Method for preparing bicyclic compounds and use of said method for preparing an interleukin-1sg(betha) conversion enzyme (ice) inhibitor

Method for preparing bicyclic compounds and use of said method for preparing an interleukin-1sg(betha) conversion enzyme (ice) inhibitor

A method for preparing compounds of formula (I)wherein R is selected from the group consisting of H. alkyl, aryl, and aralkyl of up to 18 carbon atoms and the amine function may be free or protected from a compound of formula (IA) wherein cyclization is carried out in a basic medium and in the prese...

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Hauptverfasser: CROCQ VERONIQUE, ROUSSEL PATRICK
Format: Patent
Sprache:eng ; hun
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CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
PEPTIDES
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creator CROCQ VERONIQUE
ROUSSEL PATRICK
description A method for preparing compounds of formula (I)wherein R is selected from the group consisting of H. alkyl, aryl, and aralkyl of up to 18 carbon atoms and the amine function may be free or protected from a compound of formula (IA) wherein cyclization is carried out in a basic medium and in the presence of a phosphonic acid derivative and the use of said method as an intermediate step for preparing a compound inhibiting the interleukin-1 beta conversion enzyme.
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HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
PEPTIDES
title Method for preparing bicyclic compounds and use of said method for preparing an interleukin-1sg(betha) conversion enzyme (ice) inhibitor
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