GABA RECEPTOR MODULATORS

Method, compositions, and compounds for modulating brain excitability to alleviate stress, anxiety, insomnia and seizure activity using certain steroid derivatives that act at a newly identified site on the gamma-aminobutyric acid receptor-chloride ionophore (GR) complex.

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Hauptverfasser: TAHIR, SAYED, HASAN, BOLGER, MICHAEL, BRUCE, BELELLI, DELIA, GEE, KELVIN, WELLMAN, PURDY, ROBERT, HYDE, UPASANI, RAVINDRA B, LAN, NANCY, TSAI-YUN, MIRSADEGHI, SYED
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creator TAHIR, SAYED, HASAN
BOLGER, MICHAEL, BRUCE
BELELLI, DELIA
GEE, KELVIN, WELLMAN
PURDY, ROBERT, HYDE
UPASANI, RAVINDRA B
LAN, NANCY, TSAI-YUN
MIRSADEGHI, SYED
description Method, compositions, and compounds for modulating brain excitability to alleviate stress, anxiety, insomnia and seizure activity using certain steroid derivatives that act at a newly identified site on the gamma-aminobutyric acid receptor-chloride ionophore (GR) complex.
format Patent
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source esp@cenet
subjects CHEMISTRY
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
STEROIDS
title GABA RECEPTOR MODULATORS
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