -SO2NR R where R and R are as defined above, (c) nitro, (d) amino and (e) acetamido;
and X is a group of the formula -(CH2)m- where m is an integer of from 1 to 4, -CO(CH2)n- or -CH(OH)(CH2)n- where n is 1, 2 or 3.</description><edition>4</edition><language>eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>1989</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19890106&DB=EPODOC&CC=NZ&NR=219193A$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19890106&DB=EPODOC&CC=NZ&NR=219193A$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>DICKINSON, R.P</creatorcontrib><creatorcontrib>CROSS, P.E</creatorcontrib><title>PIPERAZINYL PYRIDINES AND PIPERINYL-IMIDAZOLES AND PHARMACEUTICAL COMPOSITIONS; INTERMEDIATES</title><description>A compound of the formula:
or a pharmaceutically acceptable salt thereof, wherein <> is selected from (a) a 3- or 4-pyridinyl group optionally substituted by one or two substituents each independently selected from C1-C4 alkyl and amino, (b) a 2-pyridinyl group substituted by an amino group, (c) a 2-imidazolyl group optionally substituted by one or two C1-C4 alkyl groups and (d) a 2-, 3- or 4-pyridinyl group substituted by a nitro group, or an N-oxide thereof, or a 2-, 3- or 4-pyridinyl group substituted by a group of the formula -NHCOO(C1-C4 alkyl);
R is selected from (a) -NHSO2R where R is C1-C4 alkyl, C3-C7 cycloalkyl or -NR R where R and R are each independently M or C1-C4 alkyl, (b) -SO2NR R where R and R are as defined above, (c) nitro, (d) amino and (e) acetamido;
and X is a group of the formula -(CH2)m- where m is an integer of from 1 to 4, -CO(CH2)n- or -CH(OH)(CH2)n- where n is 1, 2 or 3.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>1989</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqFirEKwjAUALM4iPoLkh_oUDsVp0fypA-Sl5DEoYFSisRJtFD_H1F0djq4u7UYPHkMkIl7I30fSBNjlMBafsrbV2RJQ3bmFzoIFhSeEykwUjnrXaREjuNREicMFjVBwrgVq-t0W8ruy43YnzCprirzYyzLPF3KvTxHzoe6rdsGmr_DCzJgMl8</recordid><startdate>19890106</startdate><enddate>19890106</enddate><creator>DICKINSON, R.P</creator><creator>CROSS, P.E</creator><scope>EVB</scope></search><sort><creationdate>19890106</creationdate><title>PIPERAZINYL PYRIDINES AND PIPERINYL-IMIDAZOLES AND PHARMACEUTICAL COMPOSITIONS; INTERMEDIATES</title><author>DICKINSON, R.P ; CROSS, P.E</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_NZ219193A3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>1989</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>DICKINSON, R.P</creatorcontrib><creatorcontrib>CROSS, P.E</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>DICKINSON, R.P</au><au>CROSS, P.E</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>PIPERAZINYL PYRIDINES AND PIPERINYL-IMIDAZOLES AND PHARMACEUTICAL COMPOSITIONS; INTERMEDIATES</title><date>1989-01-06</date><risdate>1989</risdate><abstract>A compound of the formula:
or a pharmaceutically acceptable salt thereof, wherein <> is selected from (a) a 3- or 4-pyridinyl group optionally substituted by one or two substituents each independently selected from C1-C4 alkyl and amino, (b) a 2-pyridinyl group substituted by an amino group, (c) a 2-imidazolyl group optionally substituted by one or two C1-C4 alkyl groups and (d) a 2-, 3- or 4-pyridinyl group substituted by a nitro group, or an N-oxide thereof, or a 2-, 3- or 4-pyridinyl group substituted by a group of the formula -NHCOO(C1-C4 alkyl);
R is selected from (a) -NHSO2R where R is C1-C4 alkyl, C3-C7 cycloalkyl or -NR R where R and R are each independently M or C1-C4 alkyl, (b) -SO2NR R where R and R are as defined above, (c) nitro, (d) amino and (e) acetamido;
and X is a group of the formula -(CH2)m- where m is an integer of from 1 to 4, -CO(CH2)n- or -CH(OH)(CH2)n- where n is 1, 2 or 3.</abstract><edition>4</edition><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | PIPERAZINYL PYRIDINES AND PIPERINYL-IMIDAZOLES AND PHARMACEUTICAL COMPOSITIONS; INTERMEDIATES |
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