N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS
Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted T-type calcium channel activity, are disclosed. Specifically, a series of compounds which are N-piperidinyl acetamide derivatives as shown in formula (1) are disclosed...
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| creator | Kaul, Ramesh Pajouhesh, Hassan Ding, Yanbing Grimwood, Mike Zhang, Lingyun Zhou, Yuanxi Zhu, Yongbao Tan, Jason Chakka, Nagasree |
| description | Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted T-type calcium channel activity, are disclosed. Specifically, a series of compounds which are N-piperidinyl acetamide derivatives as shown in formula (1) are disclosed as calcium ion channel activating modulators. Compositions comprising these compounds and the use of these compounds in the treatment or prevention of conditions such as epilepsy are also disclosed. |
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Compositions comprising these compounds and the use of these compounds in the treatment or prevention of conditions such as epilepsy are also disclosed.</description><language>hrv ; eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2020</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20201113&DB=EPODOC&CC=HR&NR=P20201243T1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,778,883,25547,76298</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20201113&DB=EPODOC&CC=HR&NR=P20201243T1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>Kaul, Ramesh</creatorcontrib><creatorcontrib>Pajouhesh, Hassan</creatorcontrib><creatorcontrib>Ding, Yanbing</creatorcontrib><creatorcontrib>Grimwood, Mike</creatorcontrib><creatorcontrib>Zhang, Lingyun</creatorcontrib><creatorcontrib>Zhou, Yuanxi</creatorcontrib><creatorcontrib>Zhu, Yongbao</creatorcontrib><creatorcontrib>Tan, Jason</creatorcontrib><creatorcontrib>Chakka, Nagasree</creatorcontrib><title>N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS</title><description>Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted T-type calcium channel activity, are disclosed. 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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS |
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