5-VINYL- AND 5-ETHYNYL-QUINOLONE- AND - NAPHTHYLIDONE-CARBOXYLIC ACIDS

Quinolone and naphthyridone derivs. of formula (I), and their hydrates, acid addn. salts, and alkali-, alkaline earth, silver and guanidinium salts, are new. R1 = 1-4C alkyl (opt. substd. by OH, halo or 1-3C alkoxy), 3-6C cycloalkyl (opt. substd. by halo or 1-3C alkyl), 2-4C alkenyl, 1-3C alkoxy, am...

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Hauptverfasser: RAINAA ENDERUMAN, UBE PEETAAZEN, TOOMASU HIMURAA, KURAUSUUDEIITAA BUREMU, HAINTSUUGEORUKU BETSUSHIYUTAIN, MIHIYAERU SHIYUTEGEMAN
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creator RAINAA ENDERUMAN
UBE PEETAAZEN
TOOMASU HIMURAA
KURAUSUUDEIITAA BUREMU
HAINTSUUGEORUKU BETSUSHIYUTAIN
MIHIYAERU SHIYUTEGEMAN
description Quinolone and naphthyridone derivs. of formula (I), and their hydrates, acid addn. salts, and alkali-, alkaline earth, silver and guanidinium salts, are new. R1 = 1-4C alkyl (opt. substd. by OH, halo or 1-3C alkoxy), 3-6C cycloalkyl (opt. substd. by halo or 1-3C alkyl), 2-4C alkenyl, 1-3C alkoxy, amino, 1-3C monoalkylamino, 2-6C dialkylamino, or phenyl (opt. substd. by 1-3 halo); R2 = H, 1-4C alkyl or (5-methyl-2-oxo-1,3-dioxol-4-yl)-methyl; X = CH, C-halo, COMe, COCHF2, CMe or N; Z = CR4=CHR3 or C IDENTICAL CR5; R3 = H, 1-3C alkyl, 1-3C alkoxy, or 1-3C alkoxy-methyl; R4 = H or halo; R5 = H, 1-6C alkyl (opt. substd. by 1-3 halo or OH), 2-3C alkenyl, 1-3C alkoxy, 1-3C alkoxy-methyl, halo or SiMe3; R6 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl, 1-4C oxoalkyl, or 1-3C acyl; Y = NR'R"; NR'R" = pyrrolyl, imidazolyl or a specified satd. or mono-unsatd. mono-or bicyclic ring, (opt. contg. O or a second N, opt. substd.)
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R1 = 1-4C alkyl (opt. substd. by OH, halo or 1-3C alkoxy), 3-6C cycloalkyl (opt. substd. by halo or 1-3C alkyl), 2-4C alkenyl, 1-3C alkoxy, amino, 1-3C monoalkylamino, 2-6C dialkylamino, or phenyl (opt. substd. by 1-3 halo); R2 = H, 1-4C alkyl or (5-methyl-2-oxo-1,3-dioxol-4-yl)-methyl; X = CH, C-halo, COMe, COCHF2, CMe or N; Z = CR4=CHR3 or C IDENTICAL CR5; R3 = H, 1-3C alkyl, 1-3C alkoxy, or 1-3C alkoxy-methyl; R4 = H or halo; R5 = H, 1-6C alkyl (opt. substd. by 1-3 halo or OH), 2-3C alkenyl, 1-3C alkoxy, 1-3C alkoxy-methyl, halo or SiMe3; R6 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl, 1-4C oxoalkyl, or 1-3C acyl; Y = NR'R"; NR'R" = pyrrolyl, imidazolyl or a specified satd. or mono-unsatd. mono-or bicyclic ring, (opt. contg. O or a second N, opt. substd.)</abstract><edition>6</edition><oa>free_for_read</oa></addata></record>
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subjects AGRICULTURE
ANIMAL HUSBANDRY
BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES
CHEMISTRY
FISHING
FODDER
FOODS OR FOODSTUFFS
FOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BYSUBCLASSES A23B - A23J
FORESTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HUNTING
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PEST REPELLANTS OR ATTRACTANTS
PLANT GROWTH REGULATORS
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF
PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OFNUTRITIVE QUALITIES, PHYSICAL TREATMENT
THEIR TREATMENT, NOT COVERED BY OTHER CLASSES
TRAPPING
title 5-VINYL- AND 5-ETHYNYL-QUINOLONE- AND - NAPHTHYLIDONE-CARBOXYLIC ACIDS
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